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GPCR / G Protein

28 个项目

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  1. NNC0640
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    NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多
  2. VU0453379
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    VU0453379

    Catalog No. A18796
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    GLP-1R modulator
    VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM. 了解更多
  3. E1R
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    E1R

    Catalog No. A18825
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    sigma-1 receptors modulator
    E1R is a novel positive allosteric modulator of sigma-1 receptors. 了解更多
  4. RPC1063 (Ozanimod)
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    RPC1063 (Ozanimod)

    Catalog No. A15819
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    S1PR1 modulators
    RPC1063 (Ozanimod)是选择性的鞘氨醇1磷酸酯受体调节剂和方法，可用于治疗与S1P1-β相关的疾病。 了解更多
  5. NS13001
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    NS13001

    Catalog No. A15833
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    SK2 modulator
    NS13001是选择性的SK2/3调节剂，可作为治疗SCA2和其他可能的小脑共济失调的潜在治疗剂。 了解更多
  6. Ponesimod
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    Ponesimod

    Catalog No. A13307
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    S1P1 receptor modulator
    Ponesimod是一种口服活性，选择性鞘氨醇-1-磷酸受体1（S1P1）免疫调节剂，EC50为5.7 nM。 了解更多
  7. SBI-553
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    SBI-553

    Catalog No. A18435
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    NTR1 allosteric modulator
    SBI-553 is a potent and brain penetrant NTR1 allosteric modulator. 了解更多
  8. Org 27569
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    Org 27569

    Catalog No. A11513
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    CB1 modulator?
    Org 27569是一种强效CB1受体变构调节剂(PEC50 = 8.24)。 了解更多
  9. LUF6000
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    LUF6000

    Catalog No. A21532
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    A3 adenosine receptor allosteric modulator
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). 了解更多
  10. Endothelin Mordulator 1
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    Endothelin Mordulator 1

    Catalog No. A13040
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    endothelin receptor modulator
    Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多
  11. NSC-23026
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    NSC-23026

    Catalog No. A17151
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    CXCR4 receptor modulator
    NSC-23026是CXCR4受体调节剂。 了解更多
  12. VU 0364770
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    VU 0364770

    Catalog No. A12139
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    mGlu4 receptors modulator
    VU 0364770是mGlu4受体的正变构调节剂，在表达mGlu4的HEK 293细胞中EC50值为290 nM。 了解更多
  13. JNJ 42153605
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    JNJ 42153605

    Catalog No. A14330
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    mGluR-2 modulator
    JNJ-42153605是亲代谢型谷氨酸2受体的正变构调节剂。 了解更多
  14. ADX-47273
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    ADX-47273

    Catalog No. A11181
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    mGluR5 modulator
    ADX-47273是一种有效的，特异性的mGlu5正变构调节剂(PAM)EC50为0.17 μM，对其他亚型没有作用活性。 了解更多
  15. VU 0364439
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    VU 0364439

    Catalog No. A12664
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    GluR modulator
    VU 0364439是mGlu4受体的正变构调节剂（PAM）（对于人mGlu4，体外EC50 = 19.8 nM）。 了解更多
  16. BINA
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    BINA

    Catalog No. A11126
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    mGluR2 modulator
    BINA是mGlu2的选择性正构构调节剂（在表达人mGlu2的CHO细胞中EC50 = 33.2 nM）。 了解更多
  17. VU 0361737
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    VU 0361737

    Catalog No. A12467
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    mGlu4 receptors modulator
    VU 0361737是mGluR-4的选择性正变构调节剂（人和大鼠受体的EC50值分别为240和110 nM）。 了解更多
  18. VU0364289
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    VU0364289

    Catalog No. A15832
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    mGluR5 Modulator
    VU0364289是新型N-芳基哌嗪mGlu5阳性变构调节剂。 了解更多
  19. VU0652835
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    VU0652835

    Catalog No. A18885
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    mGlu5 modulator
    VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM. 了解更多
  20. TCN238
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    TCN238

    Catalog No. A21191
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    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  21. Lu AF21934
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    Lu AF21934

    Catalog No. A12140
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    mGlu4 receptor modulator
    Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多
  22. (R)-ADX-47273
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    (R)-ADX-47273

    Catalog No. A21887
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    mGluR5 positive allosteric modulator
    (R)-ADX-47273 is a potent mGluR5 positive allosteric modulator, with an EC50 of 168 nM for potentiation . 了解更多
  23. CBiPES HCl
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    CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂，IC50值为98.2 nM。 了解更多
  24. Basimglurant
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    Basimglurant

    Catalog No. A21225
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    mGlu5 negative allosteric modulator
    Basimglurant (RG7090) is a potent, selective and orally available mGlu5 negative allosteric modulator with a Kd of 1.1 nM. 了解更多
  25. CPPHA
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    CPPHA

    Catalog No. A15053
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    mGluR1 modulator
    CPPHA是mGluR5受体的选择性正变构调节剂。 了解更多
  26. BMT-145027
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    BMT-145027

    Catalog No. A12457
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    mGluR5 positive allosteric modulator
    BMT-145027 is an mGluR5 positive allosteric modulator without inherent agonist activity, exhibits an EC50 of 47 nM. 了解更多
  27. PU 02
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    PU 02

    Catalog No. A13757
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    5-HT3 Receptor Modulator
    PU 02是5-HT3受体的负变构调节剂。 了解更多
  28. Vortioxetine (Lu AA21004) hydrobromide
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    Vortioxetine (Lu AA21004) hydrobromide

    Catalog No. A12602
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    5-HT Receptor modulator
    Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物，可抑制5-HT（1A），5-HT（1B），5-HT（3A），5-HT（7）和SERT，IC50为15 nM，33 nM，3.7 nM，19 nM和1.6 nM。 了解更多

28 个项目

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  1. 5-HT Receptors (2)
  2. Metabotropic glutamate receptors (mGluR) (15)
  3. CXCR (1)
  4. Endothelin Receptors (1)
  5. Adenosine Receptors (1)
  6. Cannabinoid Receptors (1)
  7. Neurotensin Receptors (1)
  8. S1P Receptor (3)
  9. Sigma receptor (1)
  10. GLP-1 receptors (2)
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