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GPCR / G Protein

28 个项目

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  1. VU0453379
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    VU0453379

    Catalog No. A18796
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    GLP-1R modulator
    VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM. 了解更多
  2. NNC0640
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    NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多
  3. E1R
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    E1R

    Catalog No. A18825
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    sigma-1 receptors modulator
    E1R is a novel positive allosteric modulator of sigma-1 receptors. 了解更多
  4. NS13001
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    NS13001

    Catalog No. A15833
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    SK2 modulator
    NS13001是选择性的SK2/3调节剂，可作为治疗SCA2和其他可能的小脑共济失调的潜在治疗剂。 了解更多
  5. Ponesimod
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    Ponesimod

    Catalog No. A13307
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    S1P1 receptor modulator
    Ponesimod是一种口服活性，选择性鞘氨醇-1-磷酸受体1（S1P1）免疫调节剂，EC50为5.7 nM。 了解更多
  6. RPC1063 (Ozanimod)
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    RPC1063 (Ozanimod)

    Catalog No. A15819
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    S1PR1 modulators
    RPC1063 (Ozanimod)是选择性的鞘氨醇1磷酸酯受体调节剂和方法，可用于治疗与S1P1-β相关的疾病。 了解更多
  7. SBI-553
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    SBI-553

    Catalog No. A18435
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    NTR1 allosteric modulator
    SBI-553 is a potent and brain penetrant NTR1 allosteric modulator. 了解更多
  8. Org 27569
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    Org 27569

    Catalog No. A11513
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    CB1 modulator?
    Org 27569是一种强效CB1受体变构调节剂(PEC50 = 8.24)。 了解更多
  9. LUF6000
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    LUF6000

    Catalog No. A21532
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    A3 adenosine receptor allosteric modulator
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). 了解更多
  10. Endothelin Mordulator 1
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    Endothelin Mordulator 1

    Catalog No. A13040
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    endothelin receptor modulator
    Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多
  11. NSC-23026
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    NSC-23026

    Catalog No. A17151
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    CXCR4 receptor modulator
    NSC-23026是CXCR4受体调节剂。 了解更多
  12. ADX-47273
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    ADX-47273

    Catalog No. A11181
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    mGluR5 modulator
    ADX-47273是一种有效的，特异性的mGlu5正变构调节剂(PAM)EC50为0.17 μM，对其他亚型没有作用活性。 了解更多
  13. VU 0364439
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    VU 0364439

    Catalog No. A12664
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    GluR modulator
    VU 0364439是mGlu4受体的正变构调节剂（PAM）（对于人mGlu4，体外EC50 = 19.8 nM）。 了解更多
  14. BINA
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    BINA

    Catalog No. A11126
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    mGluR2 modulator
    BINA是mGlu2的选择性正构构调节剂（在表达人mGlu2的CHO细胞中EC50 = 33.2 nM）。 了解更多
  15. VU 0361737
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    VU 0361737

    Catalog No. A12467
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    mGlu4 receptors modulator
    VU 0361737是mGluR-4的选择性正变构调节剂（人和大鼠受体的EC50值分别为240和110 nM）。 了解更多
  16. VU0364289
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    VU0364289

    Catalog No. A15832
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    mGluR5 Modulator
    VU0364289是新型N-芳基哌嗪mGlu5阳性变构调节剂。 了解更多
  17. VU0652835
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    VU0652835

    Catalog No. A18885
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    mGlu5 modulator
    VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM. 了解更多
  18. VU 0364770
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    VU 0364770

    Catalog No. A12139
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    mGlu4 receptors modulator
    VU 0364770是mGlu4受体的正变构调节剂，在表达mGlu4的HEK 293细胞中EC50值为290 nM。 了解更多
  19. JNJ 42153605
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    JNJ 42153605

    Catalog No. A14330
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    mGluR-2 modulator
    JNJ-42153605是亲代谢型谷氨酸2受体的正变构调节剂。 了解更多
  20. Lu AF21934
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    Lu AF21934

    Catalog No. A12140
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    mGlu4 receptor modulator
    Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多
  21. (R)-ADX-47273
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    (R)-ADX-47273

    Catalog No. A21887
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    mGluR5 positive allosteric modulator
    (R)-ADX-47273 is a potent mGluR5 positive allosteric modulator, with an EC50 of 168 nM for potentiation . 了解更多
  22. CBiPES HCl
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    CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂，IC50值为98.2 nM。 了解更多
  23. Basimglurant
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    Basimglurant

    Catalog No. A21225
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    mGlu5 negative allosteric modulator
    Basimglurant (RG7090) is a potent, selective and orally available mGlu5 negative allosteric modulator with a Kd of 1.1 nM. 了解更多
  24. CPPHA
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    CPPHA

    Catalog No. A15053
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    mGluR1 modulator
    CPPHA是mGluR5受体的选择性正变构调节剂。 了解更多
  25. BMT-145027
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    BMT-145027

    Catalog No. A12457
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    mGluR5 positive allosteric modulator
    BMT-145027 is an mGluR5 positive allosteric modulator without inherent agonist activity, exhibits an EC50 of 47 nM. 了解更多
  26. TCN238
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    TCN238

    Catalog No. A21191
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    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  27. PU 02
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    PU 02

    Catalog No. A13757
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    5-HT3 Receptor Modulator
    PU 02是5-HT3受体的负变构调节剂。 了解更多
  28. Vortioxetine (Lu AA21004) hydrobromide
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    Vortioxetine (Lu AA21004) hydrobromide

    Catalog No. A12602
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    5-HT Receptor modulator
    Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物，可抑制5-HT（1A），5-HT（1B），5-HT（3A），5-HT（7）和SERT，IC50为15 nM，33 nM，3.7 nM，19 nM和1.6 nM。 了解更多

28 个项目

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  1. 5-HT Receptors (2)
  2. Metabotropic glutamate receptors (mGluR) (15)
  3. CXCR (1)
  4. Endothelin Receptors (1)
  5. Adenosine Receptors (1)
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  8. S1P Receptor (3)
  9. Sigma receptor (1)
  10. GLP-1 receptors (2)
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