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产品 1051 到 1100 共 2783个

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  1. Landiolol hydrochloride

    Catalog No. A17675
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    adrenoceptor antagonist
    Landiolol hydrochloride (ONO1101 hydrochloride) is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity?=?255:1, a half-life of 4?min)?? acts as an adrenoceptor antagonist. 了解更多
  2. Bedaquiline fumarate

    Catalog No. A17444
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    Bedaquiline fumarate, a diarylquinoline antibiotic that targets ATP synthase, is effective for the treatment of Mycobacterium tuberculosis infections. 了解更多
  3. Pinacidil monohydrate

    Catalog No. A17380
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    Pinacidil monohydrate, an antihypertensive drug, is a potassium channel activator. 了解更多
  4. Clorgyline hydrochloride

    Catalog No. A17357
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    monoamine oxidase A inhibitor
    Clorgyline hydrochloride is an irreversible and selective inhibitor of monoamine oxidase A (MAO-A) that is used in scientific research; structurally related to Pargyline. 了解更多
  5. Avibactam sodium

    Catalog No. A17306
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    non-β-lactam β-lactamase inhibitor
    Avibactam sodium (NXL-104) is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively. 了解更多
  6. Grazoprevir

    Catalog No. A17303
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    Hepatitis C virus NS3/4a protease inhibitor
    Grazoprevir (MK-5172) is a selective inhibitor of Hepatitis C virus NS3/4a protease with broad activity across genotypes and resistant variants, with Kis of 0.01 nM (gt1b), 0.01 nM (gt1a), 0.08 nM (gt2a), 0.15 nM (gt2b), 0.90 nM (gt3a), respectively. 了解更多
  7. SB-334867 free base

    Catalog No. A16695
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    orexin OX1 receptor antagonist
    SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. 了解更多
  8. Oclacitinib maleate

    Catalog No. A16640
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    JAK inhibitor
    Oclacitinib maleate (PF-03394197 maleate) is a novel JAK inhibitor. Oclacitinib maleate (PF-03394197 maleate) is most potent at inhibiting JAK1 (IC50=10 nM). 了解更多
  9. L-Glutamic acid monosodium salt

    Catalog No. A16591
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    excitatory transmitter/agonist
    L-Glutamic acid monosodium salt acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). (S)-Glutamic acid shows a direct activating effect on the release of DA from dopaminergic terminals. 了解更多
  10. Indacaterol maleate

    Catalog No. A16585
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    β-adrenoceptor agonist
    Indacaterol (QAB149) maleate is an ultra-long-acting β-adrenoceptor agonist. 了解更多
  11. Diethylcarbamazine citrate

    Catalog No. A16506
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    arachidonic acid metabolism inhibitor
    Diethylcarbamazine citrate is an inhibitor of arachidonic acid metabolism in filarial microfilaria; is highly specific for several parasites and does not contain any toxic metallic elements. 了解更多
  12. Diclofenac diethylamine

    Catalog No. A16503
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    COX inhibitor
    Diclofenac diethylamine is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor. 了解更多
  13. 2-Deoxy-D-glucose

    Catalog No. A16478
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    glucose metabolism inhibitor
    2-Deoxy-D-glucose is a glucose analog that acts as a competitive inhibitor of glucose metabolism, inhibiting glycolysis via its actions on hexokinase. 了解更多
  14. Tectochrysin

    Catalog No. A15679
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    Tectochrysin (Techtochrysin) is one of the major flavonoids of Alpinia oxyphylla Miquel. Tectochrysin (Techtochrysin) inhibits activity of NF-κB. 了解更多
  15. Kaempferide

    Catalog No. A15673
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    Kaempferide is an O-methylated flavonol, a type of chemical compound. 了解更多
  16. 2,6-Dimethoxybenzoic acid

    Catalog No. A15595
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    2,6-Dimethoxybenzoic acid is a member of organic compounds known as o-methoxybenzoic acids and derivatives. 了解更多
  17. ABT-239

    Catalog No. A14093
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    non-imidazole class of H3R antagonist
    ABT-239 is a novel, highly efficacious, non-imidazole class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist. 了解更多
  18. Talabostat

    Catalog No. A14079
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    DPP-IV inhibitor
    Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM). 了解更多
  19. N6,N6-Dimethyladenosine

    Catalog No. A13782
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    N6,N6-Dimethyladenosine is a modified ribonucleoside previously found in rRNA, and also exhibits in mycobacterium bovis Bacille Calmette-Gu??rin tRNA. 了解更多
  20. N-Bis(2-hydroxypropyl)nitrosamine

    Catalog No. A13614
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    N-Bis(2-hydroxypropyl)nitrosamine is an agent with carcinogenic activity. 了解更多
  21. 2,4-Diamino-6-hydroxypyrimidine

    Catalog No. A13500
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    GTP cyclohydrolase I inhibitor
    2,4-Diamino-6-hydroxypyrimidine is a specific GTP cyclohydrolase I inhibitor (the rate-limiting enzyme in de novo pterin synthesis), blocks BH4 synthesis and suppresses NO production. 了解更多
  22. 6-Quinoxalinecarboxylic acid, 2,3-bis(bromomethyl)-

    Catalog No. A13373
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    6-Quinoxalinecarboxylic acid, 2,3-bis(bromomethyl)-, derived from 2,3-Bis(bromomethyl)quinoxaline, shows antibacterial activity. 了解更多
  23. Benzo[a]pyrene

