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GPCR / G Protein

产品 1 到 50 共 229个

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  1. TGR5-Receptor-Agonist
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    TGR5-Receptor-Agonist

    Catalog No. A13732
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    TGR5(GPCR19) 激动剂
    TGR5 Receptor Agonist是一种有效的TGR5（GPCR19）激动剂，在U2-OS细胞分析（pEC50 = 6.8）和黑素细胞（pEC50 = 7.5）中显示出增强的效力。 了解更多
  2. SB756050
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    SB756050

    Catalog No. A12759
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    TGR5 agonist
    SB756050 is a selective TGR5 agonist currently in phase 1clinical trials for the treatment of type 2 diabetes. 了解更多
  3. INT-777
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    INT-777

    Catalog No. A21168
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    TGR5 agonist
    INT-777 is a potent TGR5 agonist with an EC50 of 0.82 μM. 了解更多
  4. INT-767
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    INT-767

    Catalog No. A21494
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    dual FXR/TGR5 agonist
    INT-767 is a dual farnesoid X receptor (FXR)/TGR5 agonist with mean EC50s of 30 and 630 nM, respectively. 了解更多
  5. Strontium ranelate (Protelos)
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    Strontium ranelate (Protelos)

    Catalog No. A11681
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    CaSR 激动剂
    Strontium ranelate是一种抗骨质疏松剂，可增加骨形成并减少骨吸收，从而导致骨转换平衡，有利于骨形成。这类似于胆碱稳定的原硅酸的作用。 了解更多
  6. Evocalcet
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    Evocalcet

    Catalog No. A17003
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    CaSR 激动剂
    Evocalcet是一种钙敏感受体激动剂。钙敏感受体（CaSR）是C类G蛋白偶联受体，可感应细胞外钙离子水平。 了解更多
  7. Lixisenatide
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    Lixisenatide

    Catalog No. A14076
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    GLP-1 receptor 激动剂
    Lixisenatide抑制胰高血糖素释放，显着降低餐后胰高血糖素。对糖尿病（T2DM）有促进作用。 了解更多
  8. BETP
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    BETP

    Catalog No. A13781
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    GLP-1 receptor 激动剂
    BETP是胰高血糖素样肽1（GLP-1）受体的选择性正构构调节剂和部分激动剂。 了解更多
  9. Liraglutide
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    Liraglutide

    Catalog No. A16115
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    GLP-1 receptor 激动剂
    Liraglutide是一种长效胰高血糖素样肽1（GLP-1）受体激动剂。 了解更多
  10. Albiglutide
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    Albiglutide

    Catalog No. A16823
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    GLP-1 激动剂
    Albiglutide是一种胰高血糖素样肽1激动剂（GLP-1激动剂）。 了解更多
  11. Dulaglutide
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    Dulaglutide

    Catalog No. A16987
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    GLP-1 receptor 激动剂
    Dulaglutide是胰高血糖素样肽1（GLP-1）受体激动剂。 了解更多
  12. Semaglutide
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    Semaglutide

    Catalog No. A18908
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    GLP-1 receptor agonist
    Semaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多
  13. Moxonidine HCl
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    Moxonidine HCl

    Catalog No. A11741
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    imidazoline receptor 1 激动剂
    Moxonidine HCl是咪唑啉受体亚型1（I1）的选择性激动剂。Moxonidine引起交感神经系统活动的减少，因此导致血压的降低。 了解更多
  14. Rilmenidine Phosphate
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    Rilmenidine Phosphate

    Catalog No. A14256
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    I(1) imidazoline receptor 激动剂
    Rilmenidine Phosphate是一种选择性的I(1)咪唑啉受体激动剂。 了解更多
  15. Moxonidine Hydrochloride
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    Moxonidine Hydrochloride

    Catalog No. A13416
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    imidazoline receptor 1 激动剂
    Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体（I1-R）选择性激动剂，为降压剂。 了解更多
  16. Capromorelin Tartrate
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    Capromorelin Tartrate

    Catalog No. A21238
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    GHSR agonist
    Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. 了解更多
  17. Linaclotide
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    Linaclotide

