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￥ 0.00 5-HT Receptors
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Lu AE58054 (Idalopirdine)
Catalog No. A12521 -
Tandospirone
Catalog No. A13293 5-HT Receptor 拮抗剂Tandospirone是5HT1A受体的部分激动剂。它以剂量依赖性方式显着降低氟哌啶醇诱导的运动迟缓。 了解更多 -
SB-742457
Catalog No. A14092 -
SB 399885 HCl
Catalog No. A14102 5-HT6 拮抗剂SB 399885 hydrochloride是一种有效的，脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍（对于人类重组，天然大鼠和天然人类SR-6受体，pKi值分别为9.11、8.81和9.02）。 了解更多 -
Cyclobenzaprine HCl
Catalog No. A14255 -
Tropisetron HCL
Catalog No. A14375 5-HT3 receptor 拮抗剂Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂，对5-HT3受体的IC50为70.1±0.9 nM。 了解更多 -
NAN-190 hydrobromide
Catalog No. A13417 5-HT1A receptor 拮抗剂NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂，但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多 -
Clozapine N-oxide
Catalog No. A15048 5-HT1C receptor 拮抗剂Clozapine N-oxide是氯氮平的主要代谢产物，在体外可降低SR-2A（5-HT2血清素受体）密度。 了解更多 -
Ziprasidone
Catalog No. A15286 5-HT/dopamine receptor 拮抗剂Ziprasidone是5-HT（5-羟色胺）和多巴胺受体拮抗剂的组合，具有抗精神病活性。 了解更多 -
Alosetron Hydrochloride
Catalog No. A14989 -
Cyproheptadine hydrochloride
Catalog No. A16169 -
Azasetron HCl
Catalog No. A16417 5-HT3 receptor 拮抗剂Azasetron HCl是一种选择性的5-HT3受体拮抗剂，IC50为0.33 nM，用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多 -
LY 334370 hydrochloride
Catalog No. A17027 5-HT1F 激动剂LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂（Ki值为1.87、16.4，> 100 (IC50)）。CAS：199673-74-0（LY 334370盐酸盐）；182563-08-2（LY 334370游离碱） 了解更多 -
Volinanserin
Catalog No. A17115 -
Dolasetron
Catalog No. A17595 5-HT3 receptor antagonistDolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多 -
Dolasetron Mesylate
Catalog No. A17729 5-HT3 receptor antagonistDolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多 -
Alprenolol hydrochloride
Catalog No. A17781 5-HT1A receptor antagonistAlprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多 -
Alosetron (Hydrochloride(1:X))
Catalog No. A11309 Serotonin 5HT3-receptor antagonistAlosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多