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产品 1101 到 1150 共 2783个

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  1. FR167344 free base

    Catalog No. A12964
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    nonpeptide bradykinin receptor B2 antagonist
    FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. 了解更多
  2. L-873724

    Catalog No. A12487
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    Cathepsin K inhibitor
    L-873724 is a potent, orally bioavailable, selective and reversible non-basic cathepsin K inhibitor. 了解更多
  3. Salsolidine

    Catalog No. A12969
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    MAO-A inhibitor
    Salsolidine is a tetrahydroisoquinoline alkaloid, acts as a stereoselective competitive MAO A inhibitor. 了解更多
  4. P-gp inhibitor 1

    Catalog No. A13384
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    P-gp inhibitor
    P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多
  5. (+)-Cloprostenol

    Catalog No. A12979
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    prostaglandin F2α (PGF2α) analogue
    (+)-Cloprostenol is a prostaglandin F2α (PGF2α) analogue, and shows selective agonistic activity at the prostaglandin receptor. 了解更多
  6. BCR-ABL-IN-1

    Catalog No. A12496
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    BCR-ABL inhibitor
    BCR-ABL-IN-1 is an inhibitor of BCR-ABL tyrosine kinase, with a pIC50 of 6.46, and may be used in the research of chronic myelogenous leukemia. 了解更多
  7. RN-18

    Catalog No. A12980
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    HIV-1 Vif inhibitor
    RN-18 is a HIV-1 viral infectivity factor (HIV-1 Vif) inhibitor with an IC50 of 6 μM in nonpermissive H9 cells. 了解更多
  8. STING agonist-1

    Catalog No. A12497
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    human-specific STING agonist
    STING agonist-1 (G10) is a novel human-specific STING agonist that elicits antiviral activity against emerging Alphaviruses. 了解更多
  9. AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  10. CX-157

    Catalog No. A12200
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    MAO-A inhibitor
    CX-157 is a reversible inhibitor of monoamine oxidase-A (MAO-A) with an EC50 of 19.3?ng/mL. 了解更多
  11. Orexin A

    Catalog No. A13009
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    Orexin A human, rat, mouse is a 33 amino acid excitatory neuropeptide. Orexin A human, rat, mouse works on 2 specific G protein-coupled receptors (GPCRs): orexin-1 (OX1) and orexin-2 (OX2). 了解更多
  12. Ruzadolane

    Catalog No. A13425
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    Ruzadolane (UP 26-91) is a non-narcotic, centrally-acting analgesic agent. 了解更多
  13. Pentiapine

    Catalog No. A12512
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    dopamine release inhibitor
    Pentiapine is a novel dopamine release inhibitor. 了解更多
  14. Benzenepentacarboxylic Acid

    Catalog No. A13012
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    Benzenepentacarboxylic acid (BA), a novel fluorescent probes to detect and scavenge HO-. 了解更多
  15. Oxypurinol

    Catalog No. A13431
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    Xanthine oxidase inhibitor
    Oxipurinol (Oxipurinol), the major active metabolite of Allopurinol, is an inhibitor of xanthine oxidase. Oxipurinol can be used to regulate blood urate levels and treat gout. 了解更多
  16. Ranolazine dihydrochloride

    Catalog No. A10781
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    Ranolazine dihydrochloride (CVT 303 dihydrochloride) is an anti-angina drug that achieves its effects by inhibiting the late phase of inward sodium current (INa and IKr with IC50 values of 6 μM and 12 μM, respectively) without affecting heart rate or blood pressure (BP). 了解更多
  17. Ziprasidone hydrochloride monohydrate

    Catalog No. A11008
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    5-HT (serotonin) and dopamine receptor antagonist
    Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  18. Medetomidine

    Catalog No. A11494
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    α2-adrenoceptor agonist
    Medetomidine(Domtor) is a potent, highly selective α2-adrenoceptor agonist (Ki values are 1.08 and 1750 nM for α2- and α1-adrenoceptors respectively). 了解更多
  19. ONO-AE3-208

    Catalog No. A11516
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    EP4 antagonist
    ONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. 了解更多
  20. Rocuronium

    Catalog No. A11551
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    neuromuscular blocker
    Rocuronium (Org-9426) is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia. 了解更多
  21. Ethylmalonic acid

    Catalog No. A12243
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    Ethylmalonic acid is non-carcinogenic potentially toxic and associated with anorexia nervosa and malonyl-CoA decarboxylase deficiency. 了解更多
  22. N-563

    Catalog No. A12245
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    N-563 is an analogue of deoxyspergualin with an immunostimulating activity,it promotes resistance to Candida albicans infection in mice. 了解更多
  23. W-2429

    Catalog No. A12246
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    non-narcotic analgesic agent
    W-2429 is a non-narcotic analgesic agent. 了解更多
  24. 2'-Hydroxy-4'-methylacetophenone

    Catalog No. A12248
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    2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. It could be used in the preparation of 4??-methyl-2??-[(p-tolylsulfonyl) oxy] acetophenone. 了解更多
  25. Norverapamil hydrochloride

    Catalog No. A12249
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    P-gp inhibitor
    Norverapamil hydrochloride ((??)-Norverapamil hydrochloride), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor. 了解更多
  26. CXD101

    Catalog No. A12253
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    HDAC inhibitor
    CXD101 is a class I-selective HDAC inhibitor (HDAC1 (IC50, 63 nM), HDAC2 (IC50, 570 nM), HDAC3 (IC50, 550 nM). CXD101 has no activity against HDAC class II. 了解更多
  27. L-690330

