AZD9496 maleate

Name: AZD9496 maleate
SKU: A21726

目录号: A21726

estrogen receptor (ERα) antagonist

AZD9496 maleate Chemical Structure

CAS NO. 1639042-28-6

AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD).

库存：现货

规格	价格	数量
2 mg	￥ 602.00
5 mg	￥ 1,211.00
10 mg	￥ 2,352.00
50 mg	￥ 6,923.00

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生物活性

AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD).

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.9 mL	89.52 mL	179.04 mL
0.5 mM	3.58 mL	17.9 mL	35.81 mL
1 mM	1.79 mL	8.95 mL	17.9 mL
5 mM	0.36 mL	1.79 mL	3.58 mL

*The above data is based on the productmolecular weight 558.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A21726
作用机制	Antagonist (拮抗剂)
M. Wt	558.55
Formula	C29H29F3N2O6
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1639042-28-6
Synonyms	AZD 9496, AZD-9496
SMILES	O=C(O)/C=C/C1=CC(F)=C([C@H]2N(CC(C)(F)C)[C@H](C)CC3=C2NC4=C3C=CC=C4)C(F)=C1.O=C(O)/C=C\C(O)=O