    Catalog No. A13158
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    Benzo[a]pyrene shows lung carcinogenicity in animal models, and it is frequently used in chemoprevention studies. 了解更多
  24. Sutezolid

    Catalog No. A12638
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    oxazolidinone antimicrobial
    Sutezolid (PNU-100480) is an oxazolidinone antimicrobial being developed for the treatment of tuberculosis. 了解更多
  25. 6-(γ,γ-Dimethylallylamino)purine

    Catalog No. A12636
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    6-(γ,γ-Dimethylallylamino)purine is a plant growth substance. 了解更多
  26. Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  27. SMND-309

    Catalog No. A11576
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    SMND-309 is a metabolite of salvianolic acid B, and exhibits neuroprotective effects in cultured neurons and in permanent middle cerebral artery occlusion rats. 了解更多
  28. R-1479

    Catalog No. A11540
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    HCV replication inhibitor
    R-1479 is a specific inhibitor of HCV replication in the HCV subgenomic replicon system (IC50=1.28 μM). 了解更多
  29. Pitolisant

    Catalog No. A11525
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    nonimidazole inverse agonist
    Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). 了解更多
  30. Poloxin

    Catalog No. A11524
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    PLK1 inhibitor
    Poloxin is a non-ATP competitive Polo-like Kinase 1 (PLK1) inhibitor that targets the polo-box domain, with an IC50 of appr 4.8 μM. 了解更多
  31. Olcegepant

    Catalog No. A11512
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    CGRP1 receptor
    Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. 了解更多
  32. JDTic dihydrochloride

    Catalog No. A11469
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    KOR antagonist
    JDTic (dihydrochloride) is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception. 了解更多
  33. HIV-1 integrase inhibitor 2

    Catalog No. A11447
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    HIV-1 integrase inhibitor
    HIV-1 integrase inhibitor 2, in the treatment of human immunodeficiency virus (HIV) infection. 了解更多
  34. CGS 21680

    Catalog No. A11354
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    adenosine A2A receptor agonist
    CGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. 了解更多
  35. Flurbiprofen

    Catalog No. A10401
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    nonsteroidal anti-inflammatory agent
    Flurbiprofen is a nonsteroidal anti-inflammatory agent (NSAIA) with antipyretic and analgesic activity. 了解更多
  36. Kynurenic acid sodium

    Catalog No. A20000
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    GPR35/CXCR8 agonist
    Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多
  37. MT-7716 hydrochloride

    Catalog No. A20004
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    NOP agonist
    MT-7716 hydrochloride (W-212393 hydrochloride) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. 了解更多
  38. SKF-96365 hydrochloride

    Catalog No. A16706
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    TRP Channel blocker
    SKF-96365 hydrochloride is a non-selective TRP Channel blocker. 了解更多
  39. Rbin-1

    Catalog No. A16682
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    Eukaryotic ribosome biogenesis inhibitor
    Rbin-1 is a potent, reversible, and specific chemical inhibitor of eukaryotic ribosome biogenesis. Rbin-1 inhibits the ATPase with GI50 of 136 nM. Rbin-1 is a potent and selective chemical inhibitor of Midasin (Mdn1). 了解更多
  40. alpha-Amanitin

    Catalog No. A14097
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    alpha-Amanitin is the principal toxin of several deadly poisonous mushrooms, exerting its toxic function by inhibiting RNA-polymerase II. 了解更多
  41. β-Chloro-L-alanine

    Catalog No. A13223
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    β-Chloro-L-alanine is a bacteriostatic amino acid analog which inhibits a number of enzymes, including threonine deaminase and alanine racemase. 了解更多
  42. Docosahexaenoic Acid methyl ester

    Catalog No. A12315
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    Docosahexaenoic Acid methyl ester is a methylated docosahexaenoic acid analog which can be intercalated into membrane phospholipids without being oxidized or hydrolyzed. 了解更多
  43. Gastrofensin AN 5 free base

    Catalog No. A13301
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    Gastrofensin AN 5 free base, a 4-phenyl-tetrahydroisoquinoline derivative, is an antiulcer agent. 了解更多
  44. Oleanolic acid hemiphthalate disodium salt

    Catalog No. A13337
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    Oleanolic acid hemiphthalate disodium salt is an anti-inflammatory agent. 了解更多
  45. 5-Amino-3H-imidazole-4-Carboxamide

    Catalog No. A12155
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    5-Amino-3H-imidazole-4-Carboxamide (AICA) is an important precursor for the synthesis of purines in general and of the nucleobases adenine and guanine in particular. 了解更多
  46. Inogatran

    Catalog No. A13356
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    synthetic thrombin inhibitor
    Inogatran (H-314-27) is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of arterial and venous thrombotic diseases. 了解更多
  47. 20-HEDE

    Catalog No. A12466
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    20-HETE antagonist
    20-HEDE (WIT 002) is an antagonist of 20-hydroxyeicosatetraenoic acid (20-HETE). 了解更多
  48. NMDI14

    Catalog No. A12958
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    NMD inhibitor
    NMDI14 is a nonsense mediated RNA decay (NMD) inhibitor. 了解更多
  49. AQ-13 dihydrochloride

    Catalog No. A12178
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    AQ-13 dihydrochloride is an aminoquinoline antimalarial drug that is effective against chloroquine-resistant strains of Plasmodium falciparum. 了解更多
  50. Pirazolac

    Catalog No. A12477
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    Pirazolac is a non-steroidal anti-inflammatory drug. 了解更多

产品 1051 到 1100 共 2783个

每页
页面:
  1. 20
  2. 21
  3. 22
  4. 23
  5. 24

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