Azilsartan (TAK-536)

Name: Azilsartan (TAK-536)
SKU: A11775

目录号: A11775

AT1 Receptor Blocker

Azilsartan (TAK-536) Chemical Structure

CAS NO. 147403-03-0

Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。

库存：现货

规格	价格	数量
10 mg	￥ 350.00
25 mg	￥ 560.00
50 mg	￥ 700.00
100 mg	￥ 910.00
10mM * 1mL in DMSO	￥ 350.00

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生物活性

Azilsartan (TAK-536)是一种用于治疗高血压的血管紧张素II受体拮抗剂。

靶点信息

AT1 receptor
2.6 nM

溶解度 *

In vitro (25°C)	DMSO	78 mg/mL (170.88 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	30% PEG400+0.5% Tween80+5% propylene glycol	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.91 mL	109.53 mL	219.06 mL
0.5 mM	4.38 mL	21.91 mL	43.81 mL
1 mM	2.19 mL	10.95 mL	21.91 mL
5 mM	0.44 mL	2.19 mL	4.38 mL

*The above data is based on the productmolecular weight 456.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11775
作用机制	Blocker (阻断剂)
M. Wt	456.5
Formula	C25H20N4O5
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	147403-03-0
Synonyms	TAK536
SMILES	CCOC1=NC2=CC=CC(=C2N1CC3=CC=C(C=C3)C4=CC=CC=C4C5=NC(=O)ON5)C(=O)O