“No”的搜索结果

产品 951 到 1000 共 2783个

每页
页面:
  1. 18
  2. 19
  3. 20
  4. 21
  5. 22

设置降序顺序
  1. OT-R antagonist 1

    Catalog No. A21216
    Quick View
    OT-R antagonist
    OT-R antagonist 1 is a new potent and selective nonpeptide low molecular weight OT-R antagonist. 了解更多
  2. MK-5046

    Catalog No. A21214
    Quick View
    BRS-3 agonist
    MK-5046 is a novel BRS-3 agonist, binds to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM). 了解更多
  3. AC-55541

    Catalog No. A21211
    Quick View
    PAR2 agonist
    AC-55541 is a highly selective protease-activated receptor 2 (PAR2) agonist (pEC50=6.7), displays no activity at other PAR subtypes or at over 30 other receptors involved in nociception and inflammation. 了解更多
  4. RAD140

    Catalog No. A21205
    Quick View
    androgen receptor modulator
    RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM). 了解更多
  5. BRD9539

    Catalog No. A21201
    Quick View
    EHMT2 inhibitor
    BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 ?M. 了解更多
  6. Zonampanel

    Catalog No. A21199
    Quick View
    glutamate receptor subtype antagonist
    Zonampanel (YM 872) is a selective antagonist of the glutamate receptor subtype, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) receptor. 了解更多
  7. Velneperit

    Catalog No. A21190
    Quick View
    NPY Y5 receptor antagonist
    Velneperit (S-2367) is a novel neuropeptide Y (NPY) Y5 receptor antagonist. 了解更多
  8. NB001

    Catalog No. A21185
    Quick View
    AC1 inhibitor
    NB001 (HTS 09836) is an adenylcyclase 1 (AC1) inhibitor which has effect on neural and non-neural pain by modulating AC1 activity. 了解更多
  9. (R)-Elagolix

    Catalog No. A21184
    Quick View
    GnRHR antagonist
    Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多
  10. IPA-3

    Catalog No. A21182
    Quick View
    PAK1 inhibitor
    IPA-3 is a selective non-ATP competitive PAK1 inhibitor with IC50 of 2.5 μM, and shows no inhibition to group II PAKs (PAKs 4-6). 了解更多
  11. Inolitazone

    Catalog No. A21180
    Quick View
    PPARγ agonist
    Inolitazone a novel high-affinity PPARγ agonist that is dependent upon PPARγ for its biological activity with IC50 of 0.8 nM for growth inhibition. 了解更多
  12. MK-0429

    Catalog No. A21173
    Quick View
    αvβ3 integrin antagonist
    MK-0429 (L-000845704) is an orally active, potent, selective and nonpeptide αvβ3 integrin antagonist with an IC50 of 80 nM. 了解更多
  13. BMS-906024

    Catalog No. A21172
    Quick View
    gamma secretase inhibitor
    BMS-906024 is an oral and selective gamma secretase inhibitor (GSI) that is a small molecule Notch inhibitor. 了解更多
  14. DL-O-Phosphoserine

    Catalog No. A21155
    Quick View
    DL-O-Phosphoserine, a normal metabolite in human biofluid, is an ester of serine and phosphoric acid. 了解更多
  15. Phenoxodiol

    Catalog No. A21147
    Quick View
    Phenoxodiol, a synthetic analog of Genestein, activates the mitochondrial caspase system, inhibits XIAP (an apoptosis inhibitor), and sensitizes the cancer cells to Fas-mediated apoptosis. 了解更多
  16. Alfacalcidol-D6

    Catalog No. A21142
    Quick View
    VDR activator
    Alfacalcidol-D6, a deuterated Alfacalcidol (1-hydroxycholecalciferol; Alpha D3; 1.alpha.-Hydroxyvitamin D3), is a non-selective VDR activator medication. 了解更多
  17. Merimepodib

    Catalog No. A21139
    Quick View
    IMPDH inhibitor
    Merimepodib is a noncompetitive and oral inhibitor of inosine monophosphate dehydrogenase (IMPDH) with broad spectrum antiviral activities. 了解更多
  18. (R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid

