微信关注
Total item
Cart Subtotal
￥ 0.00 GPCR / G Protein
-
Clonidine hydrochloride
Catalog No. A10232 Alpha adrenergic 激动剂Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。 了解更多 -
Dobutamine hydrochloride
Catalog No. A10325 Adrenoceptors 激动剂Dobutamine hydrochloride是一种直接作用剂，其主要活性来自刺激心脏的β1肾上腺素能受体，增加收缩力和心输出量。 了解更多 -
Carvedilol
Catalog No. A11843 -
Salmeterol
Catalog No. A11788 -
Adrenalone HCl
Catalog No. A11807 -
Arformoterol tartrate
Catalog No. A12795 -
Oxymetazoline hydrochloride
Catalog No. A10686 -
Tetrahydrozoline Hydrochloride
Catalog No. A13080 -
Salmeterol Xinafoate
Catalog No. A14223 -
Bambuterol HCl
Catalog No. A14251 -
Dexmedetomidine HCl
Catalog No. A11846 alpha2-adrenoceptor 激动剂Dexmedetomidine hydrochloride是美托咪啶的活性异构体，它充当有效的，高度选择性的α2-AR（α2-肾上腺素受体）激动剂。 了解更多 -
Medetomidine HCl
Catalog No. A13775 adrenergic alpha-2 receptor 激动剂Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂，Ki为1.08 nM，比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。 了解更多 -
CL 316243 disodium salt
Catalog No. A13657 β3 adrenergic 激动剂CL 316243 disodium salt是一种3β-肾上腺素能激动剂，被开发为一种抗肥胖和糖尿病的药物，并使小鼠的血糖水平迅速下降。 了解更多 -
BRL 37344 Na Salt
Catalog No. A13676 -
Guanabenz acetate
Catalog No. A13635 -
Idazoxan Hydrochloride
Catalog No. A13409 α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多 -
Tulobuterol
Catalog No. A13432 -
UK 14,304 tartrate
Catalog No. A13433 -
Xylazine HCl
Catalog No. A13434 -
(R,R)-Formoterol
Catalog No. A14964 -
Guanfacine hydrochloride
Catalog No. A15098 α2A-adrenoceptor 激动剂Guanfacine hydrochloride是一种抗高血压药，是一种选择性的α2A肾上腺素受体激动剂，Kd为31 nM，选择性是α2B肾上腺素受体的60倍。 了解更多 -
Vilanterol trifenatate
Catalog No. A15998 β2-adrenergic receptor 激动剂Vilanterol trifenatate是一种长效的β-2激动剂药物，于2013年5月与葛兰素氟替卡松合用，获葛兰素史克（Brax Elmitta）出售为Breo Ellipta，用于治疗慢性阻塞性肺疾病（COPD）。 了解更多 -
Brimonidine Tartrate
Catalog No. A15033 α-adrenergic receptor 激动剂Brimonidine Tartrate是一种高度选择性的α-肾上腺素能受体激动剂，对α2A肾上腺素能受体的EC50为0.45 nM。 了解更多 -
Clorprenaline HCl
Catalog No. A16465 -
Vilanterol
Catalog No. A13125 ultra-long-acting β? adrenoreceptor 激动剂Vilanterol是一种新的选择性β2-AR激动剂，PEC50值为10.37±0.05。 了解更多 -
Methoxamine HCl
Catalog No. A17365 alpha-1 adrenergic agonistMethoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction. 了解更多 -
Ractopamine HCl
Catalog No. A17372 beta-Adrenergic agonistRactopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多 -
Midodrine hydrochloride
Catalog No. A17757 Adrenergic alpha-1 agonistMidodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多 -
Brimonidine
Catalog No. A17899 α2-adrenergic receptor agonistBrimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 了解更多 -
Nylidrin Hydrochloride
Catalog No. A17947 beta-adrenergic agonistNylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent. 了解更多 -
Tulobuterol hydrochloride
Catalog No. A18226 β2-adrenergic receptor agonistTulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist. 了解更多 -
Norepinephrine
Catalog No. A11306 β1-selective adrenergic receptor agonistNorepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
AGN 192836
Catalog No. A13013 α2 adrenergic agonistAGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. 了解更多 -
β3-AR agonist 1
Catalog No. A12777 β3-adrenergic receptor agonistβ3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多 -
Norepinephrine hydrochloride
Catalog No. A21605 β1-selective adrenergic receptor agonistNorepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
Mosapride citrate
Catalog No. A10607 -
Tianeptine sodium
Catalog No. A10931 -
BMY 7378
Catalog No. A11208 -
Prucalopride
Catalog No. A11771 5-HT Receptor 激动剂Prucalopride是一种选择性的，高亲和力的5-HT4受体激动剂，作用于5-HT4A和5-HT4B受体，Ki分别为2.5 nM和8 nM，比作用于5-HT受体亚型选择性高290倍以上。 了解更多 -
Clomipramine HCl
Catalog No. A10231 5-HT Receptor 激动剂Clomipramine HCl是下列转运蛋白的阻滞剂：5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM)，去甲肾上腺素转运蛋白（NET）(Ki = 54 nM)，多巴胺转运蛋白（DAT）(Ki = 3，020 nM)，甘氨酸转运蛋白（GlyT/LeuT）。 了解更多 -
Almotriptan malate (Axert)
Catalog No. A11799 5-HT Receptor 激动剂Almotriptan malate (Axert)是一种选择性的5-羟色胺1B/1D（5-HT1B/1D）受体激动剂，用于治疗成人偏头痛。 了解更多 -
Aripiprazole (Abilify)
Catalog No. A11801 5-HT1A receptor 激动剂Aripiprazole (Abilify)是人5-HT1A受体部分激动剂，Ki为4.2 nM。 了解更多 -
Eletriptan hydrobromide
Catalog No. A11418 5-HT1B/1D receptor 激动剂Eletriptan hydrobromide是一种选择性SR-1B/SR-1D激动剂。 了解更多 -
Lorcaserin
Catalog No. A12378
FILTER BY:
Filtering:
- 作用机制: Agonist (激动剂) 删除该内容
购物选项
- 分类
-
- 5-HT Receptors (39)
- Adrenergic Receptors (45)
- Histamine Receptors (5)
- Opioid Receptors (15)
- Metabotropic glutamate receptors (mGluR) (14)
- Melatonin Receptors (3)
- Smoothened Receptors (2)
- CXCR (5)
- G Protein (15)
- Endothelin Receptors (1)
- LPA Receptor (2)
- Prostanoid Receptors (6)
- Adenosine Receptors (13)
- Cannabinoid Receptors (12)
- Neurotensin Receptors (1)
- Orexin Receptors (1)
- Neurokinin Receptors (1)
- S1P Receptor (4)
- Sigma receptor (6)
- Guanylate Cyclase (1)
- GHSR (1)
- Imidazoline Receptor (7)
- GLP-1 receptors (6)
- Calcium-Sensing Receptor (2)
- GPCR19 (4)
- 靶点
-
- CXCR4 (1)
ADOOQ 产品质量保证
We promise all products to perform as described.