AMPA receptor
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Becampanel
Catalog No. A21194 AMPA antagonistBecampanel (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. 了解更多 -
(S)-Willardiine
Catalog No. A21957 AMPA/kainate receptors agonist(S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. 了解更多 -
GYKI53655 Hydrochloride
Catalog No. A17032 -
CNQX disodium salt
Catalog No. A16110 -
Cyclothiazide
Catalog No. A13700 AMPA desensitization 抑制剂Cyclothiazide是苯并噻二叠氮,可作为AMPA受体的增效剂,正向调节其对谷氨酸的响应(EC50 = 3.8 M)。 了解更多 -
Aniracetam
Catalog No. A10078 -
Ampalex (CX-516)
Catalog No. A12349 Ampalex (CX-516)是ampakine和nootropic,充当ampa受体阳性变构调节剂。 了解更多 -
GYKI-52466 dihydrochloride
Catalog No. A10444 AMPA and Kainate 拮抗剂GYKI-52466 dihydrochloride是选择性非竞争性AMPA受体拮抗剂(对于AMPA、红藻氨酸和AMPA诱导的反应,IC50值分别为10-20、~ 450和> > 50 μM)。 了解更多 -
Farampator
Catalog No. A13798 -
IEM 1754 Dihydrobromide
Catalog No. A14010 -
CP 465022 hydrochloride
Catalog No. A13321 AMPA 拮抗剂CP 465022 hydrochloride是一种选择性的非竞争性AMPA拮抗剂,在大鼠皮质神经元中的IC50为25 nM,显示出有效的抗惊厥活性。 了解更多 -
Tezampanel
Catalog No. A15259 -
YM90K hydrochloride
Catalog No. A15495 AMPA 拮抗剂YM90K hydrochloride是一种选择性AMPA受体拮抗剂,在局部缺血后给药后,可延迟整体缺血模型中的神经元死亡和局部缺血模型中的脑梗塞。 了解更多 -
Philanthotoxin 74 dihydrochloride
Catalog No. A21739 AMPAR antagonistPhilanthotoxin 74 dihydrochloride (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. 了解更多 -
Mibampator
Catalog No. A21717 AMPA receptors potentiatorMibampator (LY451395) is a potent and highly selective potentiator of the AMPA receptors. 了解更多 -
Fanapanel hydrate
Catalog No. A21668 AMPA/kainate antagonistFanapanel hydrate (ZK200775 hydrate) is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively. 了解更多 -
Naspm trihydrochloride
Catalog No. A21437 CP-AMPA receptors antagonistNaspm trihydrochloride (1-Naphthylacetyl spermine trihydrochloride), a synthetic analogue of Joro spider toxin, is a calcium permeable AMPA (CP-AMPA) receptors antagonist. 了解更多 -
(S)-(-)-5-Fluorowillardiine
Catalog No. A21337 -
PF-4778574
Catalog No. A21157 AMPA receptor positive allosteric modulatorPF-4778574 is a potent AMPA receptor positive allosteric modulator (PAM) that has been shown to enhance cognition in animal models. 了解更多 -
JNJ-61432059
Catalog No. A20209 AMPAR negative modulatorJNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8, with a pIC50 of 9.7 for GluA1/γ-8. 了解更多 -
Talampanel
Catalog No. A15515