    Catalog No. A21136
    Quick View
    (R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid is a constrained Phe analogue which can fold into a beta-bend and a helical structure, and to adopt a preferred side-chain disposition in the peptide. 了解更多
  19. Ropidoxuridine

    Catalog No. A21128
    Quick View
    Ropidoxuridine (IPdR) is a novel orally available, halogenated thymidine analog and is a potential radiosensitizer for use in human tumors. 了解更多
  20. Givinostat

    Catalog No. A21126
    Quick View
    HDAC inhibitor
    Givinostat (ITF-2357) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多
  21. Roquinimex

    Catalog No. A21125
    Quick View
    Roquinimex (Linomide; PNU212616; ABR212616) is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis and reduces the secretion of TNF alpha. 了解更多
  22. Lagociclovir

    Catalog No. A21123
    Quick View
    against HBV activity
    Lagociclovir(MIV-210) is a prodrug of 3'-fluoro-2',3'-dideoxyguanosine with high oral bioavailability in humans and potent activity against HBV. 了解更多
  23. 6-FAM SE

    Catalog No. A21122
    Quick View
    6-FAM SE is another isomer of carboxyfluorescein. 6-FAM, SE is mainly used in sequencing of nucleic acids and labeling nucleotides. 了解更多
  24. 5(6)-Carboxyfluorescein

    Catalog No. A21120
    Quick View
    5(6)-Carboxyfluorescein contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid; cell-impermeant 5,6-FAM can also be used as a nonfixable polar tracer to investigate fusion, lysis and gap-junctional communication and to detect changes in cell or liposome volume. 了解更多
  25. 5(6)-FITC

    Catalog No. A21116
    Quick View
    5(6)-FITC (Fluorescein 5(6)-isothiocyanate) is an amine-reactive derivative of fluorescein dye that has wide-ranging applications as a label for antibodies and other probes, for use in fluorescence microscopy, flow cytometry and immunofluorescence-based assays such as Western blotting and ELISA. 了解更多
  26. 6-TAMRA

    Catalog No. A21109
    Quick View
    6-TAMRA has been a widely used fluorophore for preparing bioconjugates, especially fluorescent antibody and avidin derivatives used in immunochemistry. 了解更多
  27. Novaluron

    Catalog No. A21106
    Quick View
    Novaluron is a chemical with pesticide properties, belonging to the class of insecticides called insect growth regulators. 了解更多
  28. GLPG0492

    Catalog No. A21105
    Quick View
    androgen receptor modulator
    GLPG0492 is a novel selective androgen receptor modulator; exhibited anabolic activity on muscle, strongly dissociated from the androgenic activity on prostate after oral dosing. 了解更多
  29. Centanafadine

    Catalog No. A21099
    Quick View
    dual NE/DA transporter inhibitor
    Centanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively. 了解更多
  30. Meptyldinocap

    Catalog No. A21093
    Quick View
    Meptyldinocap (2,4-DNOPC) is a novel powdery mildew (Erysiphe necator) fungicide which shows protectant and post-infective activities. 了解更多
  31. Athidathion

    Catalog No. A21090
    Quick View
    Athidathion(GS-13006) is an organophosphate insecticide. 了解更多
  32. Mc-MMAE

    Catalog No. A21089
    Quick View
    tubulin inhibitor
    Mc-MMAE is a protective group (maleimidocaproyl)-conjugated monomethyl auristatin E (MMAE), which is a potent tubulin inhibitor. Mc-MMAE is a drug-linker conjugate for ADC. 了解更多
  33. Solenopsin

    Catalog No. A21087
    Quick View
    ATP-competitive AKT inhibitor
    Solenopsin is an ATP-competitive AKT inhibitor with IC50 value of 10 μM . 了解更多
  34. Gepotidacin

    Catalog No. A21086
    Quick View
    topoisomerase II inhibitor
    Gepotidacin (GSK2140944) is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor. 了解更多
  35. Benoxafos

