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Deltarasin HCl
Catalog No. A13722 -
CFTR-Inhibitor-II
Catalog No. A13723 CFTR 抑制剂CFTR inhibitor II,也称为GlyH-101，是一种甘氨酸酰肼，可选择性和可逆地阻断CFTR通道（Ki = 4.3 uM）。 了解更多 -
LB42708
Catalog No. A14020 -
R428
Catalog No. A13741 -
Atorvastatin
Catalog No. A13743 HMG-CoA reductase 抑制剂Atorvastatin是一种HMG-CoA还原酶抑制剂（IC50 = 154 nM），可有效治疗高胆固醇血症和某些血脂异常。 了解更多 -
GSK2801
Catalog No. A14015 -
CID 755673
Catalog No. A13804 PKD 抑制剂CID755673是一种具有细胞活性的泛PKD1/2/3抑制剂，IC50值分别为180 nM，280nM，以及227 nM。 了解更多 -
BAY 87-2243
Catalog No. A12978 -
CZC-25146 hydrochloride
Catalog No. A13448 -
Selinexor (KPT-330)
Catalog No. A12582 CRM1 抑制剂CRM1（XPO1）介导的核输出的KPT-330抑制剂在T细胞急性淋巴细胞白血病和急性骨髓性白血病的临床前模型中具有选择性的抗白血病活性。 了解更多 -
GDC0994 (Ravoxertinib)
Catalog No. A13420 ERK1/2 抑制剂GDC-0994是一种强效选择性Erk1/2抑制剂。GDC-0994抑制ERK磷酸化和ERK介导的信号转导通路的激活。 了解更多 -
GBR 12783 dihydrochloride
Catalog No. A13128 dopamine uptake 抑制剂GBR 12783 dihydrochloride是一种非常有效的选择性多巴胺摄取抑制剂（抑制大鼠纹状体突触体中[3H]-多巴胺摄取的IC50为1.8 nM）。 了解更多 -
ONX 0912 (Oprozomib)
Catalog No. A14181 Proteasome 抑制剂ONX 0912 (Oprozomib)是一种三肽环氧酮，可抑制对常规和硼替佐米治疗耐药的MM细胞的生长并诱导其凋亡。 了解更多 -
ML-323
Catalog No. A14030 -
SGI 1027
Catalog No. A14120 -
B-Raf-inhibitor 1
Catalog No. A14122 B-Raf 抑制剂B-Raf inhibitor 1是有效的选择性B-Raf抑制剂，对A375增殖和A375 p-ERK的细胞IC50分别为0.31 uM和2 nM。 了解更多 -
TG-02 (SB1317)
Catalog No. A11962 -
Losmapimod (GW856553X)
Catalog No. A12526 p38 MAPK 抑制剂Losmapimod，也称为GW856553或GW856553X，是葛兰素史克（GlaxoSmithKline）开发的药物，可作为酶家族的选择性抑制剂，称为p38促分裂原活化蛋白激酶，其作用于p38α和p38β的pKi分别为8.1和7.6 。 了解更多 -
Alvelestat
Catalog No. A12779 neutrophil elastase 抑制剂Avelestat，也称为AZD9668，是可口服的,高度选择性neutrophil elastase (NE)抑制剂，IC50和Ki分别为12 nM和9.4 nM,其选择性超过其他丝氨酸蛋白酶至少600倍。 了解更多 -
PF-543
Catalog No. A13039 -
E 64d (Aloxistatin)
Catalog No. A13259 Cysteine Protease 抑制剂E 64d (Aloxistatin)是组织蛋白酶B和L的抑制剂，具有溶酶体和细胞渗透性。 了解更多 -
GM 6001
Catalog No. A13320 -
Tiplaxtinin (PAI-039)
Catalog No. A14190 PAI-1 inhbitorTiplaxtinin (PAI-039)是一种纤溶酶原激活物抑制剂1（PAI-1）的选择性口服有效抑制剂，IC50为2.7μM。 了解更多 -
K-Ras(G12C) inhibitor 6
Catalog No. A14103 K-Ras(G12C) 抑制剂K-Ras(G12C) inhibitor 6 是致癌性K-Ras（G12C）的不可逆抑制剂，颠覆了天然核苷酸的偏爱性，使GDP优于GTP。 了解更多 -
GSK1324726A (I-BET726)
Catalog No. A14133 BET 抑制剂GSK1324726A (I-BET726)是一种新型、高效、选择性的BET蛋白小分子抑制剂，对BRD2（IC50 = 41 nM）、BRD3（IC50 = 31 nM）和BRD4（IC50 = 22 nM）具有高度的亲和力。 了解更多 -
Cerdulatinib
Catalog No. A14210 multi-targeted tyrosine kinase 抑制剂Cerdulatinib (PRT-062070)是多靶点酪氨酸激酶抑制剂，对JAK1/JAK2/JAK3/TYK2和Syk的IC50分别为12 nM/6 nM/8 nM/0.5 nM和32 nM。 了解更多
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