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GSK221149A (Retosiban)
Catalog No. A13106 Oxytocin Receptor 拮抗剂GSK221149A (Retosiban)是一种口服药物，可作为选择性纳摩尔（Ki = 0.65 nM）催产素受体拮抗剂，其选择性是相关血管加压素受体的> 1400倍。 了解更多 -
Atosiban
Catalog No. A14334 -
PF-3274167
Catalog No. A13754 -
Olinciguat
Catalog No. A13670 guanylate cyclase (sGC) stimulatorOlinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator with concentration-dependent stimulation of sGC in purified rat and human enzyme assays and a whole cell assay. 了解更多 -
Cinaciguat
Catalog No. A21283 sGC activatorCinaciguat is an activator of guanylate cyclase (sGC), and used for acute decompensated heart failure. 了解更多 -
Riociguat (BAY 63-2521)
Catalog No. A11549 -
YC-1 (Lificiguat)
Catalog No. A12402 -
BAY 41-2272
Catalog No. A15891 -
Vericiguat
Catalog No. A21031 guanylate cyclase stimulatorVericiguat (BAY1021189) is a potent, orally available and soluble guanylate cyclase stimulator. 了解更多 -
HJC0350
Catalog No. A14266 -
cAMPS-Sp, triethylammonium salt
Catalog No. A16060 cAMPS-Sp, triethylammonium salt是一种可透过细胞的cAMP类似物，可激活cAMP受体蛋白，例如PKA和cAMP调节的鸟嘌呤核苷酸交换因子。 了解更多 -
SQ22536
Catalog No. A16116 -
Capromorelin Tartrate
Catalog No. A21238 GHSR agonistCapromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. 了解更多 -
Anamorelin HCl
Catalog No. A12345 Anamorelin HCl目前正在开发中，是口服活性的饥饿素受体（ghrelin receptor）激动剂。用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多 -
Anamorelin
Catalog No. A12346 Anamorelin是一种新型 ghrelin receptor激动剂，FLIPR 检测中，EC50 为 0.74 nM，用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多 -
Anamorelin Fumarate
Catalog No. A15000 GHSR stimulatorAnamorelin Fumarate是一种合成的口服活性ghrelin受体激动剂，正在开发中，用于治疗与小肺癌相关的恶病质/厌食症。 了解更多 -
Moxonidine Hydrochloride
Catalog No. A13416 imidazoline receptor 1 激动剂Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体（I1-R）选择性激动剂，为降压剂。 了解更多 -
Moxonidine HCl
Catalog No. A11741 imidazoline receptor 1 激动剂Moxonidine HCl是咪唑啉受体亚型1（I1）的选择性激动剂。Moxonidine引起交感神经系统活动的减少，因此导致血压的降低。 了解更多 -
Rilmenidine Phosphate
Catalog No. A14256 I(1) imidazoline receptor 激动剂Rilmenidine Phosphate是一种选择性的I(1)咪唑啉受体激动剂。 了解更多 -
KU14R
Catalog No. A13987 -
Proglumide
Catalog No. A18171 CCK antagonistProglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. IProglumide is a known cholecystokinin (CCK) antagonist. 了解更多 -
Dexloxiglumide
Catalog No. A18541 CCKA receptor antagonistDexloxiglumide is a selective cholecystokinin type A (CCKA) receptor antagonist. Dexloxiglumide, the active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). 了解更多 -
Loxiglumide (CR1505)
Catalog No. A11769 -
Proglumide sodium salt
Catalog No. A13713 CCK 拮抗剂Proglumide sodium salt是一种非选择性胆囊收缩素（CCK）拮抗剂。它抑制CCK刺激的淀粉酶分泌，并防止CCK诱导的小鼠胰腺腺泡中的2-脱氧葡萄糖摄取。 了解更多 -
Z-360 calcium salt (Nastorazepide calcium salt)
Catalog No. A13671 CCK-2 receptor 拮抗剂Z-360 calcium salt (Nastorazepide calcium salt)是一种选择性口服可口服的1,5-苯并二氮杂卓衍生物胃泌素/胆囊收缩素2（CCK-2）受体拮抗剂，具有潜在的抗肿瘤活性。 了解更多 -
Nastorazepide (Z-360)
Catalog No. A15984 CCK-2 receptor 拮抗剂Nastorazepide (Z-360) 是一种选择性的，口服的1,5-苯二氮杂卓衍生物胃泌素/胆囊收缩素2（CCK-2）受体拮抗剂，具有潜在的抗肿瘤活性。 了解更多 -
Semaglutide
Catalog No. A18908 GLP-1 receptor agonistSemaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多 -
Lixisenatide
Catalog No. A14076 -
BETP
Catalog No. A13781 -
Liraglutide
Catalog No. A16115 -
Albiglutide
Catalog No. A16823 -
Dulaglutide
Catalog No. A16987 -
NPS-2143 hydrochloride
Catalog No. A11505 CaSR antagonistNPS-2143 hydrochloride (SB-262470A hydrochloride), an orally active calcilytic agent, is a selective and potent calcium ion-sensing receptor (CaSR) antagonist. 了解更多 -
NPS-2143 (SB-262470)
Catalog No. A11140 CaSR 拮抗剂NPS-2143 (SB-262470)是一种选择性的Ca2+感应受体拮抗剂，显示可阻止HEK293细胞中表达的人Ca2+受体引起的细胞质Ca2+浓度增加，IC50为43 nM。 了解更多 -
AMG-073 HCl (Cinacalcet HCl)
Catalog No. A10219 CaSR activatorAMG-073 HCl（Cinacalcet HCl）是一种用于治疗甲状旁腺功能亢进的化合物，称为拟钙剂，通过增加甲状旁腺钙敏感受体（CaR）对细胞外钙的敏感性来减少甲状旁腺激素（PTH）的合成和分泌 。 了解更多 -
Strontium ranelate (Protelos)
Catalog No. A11681 CaSR 激动剂Strontium ranelate是一种抗骨质疏松剂，可增加骨形成并减少骨吸收，从而导致骨转换平衡，有利于骨形成。这类似于胆碱稳定的原硅酸的作用。 了解更多 -
AMG 073 (Cinacalcet)
Catalog No. A11314 -
Evocalcet
Catalog No. A17003 -
INT-777
Catalog No. A21168
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