    Catalog No. A21085
    Quick View
    Benoxafos (HOE 2910) is an insecticide. 了解更多
  36. Squalamine lactate

    Catalog No. A21076
    Quick View
    Squalamine lactate is an aminosterol compound discovered in the tissues of the dogfish shark, with antimicrobial activity, and used for the treatment of neovascular age-related macular degeneration. 了解更多
  37. Cyhalofop

    Catalog No. A21075
    Quick View
    Cyhalofop(Cyhalofop acid) is a recently registered herbicide from the aryloxyphenoxy propionate group in India to control a wide range of grass weed species at various growth stages in rice crop. 了解更多
  38. Ralinepag

    Catalog No. A21073
    Quick View
    IP receptor agonist
    Ralinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively. 了解更多
  39. VBY-825

    Catalog No. A21069
    Quick View
    cathepsin inhibitor
    VBY-825 is a novel, reversible cathepsin inhibitor with high potency against cathepsins B, L, S and V. 了解更多
  40. Ridinilazole

    Catalog No. A21068
    Quick View
    Ridinilazole is a novel antibacterial with MICs range of 0.06-0.25??g/mL (MIC90=8??g/mL) against C.?difficile. 了解更多
  41. Haloxon

    Catalog No. A21067
    Quick View
    Haloxon is an organophosphorus anthelmintic once used against nematodes of the abomasum and small intestine in ruminants. 了解更多
  42. N6-(4-Hydroxybenzyl)adenosine

    Catalog No. A21066
    Quick View
    platelet aggregation inhibitor
    N6-(4-Hydroxybenzyl)adenosine is a inhibitor of platelet aggregation induced in vitro by collagen and their activity range was demonstrated (IC50: 6.77-141 μM). 了解更多
  43. Chromafenozide

    Catalog No. A21065
    Quick View
    Chromafenozide (ANS118) is a lepidopteran insecticide; it is highly effective in controlling various lepidopteran pests. 了解更多
  44. Lisinopril

    Catalog No. A21064
    Quick View
    angiotensin-converting enzyme inhibitor
    Lisinopril (MK-521) is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks. 了解更多
  45. Artefenomel

    Catalog No. A21050
    Quick View
    Artefenomel (OZ439) is a synthetic antimalarial agent with the artemisinin pharmacophore. Artefenomel (OZ439) is a long-acting artemisinin-related agent. 了解更多
  46. Azimilide

    Catalog No. A20944
    Quick View
    class III antiarrhythmic compound
    Azimilide(NE-10064) is a class III antiarrhythmic compound, inhibits I(Ks) and I(Kr) in guinea-pig cardiac myocytes and I(Ks) (minK) channels expressed in Xenopus oocytes. 了解更多
  47. Carboxyamidotriazole

    Catalog No. A20940
    Quick View
    non-voltage dependent calcium channel blocker
    Carboxyamidotriazole (L 651582) is a blocker of non-voltage dependent calcium channel. 了解更多
  48. K-Ras G12C-IN-1

    Catalog No. A20937
    Quick View
    K-ras G12C inhibitor
    K-Ras G12C-IN-1 is a novel and irreversible inhibitor of mutant K-ras G12C extracted from patent WO 2014152588 A1. 了解更多
  49. ITX3

    Catalog No. A20934
    Quick View
    TrioN inhibitor
    ITX3 is a specific and nontoxic inhibitor of the TrioN (N-terminal GEF domain of the multidomain Trio protein) with IC50 of 76 uM; inhibits TrioN-stimulated RhoG exchange in vitro. 了解更多
  50. Dihexa

    Catalog No. A20933
    Quick View
    Dihexa, an oligopeptide drug, is an orally active and blood-brain barrier-permeable angiotensin IV analog. 了解更多

产品 951 到 1000 共 2783个

每页
页面:
  1. 18
  2. 19
  3. 20
  4. 21
  5. 22

设置降序顺序
Rewards