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产品 851 到 900 共 2783个

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  1. Thalidomide-O-amido-PEG2-C2-NH2 (TFA)

    Catalog No. A21634
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    E3 ligase ligand-linker conjugate
    Thalidomide-O-amido-PEG2-C2-NH2 TFA is a synthesized E3 ligase ligand-linker conjugate that incorporates the Thalidomide based cereblon ligand and 2-unit PEG linker used in PROTAC technology. 了解更多
  2. SCH 50911

    Catalog No. A21630
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    γ-Aminobutyric acid B GABA(B) receptor antagonist
    SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist. 了解更多
  3. Fasudil

    Catalog No. A21628
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    ROCK inhibitor
    Fasudil (HA-1077; AT877), is a nonspecific ROCK inhibitor and also has inhibitory effect on protein kinases. 了解更多
  4. Mirogabalin

    Catalog No. A21626
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    Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS. 了解更多
  5. Nanatinostat

    Catalog No. A21625
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    HDAC inhibitor
    Nanatinostat (CHR-3996) is a potent, class I selective and orally active histone deacetylase (HDAC) inhibitor with an IC50 of 8 nM. 了解更多
  6. Pardoprunox hydrochloride

    Catalog No. A21624
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    partial dopamine D2 and D3 receptor agonist
    Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist. 了解更多
  7. Acetoacetic acid sodium salt

    Catalog No. A21621
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    Acetoacetic acid sodium salt is a metabolite of non-esterified fatty acids, involved in the development of human diabetes. Acetoacetic acid sodium salt induces oxidative stress to inhibit the assembly of very low density lipoprotein in bovine hepatocytes. 了解更多
  8. Tenosal

    Catalog No. A21619
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    Tenosal is a new compound obtained by esterifying salicylic acid with 2-thiophene-carboxylic acid and displays anti-inflammatory, analgesic and antipyretic properties. 了解更多
  9. Dasotraline

    Catalog No. A21618
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    triple reuptake inhibitor
    Dasotraline is a triple reuptake inhibitor that blocks dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respectively. 了解更多
  10. Ecteinascidin-Analog-1

    Catalog No. A21614
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    Ecteinascidin-Analog-1 is a useful intermediate for chemical sythesis of Ecteinascidin analogues; Ecteinascidins is a family of tetrahydroisoquinoline alkaloids with wide range of antitumor and antimicrobial activities. 了解更多
  11. Ionomycin

    Catalog No. A21611
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    Ionomycin (SQ23377) is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. 了解更多
  12. Cyantraniliprole D3

    Catalog No. A21610
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    Cyantraniliprole D3 is the deuterium labeled Cyantraniliprole, which is an insecticide of the ryanoid class. 了解更多
  13. Norepinephrine hydrochloride

    Catalog No. A21605
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    β1-selective adrenergic receptor agonist
    Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  14. 5-Hydroxy Propafenone D5 Hydrochloride

    Catalog No. A21604
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    5-Hydroxy Propafenone D5 Hcl is the deuterium labeled 5-Hydroxy Propafenone. 了解更多
  15. Ned 19

    Catalog No. A21597
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    NAADP antagonist
    Ned 19 is a selective membrane-permeant non competitive NAADP antagonist and inhibits NAADP-mediated Ca2+ signaling, with an IC50 of 65 nM. 了解更多
  16. BAY1217389

    Catalog No. A21595
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    MPS1 kinase inhibitor
    BAY 1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM. 了解更多
  17. Notch inhibitor 1

    Catalog No. A21591
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    Notch inhibitor
    Notch inhibitor 1 is a potent Notch inhibitor, with IC50s of 7.8 and 8.5 nM for Notch 1 and Notch 3, respectively. Used in the research of cancer. 了解更多
  18. Bupropion morpholinol D6

    Catalog No. A21587
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    Bupropion morpholinol D6 is a useful labeled metabolite of Bupropion. 了解更多
  19. EHNA hydrochloride

    Catalog No. A21585
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    Adenosine deaminase inhibitor
    EHNA hydrochloride is a specific inhibitor of adenosine deaminase, prevents dAdo degradation and increases mitochondrial dATP levels in fibroblasts. 了解更多
  20. AS2521780

