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Doxazosin
Catalog No. A17779 α-1 adrenergic receptor blockerDoxazosin is an α-1 adrenergic receptor blocker that inhibits the binding of norepinephrine, which is released from sympathetic nerve terminals, to the α-1 receptors on the membrane of vascular smooth muscle cells. Blockages of the alpha-1 adrenergic action on the vascular smooth muscles lead to a decrease in vascular resistance and antihypertensive activity. 了解更多 -
Brimonidine
Catalog No. A17899 α2-adrenergic receptor agonistBrimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 了解更多 -
Nylidrin Hydrochloride
Catalog No. A17947 beta-adrenergic agonistNylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent. 了解更多 -
Metipranolol hydrochloride
Catalog No. A18064 β-adrenergic receptor antagonistMetipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多 -
Anisodamine
Catalog No. A18215 alpha-1 adrenergic receptors / mAChRs inhibitorAnisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多 -
Tulobuterol hydrochloride
Catalog No. A18226 β2-adrenergic receptor agonistTulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多 -
Atenolol
Catalog No. A21962 -
Norepinephrine
Catalog No. A11306 β1-selective adrenergic receptor agonistNorepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
Ancarolol
Catalog No. A12534 -
AGN 192836
Catalog No. A13013 α2 adrenergic agonistAGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多 -
β3-AR agonist 1
Catalog No. A12777 β3-adrenergic receptor agonistβ3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多 -
Norepinephrine hydrochloride
Catalog No. A21605 β1-selective adrenergic receptor agonistNorepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
Mosapride citrate
Catalog No. A10607 -
Tianeptine sodium
Catalog No. A10931 -
Agomelatine
Catalog No. A10048 -
5-hydroxytryptophan (5-HTP)
Catalog No. A10017 5-hydroxytryptophan (5-HTP)是天然存在的氨基酸和化学前体，也是色氨酸在神经递质5-羟色胺和褪黑素生物合成中的代谢中间体。 了解更多 -
BRL-15572 dihydrochloride
Catalog No. A11178 5-HT1D receptor 拮抗剂BRL-15572是一种选择性的h5-HT1D拮抗剂，相对于h5-HT1B表现出60倍的选择性，对一系列其他受体类型的亲和力很小或没有亲和力。 了解更多 -
WAY-100635
Catalog No. A11182 -
BMY 7378
Catalog No. A11208 -
Naftopidil 2HCl
Catalog No. A10619 5-HT1A and α1-adrenergic receptor 拮抗剂Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂，IC50分别为0.1μM和0.2μM。 了解更多 -
Puerarin (Kakonein)
Catalog No. A10759 5-HT2C receptor 拮抗剂Puerarin (Kakonein)是几种已知的异黄酮之一。Puerarin是5-HT2C受体和苯二氮卓类拮抗剂。Puerarin正在研究作为一种自微乳化药物递送系统。 了解更多 -
Risperidone (Risperdal)
Catalog No. A10797 Risperidone (Risperdal)是一种非典型的抗精神病药，用于治疗精神分裂症（包括青少年精神分裂症），精神分裂症，躁郁症的躁狂和躁狂状态，以及自闭症儿童的烦躁不安。 了解更多 -
Tropisetron (ICS 205930)
Catalog No. A11226 -
Vilazodone
Catalog No. A11116 Serotonin reuptake 抑制剂Vilazodone充当5-羟色胺再摄取抑制剂（IC50 = 0.5 nM）和5-HT1A受体部分激动剂（IC50 = 0.2 nM； IA =?60-70％）。 了解更多 -
Prucalopride
Catalog No. A11771 5-HT Receptor 激动剂Prucalopride是一种选择性的，高亲和力的5-HT4受体激动剂，作用于5-HT4A和5-HT4B受体，Ki分别为2.5 nM和8 nM，比作用于5-HT受体亚型选择性高290倍以上。 了解更多 -
Alosetron
Catalog No. A11310 -
SB269970 HCl
Catalog No. A11925 -
Ondansetron (Zofran)
Catalog No. A11701 Ondansetron (Zofran)是一种5-羟色胺5-HT3受体拮抗剂，主要用作止吐药（用于治疗恶心和呕吐）。 了解更多 -
Mirtazapine
Catalog No. A11702 Mirtazapine是一种去甲肾上腺素能和特异性血清素能抗抑郁药（NaSSA）。在结构上，米氮平也可以归类为四环抗抑郁药（TeCA）。 了解更多 -
Urapidil hydrochloride
Catalog No. A11704 Urapidil hydrochloride是α1肾上腺素受体拮抗剂、5-HT1A血清素受体部分激动剂和抗高血压药。 了解更多 -
Duloxetine HCl
Catalog No. A11717 Duloxetine Hydrochloride是一种5-羟色胺和去甲肾上腺素再摄取抑制剂（SNRI），Ki为 4.6 nM。用于治疗压力性尿失禁和抑郁症。 了解更多 -
Tegaserod maleate
Catalog No. A11743 Tegaserod maleate作为运动刺激剂发挥作用，通过激活胃肠道中肠神经系统的5-ht4受体达到其所需的治疗效果。它还能刺激胃肠动力和蠕动反射，据称还能减轻腹痛。此外，替加色罗是5-ht2b受体拮抗剂。 了解更多 -
Asenapine maleate
Catalog No. A10091 H1 拮抗剂Asenapine maleate平对多种受体具有高亲和力（pKi），包括5-羟色胺5-HT1A（8.6），5-HT1B（8.4），5-HT2A（10.2），5-HT2B（9.8），5-HT2C（10.5），5 -HT5A（8.8），5-HT6（9.5）和5-HT7（9.9）受体，肾上腺素α1（8.9），α2A（8.9），α2B（9.5）和α2C（8.9）受体，多巴胺D1（ 8.9），D2（8.9），D3（9.4）和D4（9.0）受体以及组胺H1（9.0）和H2（8.2）受体。 了解更多 -
Clomipramine HCl
Catalog No. A10231 5-HT Receptor 激动剂Clomipramine HCl是下列转运蛋白的阻滞剂：5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM)，去甲肾上腺素转运蛋白（NET）(Ki = 54 nM)，多巴胺转运蛋白（DAT）(Ki = 3，020 nM)，甘氨酸转运蛋白（GlyT/LeuT）。 了解更多 -
Dapoxetine hydrochloride
Catalog No. A10287 Dapoxetine hydrochloride是通过抑制5-羟色胺转运蛋白，增加5-羟色胺在突触后裂隙中的作用并因此促进射精延迟而起作用。 了解更多 -
Citalopram Hydrobromide
Catalog No. A10222 Citalopram Hydrobromide是ST（5-羟色胺/5-羟色胺转运蛋白）的选择性抑制剂，因此是一种有效且选择性的5-羟色胺再摄取抑制剂。 了解更多 -
Ketanserin (Vulketan Gel)
Catalog No. A10497 5-HT2A serotonin receptor 拮抗剂Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂，Ki为2.5 nM。 了解更多 -
Granisetron Hydrochloride
Catalog No. A10437 -
Almotriptan malate (Axert)
Catalog No. A11799 5-HT Receptor 激动剂Almotriptan malate (Axert)是一种选择性的5-羟色胺1B/1D（5-HT1B/1D）受体激动剂，用于治疗成人偏头痛。 了解更多 -
Aripiprazole (Abilify)
Catalog No. A11801 5-HT1A receptor 激动剂Aripiprazole (Abilify)是人5-HT1A受体部分激动剂，Ki为4.2 nM。 了解更多
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