    Catalog No. A13834
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    Guanylate cyclase C 激动剂
    Linaclotide是鸟苷酸环化酶2C的肽激动剂。 了解更多
  18. Carbetocin
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    Carbetocin

    Catalog No. A18080
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    peripheral oxytocin receptors agonist
    Carbetocin (Lonactene; Duratocin) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth; an agonist at peripheral oxytocin receptors. 了解更多
  19. Siramesine Hydrochloride
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    Siramesine Hydrochloride

    Catalog No. A12479
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    Sigma-2 receptor 激动剂
    Siramesine Hydrochloride是一种选择性sigma-2受体激动剂，已被证明可触发癌细胞的细胞死亡并在体内表现出强大的抗癌活性。 了解更多
  20. Siramesine
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    Siramesine

    Catalog No. A13036
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    Sigma-2 receptor 激动剂
    Siramesine是一种溶酶体去污剂，诱导细胞保护性自噬体积累。 了解更多
  21. SA-4503
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    SA-4503

    Catalog No. A12984
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    sigma 1 receptor(σ1R) 激动剂
    SA4503是选择性sigma 1受体（σ1R）激动剂；对（+）-[3H]喷他佐辛标记的sigma 1受体亚型具有高亲和力（IC50 = 17.4+/-1.9 nM）；对sigma 2受体的亲和力低100倍。 了解更多
  22. 4-IBP
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    4-IBP

    Catalog No. A12314
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    σ1 激动剂
    4-IBP is a selective ??1 agonist with a high level of affinity for the ??1 receptor (Ki = 1.7 nM) and a moderate affinity for the ??2 receptor (Ki = 25.2 nM) . 了解更多
  23. Cutamesine
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    Cutamesine

    Catalog No. A21152
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    sigma 1 receptor agonist
    Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多
  24. Ditolylguanidine
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    Ditolylguanidine

    Catalog No. A21268
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    Sigma receptor agonist
    Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多
  25. CYM 5442 HCl
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    CYM 5442 HCl

    Catalog No. A13637
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    EDG-1 (S1P1) 激动剂
    CYM 5442 HCl是一种有效的体外选择性EDG-1（S1P1）激动剂（EC50 = 1.35 nM）。 了解更多
  26. ASP1126
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    ASP1126

    Catalog No. A18432
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    S1P agonist
    ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist, with EC50 values of 7.12 nM, 517 nM for hS1P1 and hS1P3, respectively. 了解更多
  27. Cenerimod
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    Cenerimod

    Catalog No. A20913
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    S1P1 agonist
    Cenerimod (ACT-334441) is a potent and orally available sphingosine 1-phosphate 1 receptor (S1P1) agonist extracted from patent WO 2016184939 A1 and WO 2011007324 A1, example 1, with an EC50 of 2.7 nM. 了解更多
  28. FTY720 (S)-Phosphate
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    FTY720 (S)-Phosphate

    Catalog No. A21324
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    S1PR1 agonist
    FTY720 (S)-Phosphate is an agonist of S1P receptor 1 (S1PR1), used in the research of acute inflammatory diseases such as acute lung injury. 了解更多
  29. Senktide
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    Senktide

    Catalog No. A16945
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    NK3 receptor 激动剂
    Senktide是神经介素K3（NK3）受体的有效选择性激动剂（EC50 = 0.5-3 nM）。 了解更多
  30. Orexin 2 Receptor Agonist
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    Orexin 2 Receptor Agonist

    Catalog No. A15982
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    Orexin 2 receptor 激动剂
    Orexin 2 Receptor Agonist一种有效的选择性Orexin2受体激动剂。 了解更多
  31. ML314
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    ML314

    Catalog No. A13570
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    NTR1 激动剂
    ML-314是神经降压素NTR1受体的脑渗透性非肽β-arrestin偏向性激动剂，在主要试验中对NTR1（EC50 = 2.0μM）表现出完全的激动剂行为，对NTR2具有选择性。 了解更多
  32. WIN 55,212-2 mesylate
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    WIN 55,212-2 mesylate