    Catalog No. A21581
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    PKCθ selective inhibitor
    AS2521780 is a novel PKCθ selective inhibitor with an IC50 of 0.48 nM. 了解更多
  21. Ipragliflozin L-Proline

    Catalog No. A21579
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    SGLT2 inhibitor
    Ipragliflozin (L-Proline) is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6. 了解更多
  22. L-NIL

    Catalog No. A21576
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    inducible NO synthase inhibitor
    L-NIL is a potent and selective inhibitor of inducible NO synthase with IC50s of 3.3 and 92 μM for mouse inducible NO synthase and rat brain constitutive NO synthase, respectively. 了解更多
  23. SCH 546738

    Catalog No. A21554
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    CXCR3 antagonist
    SCH 546738 is a potent, orally active and non-competitive CXCR3 antagonist, the affinity constant (Ki) of SCH 546738 binding to human CXCR3 receptor is determined to be 0.4 nM in multiple experiments. 了解更多
  24. CDK9-IN-1

    Catalog No. A21552
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    CDK9 inhibitor
    CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87. 了解更多
  25. Gusperimus trihydrochloride

    Catalog No. A21551
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    Gusperimus trihydrochloride (Spanidin) is a derivative of the antitumor antibiotic spergualin with immunosuppressant activity. 了解更多
  26. BMS-983970

    Catalog No. A21547
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    pan-Notch inhibitor
    BMS-983970 is an oral pan-Notch inhibitor for the treatment of multiplecancers. 了解更多
  27. Diethyl aminoethyl hexanoate citrate

    Catalog No. A21544
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    plant growth regulator
    Diethyl aminoethyl hexanoate citrate is a compound that is widely used as a plant growth regulator. 了解更多
  28. Droxidopa

    Catalog No. A21541
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    Droxidopa(L-DOPS), the mixture of Droxidopa (w/w80%) and Pharmaceutical starch (w/w20%), acts as a prodrug to the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline). 了解更多
  29. Omadacycline hydrochloride

    Catalog No. A21540
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    Omadacycline hydrochloride is novel, aminomethyl tetracycline antibiotic being developed for the treatment of community-acquired bacterial infections. The ED50 for Escherichia coli is 2.02 mg/kg. 了解更多
  30. CCMI

    Catalog No. A21534
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    α7 nAChR-positive allosteric modulator
    CCMI is a potent and selective α7 nAChR-positive allosteric modulator, does not bind to or activate α7 nAChRs via the orthosteric site, and causes significant positive modulation of agonist-induced currents at α7 nAChRs. 了解更多
  31. LUF6000

    Catalog No. A21532
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    A3 adenosine receptor allosteric modulator
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). 了解更多
  32. Taribavirin

    Catalog No. A21525
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    inosine monophosphate dehydrogenase inhibitor
    Taribavirin is an orally active inosine monophosphate dehydrogenase inhibitor, has activity against a wide range of viruses, especially the hepatitis C virus and influenza virus. 了解更多
  33. (S)-(-)-Citronellal

    Catalog No. A21520
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    (S)-(-)-Citronellal ((-)-Citronellal) is a monoterpenoid compound found in Corymbia citriodora and Cymbopogon nardus essential oils. 了解更多
  34. 5'-GTP trisodium salt hydrate

    Catalog No. A21514
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    signal transducing G proteins activator
    5'-GTP trisodium salt hydrate is an activator of the signal transducing G proteins and also serves as an energy-rich precursor of mononucleotide units in the enzymatic biosynthesis of DNA and RNA. 了解更多
  35. Beclabuvir

    Catalog No. A21511
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    HCV NS5B RNA-dependent RNA polymerase inhibitor
    Beclabuvir is an allosteric inhibitor that binds to thumb site 1 of the hepatitis C virus (HCV) NS5B RNA-dependent RNA polymerase, and inhibits recombinant NS5B proteins from HCV genotypes 1, 3, 4, and 5 with IC50 of < 28 nM. 了解更多
  36. Tecarfarin sodium

