GPCR / G Protein
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TGR5-Receptor-Agonist
Catalog No. A13732 TGR5(GPCR19) 激动剂TGR5 Receptor Agonist是一种有效的TGR5(GPCR19)激动剂,在U2-OS细胞分析(pEC50 = 6.8)和黑素细胞(pEC50 = 7.5)中显示出增强的效力。 了解更多 -
Verucerfont
Catalog No. A16950 CRF-1 拮抗剂Verucerfont,也称为GSK561679和NBI77860,是CRF-1拮抗剂。Verucerfont阻止CRH-1受体,因此减少了慢性应激后ACTH的释放。 了解更多 -
Emicerfont
Catalog No. A14047 -
Pexacerfont
Catalog No. A14105 CRF1 receptor antagonistPexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多