微信关注
Total item
Cart Subtotal
￥ 0.00 GPCR / G Protein
-
Kynurenic acid
Catalog No. A16581 GPR35/CXCR8 拮抗剂Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多 -
AF64394
Catalog No. A21574 -
(1R,2R)-2-PCCA(hydrochloride)
Catalog No. A21655 GPR88 receptor agonist(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多 -
AMG 837 sodium salt
Catalog No. A21793 GPR40 agonistAMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多 -
Radioprotectin-1
Catalog No. A18628 LPA2 agonistRadioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. 了解更多 -
GRI 977143
Catalog No. A15343 -
GSK726701A
Catalog No. A20101 EP4 partial agonistGSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. 了解更多 -
AGN 210676
Catalog No. A21281 prostaglandin EP2 agonistAGN 210676 is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. 了解更多 -
Treprostinil sodium
Catalog No. A21046 DP1/EP2 agonistTreprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6??0.1 and 6.2??1.2 nM, respectively. 了解更多 -
NS-304 (Selexipag)
Catalog No. A13880 prostacyclin receptor 激动剂NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂（人和大鼠IP受体的Ki值为260和2100 nM，EP1-4，DP，FP和TP受体的Ki值为> 10μM）。 了解更多 -
CP544326 (Taprenepag)
Catalog No. A15853 -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多 -
CGS 21680 HCl Hydrate
Catalog No. A11619 -
2-Chloroadenosine (CADO)
Catalog No. A16105 Adenosine A Receptor 激动剂2-Chloroadenosine (CADO)是腺苷的代谢稳定的类似物，其表现为腺苷A受体激动剂（腺苷A1-R，腺苷A2A-R和腺苷A3-R的Ki值分别为300、80和1900 nM）。 了解更多 -
CGS 21680 HCl
Catalog No. A16441 -
Regadenoson
Catalog No. A12541 A2A adenosine 激动剂Regadenoson是A2A腺苷受体相对于A1，A2B和A3受体的选择性激动剂。还发现Regadenoson是引起冠状动脉血管扩张的完全而有效的激动剂，这种反应具有非常大的A2A受体储备。 了解更多 -
Tecadenoson
Catalog No. A13302 A1 adenosine receptor agonistTecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多 -
Taranabant
Catalog No. A11578 CB1 receptor inverse agonistTaranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多 -
Taranabant ((1R,2R)stereoisomer)
Catalog No. A21705 CB1 receptor inverse agonistTaranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多 -
WIN 55,212-2 mesylate
Catalog No. A11932 CB receptor 激动剂WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多 -
GW842166X
Catalog No. A11253 -
Bay 59-3074
Catalog No. A16328 CB1/CB2 receptor 激动剂Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂，对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多 -
AM1241
Catalog No. A16397 -
Rimonabant hydrochloride
Catalog No. A11548 -
Orexin 2 Receptor Agonist
Catalog No. A15982
FILTER BY:
Filtering:
- 作用机制: Agonist (激动剂) 删除该内容
购物选项
- 分类
-
- 5-HT Receptors (39)
- Adrenergic Receptors (45)
- Histamine Receptors (5)
- Opioid Receptors (15)
- Metabotropic glutamate receptors (mGluR) (14)
- Melatonin Receptors (3)
- Smoothened Receptors (2)
- CXCR (5)
- G Protein (15)
- Endothelin Receptors (1)
- LPA Receptor (2)
- Prostanoid Receptors (6)
- Adenosine Receptors (13)
- Cannabinoid Receptors (12)
- Neurotensin Receptors (1)
- Orexin Receptors (1)
- Neurokinin Receptors (1)
- S1P Receptor (4)
- Sigma receptor (6)
- Guanylate Cyclase (1)
- GHSR (1)
- Imidazoline Receptor (7)
- GLP-1 receptors (6)
- Calcium-Sensing Receptor (2)
- GPCR19 (4)
- 靶点
-
- CXCR4 (1)
ADOOQ 产品质量保证
We promise all products to perform as described.