    Catalog No. A21509
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    VKOR antagonist
    Tecarfarin sodium (ATI-5923 sodium) is a novel orally active non-competitive vitamin K epoxide reductase (VKOR) antagonist, impairs the activation of the vitamin K-dependent clotting factors II, VII, IX and X. 了解更多
  37. Rhosin

    Catalog No. A21504
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    RhoA subfamily Rho GTPases inhibitor
    Rhosin is a potent, specific RhoA subfamily Rho GTPases inhibitor, which specifically binds to RhoA to inhibit RhoA-GEF interaction with a Kd of ~ 0.4 uM, and does not interact with Cdc42 or Rac1, nor the GEF, LARG. Rhosin induces cell apoptosis. 了解更多
  38. Prinomastat

    Catalog No. A21501
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    metalloproteinase inhibitor
    Prinomastat (AG3340) is a broad spectrum, potent, orally active metalloproteinase (MMP) inhibitor with IC50s of 79, 6.3 and 5.0 nM for MMP-1, MMP-3 and MMP-9, respectively. 了解更多
  39. UAA crosslinker 1 hydrochloride

    Catalog No. A21496
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    UAA crosslinker 1 hydrochloride is an amber codon used for non-canonical amino acids (ncAAs) incorporation. The ncAAs can be incorporated into proteins in vivo by making use of the promiscuous activity of certain wildtype and engineered aminoacyl-tRNA synthetases. 了解更多
  40. Docebenone

    Catalog No. A21493
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    5-LO (5-lipoxygenase) inhibitor
    Docebenone (AA 861) is a potent, selective and orally active 5-LO (5-lipoxygenase) inhibitor. 了解更多
  41. Macozinone

    Catalog No. A21488
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    DprE inhibitor
    Macozinone (PBTZ169) is a bactericidal benzothiazinone and a potent DprE1 (decaprenylphosphoryl-β-d-ribose 2??-oxidase) inhibitor. 了解更多
  42. Givinostat hydrochloride

    Catalog No. A21487
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    HDAC inhibitor
    Givinostat hydrochloride (ITF-2357 hydrochloride) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多
  43. Delavirdine

    Catalog No. A21469
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    non-nucleoside reverse transcriptase inhibitor
    Delavirdine(U 90152) is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI). 了解更多
  44. Elinogrel

    Catalog No. A21468
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    platelet P2Y12 antagonist
    Elinogrel (PRT060128) is a potent, direct acting, competitive, and reversible platelet P2Y12 antagonist (IC50=20 nM). It is orally and intravenously available and has potent antiplatelet effects. 了解更多
  45. CDKI-73

    Catalog No. A21467
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    CDK9 inhibitor
    CDKI-73 is a potent CDK9 inhibitor with Ki of 4 nM; shows selective toxicity to CLL cells(LD50=80 nM) versus normal B cell and normal CD34+ cell(LD50>20 uM). 了解更多
  46. β-Apo-13-carotenone D3

    Catalog No. A21462
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    RXRα antagonist
    β-Apo-13-carotenone D3 is the deuterium labeled β-Apo-13-carotenone. β-Apo-13-carotenone (D'Orenone) is a naturally occurring β-apocarotenoid functioned as an antagonist of RXRα. 了解更多
  47. Betamethasone hydrochloride

    Catalog No. A21455
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    Betamethasone (hydrochloride) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties. 了解更多
  48. (±)-ANAP

    Catalog No. A21453
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    fluorescent probes
    (±)-ANAP is the unnatural amino acid analog of prodan, acts as a fluorescent probes, and enhances environmental sensitivity. 了解更多
  49. (-)-Talarozole

    Catalog No. A21451
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    retinoic acid metabolism inhibitor
    (-)-Talarozole is a potent inhibitor of retinoic acid metabolism extracted from patent WO 1997049704 A1. 了解更多
  50. DPN

    Catalog No. A21446
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    DPN (Diarylpropionitrile) is a non-steroidal estrogen receptor β(ER β) selective ligand. 了解更多

产品 851 到 900 共 2783个

每页
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  2. 17
  3. 18
  4. 19
  5. 20

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