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Belinostat (PXD101)

Belinostat (PXD101)

Name: Belinostat (PXD101)
SKU: A10122

目录号: A10122

HDAC 抑制剂

Product Citations (1)

Belinostat (PXD101) Chemical Structure

CAS NO. 414864-00-9

Belinostat（PXD101）是一种HDAC抑制剂，可抑制HeLa细胞提取物中的HDAC活性，IC50为27 nM。

库存：现货

规格	价格	数量
10 mg	￥ 420.00
50 mg	￥ 1,400.00
100 mg	￥ 2,100.00
200 mg	￥ 3,500.00
10mM * 1mL in DMSO	￥ 546.00

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生物活性

Belinostat（PXD101）是一种HDAC抑制剂，可抑制HeLa细胞提取物中的HDAC活性，IC50为27 nM。

靶点信息

HDAC (Cell-free assay)
27 nM

溶解度 *

In vitro (25°C)	DMSO	56 mg/mL (175.9 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	2% DMSO+30% PEG 300+ddH2O	9 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	31.41 mL	157.04 mL	314.07 mL
0.5 mM	6.28 mL	31.41 mL	62.81 mL
1 mM	3.14 mL	15.7 mL	31.41 mL
5 mM	0.63 mL	3.14 mL	6.28 mL

*The above data is based on the productmolecular weight 318.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10122
作用机制	Inhibitor (抑制剂)
M. Wt	318.4
Formula	C15H14N2O4S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	414864-00-9
Synonyms	PX105684
SMILES	C1=CC=C(C=C1)NS(=O)(=O)C2=CC=CC(=C2)/C=C/C(=O)NO