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￥ 0.00 GPCR / G Protein
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Tecadenoson
Catalog No. A13302 A1 adenosine receptor agonistTecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多 -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多 -
NS-304 (Selexipag)
Catalog No. A13880 prostacyclin receptor 激动剂NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂（人和大鼠IP受体的Ki值为260和2100 nM，EP1-4，DP，FP和TP受体的Ki值为> 10μM）。 了解更多 -
CP544326 (Taprenepag)
Catalog No. A15853 -
GSK726701A
Catalog No. A20101 EP4 partial agonistGSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. 了解更多 -
AGN 210676
Catalog No. A21281 prostaglandin EP2 agonistAGN 210676 is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. 了解更多 -
Treprostinil sodium
Catalog No. A21046 DP1/EP2 agonistTreprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6??0.1 and 6.2??1.2 nM, respectively. 了解更多 -
GRI 977143
Catalog No. A15343 -
Radioprotectin-1
Catalog No. A18628 LPA2 agonistRadioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. 了解更多 -
AF64394
Catalog No. A21574 -
(1R,2R)-2-PCCA(hydrochloride)
Catalog No. A21655 GPR88 receptor agonist(1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多 -
AMG 837 sodium salt
Catalog No. A21793 GPR40 agonistAMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多 -
Kynurenic acid
Catalog No. A16581 GPR35/CXCR8 拮抗剂Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多 -
GPR35 agonist 1
Catalog No. A12462 GPR35/CXCR8 agonistGPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability. 了解更多 -
Kynurenic acid sodium
Catalog No. A20000 GPR35/CXCR8 agonistKynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多 -
SAG
Catalog No. A13627 -
SAG hydrochloride
Catalog No. A21678 Smo receptor agonistSAG (hydrochloride) is a potent Smo receptor agonist, and activates the Hedgehog signaling pathway, with a Kd of 59 nM. 了解更多 -
Melatonin
Catalog No. A10564 -
Ramelteon (TAK-375)
Catalog No. A10777 MT1/MT2-Receptor 激动剂Ramelteon (TAK-375)是melatonin受体激动剂，对褪黑激素MT1（IC50 = 28.5±8.55 pM）和MT2（20.1±9.25 pM）受体均具有高亲和力，并且相对于MT3受体具有选择性。 了解更多 -
Tasimelteon
Catalog No. A17351 MT1 and MT2 receptor agonistTasimelteon is a melatonin MT1 and MT2 receptor agonist. 了解更多 -
LY2140023 (LY404039)
Catalog No. A10544 mGluR 激动剂LY-404039是一种用于科学研究的药物，用作代谢型谷氨酸受体II亚型mGluR2和mGluR3的选择性激动剂。它在动物研究中具有抗焦虑和抗精神病作用，但不会引起镇静作用。早期的人体试验使用LY-404，039前药形式LY-214，0023，也取得了令人鼓舞的结果。 了解更多 -
Ibotenic Acid
Catalog No. A14006 NMDA& mGlu receptor 激动剂Ibotenic Acid是最初从鹅膏菌属物种中分离出来的一种神经兴奋性氨基酸，它起着NMDA和代谢型谷氨酸受体激动剂的作用。 了解更多 -
Kainic acid monohydrate
Catalog No. A13485 Kainate receptor 激动剂Kainic acid monohydrate是海藻酸酯类离子型谷氨酸受体激动剂。可在体内诱发癫痫发作和神经退行性变，也已用于在啮齿动物中诱发实验性癫痫和检查兴奋性诱发的神经元凋亡机制。 了解更多 -
(S)-3,5-DHPG
Catalog No. A16108 mGluR 激动剂(S)-3,5-DHPG是I类代谢型谷氨酸受体（mGluRs）的激动剂，与mGluR1a和mGluR5a（分别为Ki = 0.9和3.9 uM）结合，但不与离子型谷氨酸受体结合。 了解更多 -
O-Phospho-L-serine
Catalog No. A21159 group III mGluR receptors agonistO-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2. 了解更多 -
(1R,2S)-VU0155041
Catalog No. A21933 partial mGluR4 agonist(1R,2S)-VU0155041, Cis regioisomer of VU0155041, is a partial mGluR4 agonist with an EC50 of 2.35 μM. 了解更多 -
CHPG sodium salt
Catalog No. A21968 mGluR5 agonistCHPG sodium salt is a selective mGluR5 agonist, and attenuates SO2-induced oxidative stress and inflammation through TSG-6/NF-κB pathway in BV2 microglial cells. 了解更多
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