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Amineptine
Catalog No. A14998 Amineptine是一种三环抗抑郁药物，可选择性地阻断3H-imipramine结合，吸收多巴胺，并结合临床状态的变化对主要抑郁症患者的血小板进行了研究。 了解更多 -
SCH 23390 HCl
Catalog No. A13066 -
C-DIM12
Catalog No. A15936 -
ACR 16 hydrochloride
Catalog No. A16074 dopaminergic stabilizerACR 16 hydrochloride是一种多巴胺能稳定剂（对于D2（低）和D2（高），Ki值分别为17550 nM和7521），通过功能性多巴胺D2受体拮抗作用和皮质谷氨酸功能的双重作用，稳定地稳定精神运动活动。在各种情况下神经传递受到干扰。 了解更多 -
UNC 9994 hydrochloride
Catalog No. A16087 dopamine D2 receptor 激动剂UNC 9994 hydrochloride，独特的，β-arrestin偏向的功能选择性多巴胺D2受体（D2R）激动剂（Ki值为30 nM；在ε-arrestin-2募集试验中EC50值为50 nM），在体内具有抗精神病活性。UNC9994在野生型小鼠中显着抑制了PCP诱导的超运动，而在Δr-arrestin-2基因敲除小鼠中这种作用被完全消除。 了解更多 -
Prochlorperazine
Catalog No. A16172 -
Alizapride HCl
Catalog No. A16394 -
Azaperone
Catalog No. A16416 -
Melitracen hydrochloride
Catalog No. A17494 dopamine D1/2 receptor antagonistMelitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多 -
Metoclopramide hydrochloride hydrate
Catalog No. A18072 Dopamine D2 antagonistMetoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. 了解更多 -
NRA-0160
Catalog No. A20128 Dopamine D4 receptor antagonistNRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多 -
Dicarbine
Catalog No. A18925 Dopamine receptor blockerDicarbine blocks dopamine receptors in various brain parts and prevents the depression of the conditioned defence reflexes caused by stimulation of the mesencephalic portion of the reticular formation. Dicarbine could be used to treat patients with schizophrenia and alcoholic psychosis in clinical. 了解更多 -
Nepicastat (free base) (SYN-117)
Catalog No. A10637 dopamine beta-hydroxylase 抑制剂Nepicastat (free base) (SYN-117)是多巴胺β-羟化酶的抑制剂，该酶催化多巴胺向去甲肾上腺素的转化。 了解更多 -
Nalmefene hydrochloride
Catalog No. A13843 dopamine receptor 激动剂Nalmefene hydrochloride是opioid receptor拮抗剂。 了解更多 -
Cariprazine hydrochloride
Catalog No. A15036 D3/D2 Dopamine Receptor 拮抗剂Cariprazine hydrochloride是一种新型的抗精神病药物，对多巴胺D3（Ki = 0.09 nM）和D2（Ki = 0.5 nM）受体具有高选择性和亲和力，对5-羟色胺5-HT（1A）受体具有中等亲和力。 了解更多 -
Metoclopramide
Catalog No. A15161 -
Phenylpiracetam
Catalog No. A15211 -
SKF38393 HCl
Catalog No. A15839 -
Loxapine Succinate
Catalog No. A17347 D2DR and D4DR inhibitorLoxapine Succinate is a D2DR and D4DR inhibitor and serotonergic receptor antagonist. Loxapine succinate is an antipsychotic agent used in schizophrenia. 了解更多 -
Promazine hydrochloride
Catalog No. A17638 D2DR inhibitorPromazine Hydrochloride is a phenothiazine compound and D2DR inhibitor. Promazine Hydrochloride has been employed in studies investigating dopamine-stimulated glycosylation of brain proteins in vitro. It has actions similar to chlorpromazine but with less antipsychotic activity. 了解更多 -
PF-06256142
Catalog No. A18872 D1 receptor agonistPF-06256142 is a potent and selective orthosteric agonist of the D1 receptor, with D1 EC50=30 nM and D1 binding Ki = 12 nM. 了解更多 -
Zamicastat
Catalog No. A13672 dopamine β-hydroxylase (DBH) inhibitorZamicastat (BIA 5-1058) is a dopamine β-hydroxylase (DBH) inhibitor that could cross the blood-brain barrier (BBB) and cause central as well as peripheral effects. 了解更多 -
Veralipride
Catalog No. A13132 D2 receptor antagonistVeralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多 -
Pipamperone
Catalog No. A12621 D2 receptor antagonistPipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7). 了解更多 -
SPD-473 citrate
Catalog No. A12617 serotonin/dopamine/norepinephrine reuptake inhibitiorSPD-473 citrate is a serotonin/dopamine/norepinephrine reuptake inhibitior. 了解更多 -
Pentiapine
Catalog No. A12512 -
Trimethobenzamide hydrochloride
Catalog No. A17648 D2 receptor blockerTrimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多 -
Quinagolide hydrochloride
Catalog No. A18038 dopamine D2 receptor agonistQuinagolide hydrochloride is a selective dopamine D2 receptor agonist, also is a prolactin inhibitor. 了解更多 -
Haloperidol hydrochloride
Catalog No. A18304 dopamine D2 receptor antagonistHaloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多 -
SB-277011 dihydrochloride
Catalog No. A21353 dopamine D3 receptor antagonistSB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多 -
Risperidone hydrochloride
Catalog No. A21458 dopamine D2 receptor antagonistRisperidone hydrochloride is a serotonin 5-HT2 receptor blocker and a potent dopamine D2 receptor antagonist, with Kis of 0.16, 1.4 nM for 5-HT2 and D2 receptor, respectively. 了解更多 -
Risperidone mesylate
Catalog No. A21463 dopamine D2 receptor antagonistRisperidone mesylate(R 64 766 mesylate) is a serotonin 5-HT2 receptor blocker(Ki= 0.16 nM) and a potent dopamine D2 receptor antagonist(Ki= 1.4 nM). 了解更多 -
JNJ-37822681 dihydrochloride
Catalog No. A21470 dopamine D2 receptor antagonistJNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多 -
Pardoprunox hydrochloride
Catalog No. A21624 partial dopamine D2 and D3 receptor agonistPardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist. 了解更多 -
SKF-82958 hydrobromide
Catalog No. A21763 D1/D5 receptor full agonistSKF-82958 hydrobromide is a D1/D5 receptor full agonist. 了解更多 -
Vanoxerine
Catalog No. A21922 dopamine reuptake inhibitorVanoxerine (GBR-12909) is a competitive, potent, and highly selective dopamine reuptake inhibitor (Ki=1 nM). 了解更多 -
Dihydrexidine
Catalog No. A21949 D1-like dopamine receptor (D1/D5) agonistDihydrexidine (DAR-0100) is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist with an IC50 of 10 nM for D1 receptor. Dihydrexidine exhibits potent antiparkinsonian activity. 了解更多 -
Haloperidol D4
Catalog No. A21961 dopamine D2 receptor antagonistHaloperidol D4 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
Haloperidol D4'
Catalog No. A21971 dopamine D2 receptor antagonistHaloperidol D4' is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
Ro 10-5824 dihydrochloride
Catalog No. A21986 dopamine D4 receptor partial agonistRo 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多 -
Amisulpride hydrochloride
Catalog No. A21994 dopamine D2/D3 receptor antagonistAmisulpride hydrochloride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. 了解更多
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