    Catalog No. A11932
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    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多
  33. MDA 19
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    MDA 19

    Catalog No. A11939
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    CB2 激动剂
    MDA 19是CB2的有效选择性激动剂，对精神活性CB1受体具有合理的选择性。 了解更多
  34. GW842166X
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    GW842166X

    Catalog No. A11253
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    CB2 receptor 激动剂
    GW842166X是一种选择性的非大麻类CB2受体激动剂，EC50为63 nM，对CB1受体没有显著的活性。 了解更多
  35. Tedalinab
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    Tedalinab

    Catalog No. A14189
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    CB2 receptor 激动剂
    Tedalinab (GRC-10693)是开发用于治疗骨关节炎和神经性疼痛的药物，它可作为有效的选择性大麻素CB2受体激动剂。与相关的CB1受体相比，它对CB2的选择性为4700x，具有很高的口服生物利用度，并在早期临床试验中显示出令人鼓舞的安全性结果以及有效的镇痛和抗炎作用。 了解更多
  36. Bay 59-3074
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    Bay 59-3074

    Catalog No. A16328
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    CB1/CB2 receptor 激动剂
    Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂，对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多
  37. AM1241
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    AM1241

    Catalog No. A16397
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    CB2 receptor 激动剂
    AM1241是选择性的大麻素CB2受体激动剂，Ki为3.4 nM，相对于CB1受体具有82倍的选择性。 了解更多
  38. Rimonabant hydrochloride
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    Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  39. SR 144528
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    SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  40. VCE-004.8
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    VCE-004.8

    Catalog No. A18549
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    PPARγ and CB2 receptor dual agonist
    VCE-004.8, a semi-synthetic multitarget cannabinoquinoid, is a specific PPARγ and CB2 receptor dual agonist with potent anti-inflammatory activity. 了解更多
  41. CB2R-IN-1
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    CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  42. Taranabant
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    Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  43. Taranabant ((1R,2R)stereoisomer)
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    Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  44. CGS 21680 HCl Hydrate
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    CGS 21680 HCl Hydrate

    Catalog No. A11619
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    Adenosine A2A Receptor 激动剂
    CGS 21680 HCl是一种特定的腺苷A2A亚型受体激动剂。 了解更多
  45. Capadenoson
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    Capadenoson

    Catalog No. A14159
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    Adenosine Receptor 激动剂
    Capadenoson是腺苷A1受体的选择性激动剂。 了解更多
  46. IB-MECA
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    IB-MECA

    Catalog No. A14345
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    Adenosine A3-R 激动剂
    IB-MECA已被证明是一种有效的选择性腺苷A3-R激动剂，腺苷A3-R，腺苷A1-R和腺苷A2A-R的Ki值分别为1.1、54和56 nM。 了解更多
  47. 2-Chloroadenosine (CADO)
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    2-Chloroadenosine (CADO)

    Catalog No. A16105
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    Adenosine A Receptor 激动剂
    2-Chloroadenosine (CADO)是腺苷的代谢稳定的类似物，其表现为腺苷A受体激动剂（腺苷A1-R，腺苷A2A-R和腺苷A3-R的Ki值分别为300、80和1900 nM）。 了解更多
  48. CGS 21680 HCl
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    CGS 21680 HCl

    Catalog No. A16441
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    Adenosine A2 receptor 激动剂
    CGS 21680 HCl是腺苷A2受体激动剂，IC50为22 nM，比A1受体高140倍。 了解更多
  49. Regadenoson
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    Regadenoson

    Catalog No. A12541
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    A2A adenosine 激动剂
    Regadenoson是A2A腺苷受体相对于A1，A2B和A3受体的选择性激动剂。还发现Regadenoson是引起冠状动脉血管扩张的完全而有效的激动剂，这种反应具有非常大的A2A受体储备。 了解更多
  50. NECA
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    NECA

    Catalog No. A16962
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    adenosine receptor 激动剂
    NECA是一种高亲和力的腺苷受体激动剂（human A3，A1和A2A受体的Ki值分别为6.2、14和20 nM；human A2B的EC50 = 2.4 μM）。 了解更多

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