微信关注
China
Total item
Cart Subtotal
￥ 0.00 GPCR / G Protein
-
GSK726701A
Catalog No. A20101 EP4 partial agonistGSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. 了解更多 -
CAY10471 Racemate
Catalog No. A11760 Prostaglandin D2 receptor CRTH2 antagonistCAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多 -
ONO-AE3-208
Catalog No. A11516 EP4 antagonistONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. 了解更多 -
(+)-Cloprostenol
Catalog No. A12979 prostaglandin F2α (PGF2α) analogue(+)-Cloprostenol is a prostaglandin F2α (PGF2α) analogue, and shows selective agonistic activity at the prostaglandin receptor. 了解更多 -
MK-2894 sodium salt
Catalog No. A11498 EP4 antagonistMK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多 -
Terutroban
Catalog No. A20884 thromboxane-prostaglandin receptor antagonistTerutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多 -
AGN 210676
Catalog No. A21281 prostaglandin EP2 agonistAGN 210676 is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. 了解更多 -
CJ-42794
Catalog No. A21948 EP4 antagonistCJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多 -
Treprostinil sodium
Catalog No. A21046 DP1/EP2 agonistTreprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6??0.1 and 6.2??1.2 nM, respectively. 了解更多 -
Laropiprant (MK0524)
Catalog No. A11483 DP1 抑制剂Laropiprant (MK0524)与烟酸合用可降低血液胆固醇。是一种有效的，选择性的 DP receptor 拮抗剂，Ki 值为 0.57 nM，对 TP 受体的 Ki 值为 2.95 nM。 了解更多 -
Ozagrel hydrochloride
Catalog No. A11742 Thromboxane A2 synthesis 抑制剂Ozagrel hydrochloride是一种抗血小板剂，用作血栓烷a2合成抑制剂。 了解更多 -
Cloprostenol (sodium salt)
Catalog No. A13498 cloprostenol是前列腺素F2α（PGF2α）的合成类似物。它在仓鼠和大鼠中终止妊娠的效力分别是PGF2α的200倍和100倍，而没有与PGF2α相关的副作用。 了解更多 -
BAY-u 3405
Catalog No. A13751 -
NS-304 (Selexipag)
Catalog No. A13880 prostacyclin receptor 激动剂NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂（人和大鼠IP受体的Ki值为260和2100 nM，EP1-4，DP，FP和TP受体的Ki值为> 10μM）。 了解更多 -
MF498
Catalog No. A15532 -
PF-04418948
Catalog No. A12894 -
CP544326 (Taprenepag)
Catalog No. A15853 -
TG6-10-1
Catalog No. A15968 -
Grapiprant (CJ-023423)
Catalog No. A15964 prostaglandin EP4 receptor 拮抗剂Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型，有效且选择性的前列腺素EP4受体拮抗剂。 了解更多 -
MT-DADMe-ImmA
Catalog No. A13651 human 5'-methylthioadenosine phosphorylase inhibitorMT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM. 了解更多 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
EHNA hydrochloride
Catalog No. A21585 Adenosine deaminase inhibitorEHNA hydrochloride is a specific inhibitor of adenosine deaminase, prevents dAdo degradation and increases mitochondrial dATP levels in fibroblasts. 了解更多 -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多 -
Istradefylline (KW-6002)
Catalog No. A11451 -
SYN-115 (Tozadenant)
Catalog No. A11560 A2a receptor 拮抗剂SYN115是口服，有效和选择性的腺苷2a（A2a）受体抑制剂，作用于人类和恒河猴的 adenosine A2A 受体，Ki 值分别为 11.5 nM 和 6 nM。 了解更多 -
CGS 21680 HCl Hydrate
Catalog No. A11619 -
Aminophylline
Catalog No. A10066 Adenosine receptor 拮抗剂Aminophylline是一种非选择性的腺苷受体拮抗剂和磷酸二酯酶抑制剂，能够逆转局部缺血引起的bradyasystole。 了解更多 -
Dyphylline
Catalog No. A10339 Adenosine receptor 拮抗剂Dyphylline是黄嘌呤衍生物，具有支气管扩张药和血管扩张药的作用。 它充当腺苷受体拮抗剂和磷酸二酯酶抑制剂。 了解更多 -
SCH 442416
Catalog No. A12695 A2A Receptor 拮抗剂SCH 442416是一种选择性的腺苷A2A受体拮抗剂。以高亲和力结合人和大鼠A2A受体（Ki值分别为0.048和0.5 nM）。在体外对hA2A的选择性比hA1高> 23000倍，并且对hA2B和hA3受体的亲和力最小（IC50> 10μM）。 了解更多 -
CVT 6883
Catalog No. A13745 -
5-Iodotubercidin
Catalog No. A13948 Adenosine kinase 抑制剂5-Iodotubercidin是一种有效的腺苷激酶抑制剂，IC50为26 nM。 了解更多
FILTER BY:
购物选项
- 分类
-
- 5-HT Receptors (143)
- Adrenergic Receptors (110)
- Histamine Receptors (62)
- Opioid Receptors (28)
- Metabotropic glutamate receptors (mGluR) (50)
- Melatonin Receptors (4)
- Peptide Receptors (6)
- Smoothened Receptors (14)
- CXCR (30)
- G Protein (26)
- Platelet-Activating Factor (PAF) Receptors (10)
- Endothelin Receptors (21)
- LPA Receptor (13)
- Prostanoid Receptors (28)
- Adenosine Receptors (48)
- Cannabinoid Receptors (26)
- Neurotensin Receptors (4)
- Orexin Receptors (20)
- Somatostatin Receptors (3)
- Neurokinin Receptors (20)
- Protease-Activated Receptors (PAR) (2)
- S1P Receptor (21)
- CGRP Receptor (8)
- Sigma receptor (13)
- Guanylate Cyclase (8)
- cAMP (6)
- GHSR (5)
- Bombesin Receptors (1)
- Imidazoline Receptor (8)
- CCK (6)
- GLP-1 receptors (8)
- Calcium-Sensing Receptor (6)
- GPCR19 (5)
- CRFR (7)
- 作用机制
-
- Inhibitor (抑制剂) (86)
- Agonist (激动剂) (229)
- Antagonist (拮抗剂) (385)
- Activator (激活剂) (12)
- Modulator (调节剂) (28)
- Blocker (阻断剂) (12)
- Stabilizer (稳定剂) (1)
- Stimulator (刺激物) (4)
- 靶点
-
- A1 adenosine receptor (1)
- A3 adenosine receptor (1)
- Aurora A (1)
- Aurora B (1)
- Aurora C (1)
- COX-1 (1)
- COX-2 (1)
- CXCL12 (1)
- CXCL8 (2)
- CXCR1 (4)
- CXCR2 (9)
- CXCR4 (11)
- Histamine H1 receptor (1)
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
ADOOQ 产品质量保证
We promise all products to perform as described.