    Catalog No. A12255
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    IMPase inhibitor
    L-690330 is a competitive inhibitor of inositol monophosphatase (IMPase) with Kis of 0.27 and 0.19 μM for recombinant human and bovine IMPase, 0.30 and 0.42 μM for human and bovine frontal cortex IMPase, respectively. 了解更多
  28. Aglafoline

    Catalog No. A12257
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    PAF antagonist
    Aglafoline is an effective PAF antagonist not only in vitro, but also in vivo. 了解更多
  29. Nicainoprol

    Catalog No. A12269
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    Nicainoprol is a fast-sodium-channel blocking drug, which is a potent antiarrhythmic agent. 了解更多
  30. 2',3'-cGAMP

    Catalog No. A12277
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    2',3'-cGAMP (2'-3'-cyclic GMP-AMP) is a endogenous cGAMP in mammalian cells. 了解更多
  31. Kinetin riboside

    Catalog No. A12284
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    PINK1 activator
    Kinetin riboside is an activator of the Parkinson's Disease-associated PTEN-induced Putative Kinase 1 (PINK1), and acts independently from mitochondrial depolarization. 了解更多
  32. TOK-8801

    Catalog No. A12288
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    immunomodulator
    TOK-8801 is a synthesized dihydroimidazothiazole carboxamide and is under development as an immunomodulator. 了解更多
  33. 3-arylisoquinolinamine derivative

    Catalog No. A12292
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    3-arylisoquinolinamine derivative is a 3-arylisoquinolinamine derivative with antitumor activity. 了解更多
  34. LR-90

    Catalog No. A12296
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    AGE inhibitor
    LR-90 is an advanced glycation end product (AGE) inhibitor, inhibits inflammatory responses in human monocytes. LR-90 is also used in the research of diabetic animal model. 了解更多
  35. RP 54275

    Catalog No. A12302
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    RP 54275 (2-Octadecyl-1H-indole-5-carboxylic acid) is a novel hypocholesterolaemic drug. 了解更多
  36. CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  37. Ipenoxazone

    Catalog No. A12307
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    Ipenoxazone is a potent and centrally acting muscle relaxant. 了解更多
  38. Indole-3-carboxylic acid

    Catalog No. A12338
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    Indole-3-carboxylic acid is a normal urinary indolic tryptophan metabolite and has been found elevated in patients with liver diseases. 了解更多
  39. Tepilamide fumarate

    Catalog No. A12525
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    Tepilamide fumarate (XP-23829) is an oral fumaric acid ester, acts as a prodrug of monomethyl fumarate, and is used in the research of moderate to severe chronic plaque psoriasis. 了解更多
  40. 9-amino-CPT

    Catalog No. A12540
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    Topoisomerase I inhibitor
    9-Aminocamptothecin is a topoisomerase I inhibitor with potent anticancer activity. 了解更多
  41. CCT251236

    Catalog No. A12543
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    CCT251236 is an orally available pirin ligand from a heat shock transcription factor 1 (hsf1) phenotypic screen with an IC50 of 19 nM for inhibition of HSF1-mediated HSP72 induction. 了解更多
  42. Dot1L-IN-1

    Catalog No. A12552
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    Dot1L inhibitor
    Dot1L-IN-1 is a highly potent, selective and structurally novel Dot1L inhibitor with a Ki of 2 pM. 了解更多
  43. BETd-260

    Catalog No. A12563
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    BET degrader
    BETd-260 is a potent BET degrader based on PROTAC technology, with as low as 30 pM against BRD4 protein in RS4;11 leukemia cell line. 了解更多
  44. ITE

    Catalog No. A12565
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    AhR agonist
    ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR), binding directly to AHR, with a Ki of 3 nM. ITE also has immunosuppressive activity. 了解更多
  45. (S)-2-Hydroxy-3-phenylpropanoic acid

    Catalog No. A12566
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    (S)-2-Hydroxy-3-phenylpropanoic acid is a product of phenylalanine catabolism. An elevated level of phenyllactic acid is found in body fluids of patients with or phenylketonuria. 了解更多
  46. A2A receptor antagonist 1

    Catalog No. A12567
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    adenosine A2A/A1 receptor antagonist
    A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多
  47. ABT-639 hydrochloride

    Catalog No. A12571
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    T-type Ca2+ channel blocker
    ABT-639 hydrochloride is a novel, peripherally acting, selective T-type Ca2+ channel blocker. 了解更多
  48. NSC632839

    Catalog No. A12573
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    isopeptidase inhibitor
    NSC632839 is a nonselective isopeptidase inhibitor, which inhibits USP2, USP7, and SENP2 with EC50s of 45??4 μM, 37??1 μM, and 9.8??1.8 μM, respectively. 了解更多
  49. 2-Aminoethyl-mono-amide-DOTA-tris(tBu ester)

    Catalog No. A12574
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    2-Aminoethyl-mono-amide-DOTA-tris(tBu ester) is a macrocycle DOTA derivative for tumor pretargeting. 了解更多
  50. (R)-(+)-Citronellal

    Catalog No. A12577
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    (R)-(+)-Citronellal, isolated from citrus, lavender and eucalyptus oils, is a monoterpenoid and main component of citronellal oil with a distinct lemon scent. A flavouring agent. Used for insect repellent and antifungal properties. 了解更多

产品 1101 到 1150 共 2783个

每页
页面:
  1. 21
  2. 22
  3. 23
  4. 24
  5. 25

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