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SIB 1757
Catalog No. A13758 -
A-841720
Catalog No. A13854 -
MTEP hydrochloride
Catalog No. A15174 -
Dipraglurant
Catalog No. A11382 mGluR5 antagonistsDipraglurant (ADX 48621) is a mGluR5 antagonists with IC50 of 0.021 μM. 了解更多 -
Mavoglurant
Catalog No. A21223 mGlu5 receptor antagonistMavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist, has an IC50 of 30 nM in a functional assay with human mGluR5. 了解更多 -
Mavoglurant racemate
Catalog No. A21799 mGlu5 receptor antagonistMavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. 了解更多 -
Methoxy-PEPy
Catalog No. A21899 mGlu5 receptor antagonistMethoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. 了解更多 -
Alvimopan (ADL 8-2698)
Catalog No. A11292 Opioid 拮抗剂Alvimopan (ADL 8-2698)表现为外周作用的opioid拮抗剂，Alvimopan竞争性结合胃肠道中的mu-opioid receptor。 了解更多 -
Naloxegol Oxalate
Catalog No. A15972 -
BTRX-335140
Catalog No. A18583 κ opioid receptor antagonistBTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. 了解更多 -
Methylnaltrexone Bromide
Catalog No. A15159 -
GSK1521498 free base
Catalog No. A18994 μ-opioid receptor antagonistGSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多 -
GSK1521498 free base (hydrochloride)
Catalog No. A21792 μ-opioid receptor (MOR) antagonistGSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多 -
Amisulpride
Catalog No. A10067 -
Adoprazine (SLV313)
Catalog No. A11297 -
cis-(Z)-Flupentixol dihydrochloride
Catalog No. A12347 Dopamine receptor 拮抗剂cis-(Z)-Flupentixol dihydrochloride是多巴胺受体拮抗剂、抗精神病药物、抗精神病药物。 了解更多 -
SB269652
Catalog No. A14191 -
Metoclopramide HCl
Catalog No. A14247 dopamine D2 receptor 拮抗剂Metoclopramide HCl是一种选择性的多巴胺D2受体拮抗剂。 了解更多 -
SCH 23390 HCl
Catalog No. A13066 -
Prochlorperazine
Catalog No. A16172 -
Alizapride HCl
Catalog No. A16394 -
Azaperone
Catalog No. A16416 -
Melitracen hydrochloride
Catalog No. A17494 dopamine D1/2 receptor antagonistMelitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多 -
Metoclopramide hydrochloride hydrate
Catalog No. A18072 Dopamine D2 antagonistMetoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. 了解更多 -
NRA-0160
Catalog No. A20128 Dopamine D4 receptor antagonistNRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多 -
Cariprazine hydrochloride
Catalog No. A15036 D3/D2 Dopamine Receptor 拮抗剂Cariprazine hydrochloride是一种新型的抗精神病药物，对多巴胺D3（Ki = 0.09 nM）和D2（Ki = 0.5 nM）受体具有高选择性和亲和力，对5-羟色胺5-HT（1A）受体具有中等亲和力。 了解更多 -
Metoclopramide
Catalog No. A15161 -
Veralipride
Catalog No. A13132 D2 receptor antagonistVeralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多 -
Pipamperone
Catalog No. A12621 D2 receptor antagonistPipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7). 了解更多 -
Haloperidol hydrochloride
Catalog No. A18304 dopamine D2 receptor antagonistHaloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多 -
SB-277011 dihydrochloride
Catalog No. A21353 dopamine D3 receptor antagonistSB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多 -
Risperidone hydrochloride
Catalog No. A21458 dopamine D2 receptor antagonistRisperidone hydrochloride is a serotonin 5-HT2 receptor blocker and a potent dopamine D2 receptor antagonist, with Kis of 0.16, 1.4 nM for 5-HT2 and D2 receptor, respectively. 了解更多 -
Risperidone mesylate
Catalog No. A21463 dopamine D2 receptor antagonistRisperidone mesylate(R 64 766 mesylate) is a serotonin 5-HT2 receptor blocker(Ki= 0.16 nM) and a potent dopamine D2 receptor antagonist(Ki= 1.4 nM). 了解更多
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