“bsj 03 123”的搜索结果

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  1. BSJ-03-123

    Catalog No. A22336
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    CDK6-selective small-molecule degrader
    BSJ-03-123 is a potent and novel CDK6-selective small-molecule degrader (PROTAC). 了解更多
  2. Dihydrorhodamine 123

    Catalog No. A19716
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    fluorescent probe
    Dihydrorhodamine 123 is a fluorescent probe (λex=488 nm, λem=525 nm). 了解更多
  3. BQ-123

    Catalog No. A15912
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    ETA receptor 拮抗剂
    BQ-123是一种选择性内皮素A受体(ETA)拮抗剂,IC50为7.3 nM。 了解更多
  4. BAY1238097

    Catalog No. A16881
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    BET 抑制剂
    BAY1238097是一种有效的选择性BET抑制剂。BAY1238097与BET蛋白BRD上的乙酰化赖氨酸识别基序结合,从而防止BET蛋白与组蛋白之间的相互作用。 了解更多
  5. LSD1-IN-6

    Catalog No. A20474
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    LSD1 inhibitor
    LSD1-IN-6 (Compound 4m) is a potent and reversible inhibitor of lysine-specific demethylase 1 (LSD1), with an IC50 of 123 nM. LSD1-IN-6 increases dimethylated Lys4 of histone H3, shows no effect on expression of LSD1. 了解更多
  6. D-erythro-Sphingosine

    Catalog No. A12304
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    p32-kinase activator
    D-erythro-Sphingosine (Erythrosphingosine) is a very potent activator of p32-kinase with an EC50 of 8 μM, and inhibits protein kinase C (PKC). D-erythro-Sphingosine (Erythrosphingosine) is also a PP2A activator. 了解更多
  7. 4-Aminophenol

    Catalog No. A17667
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    4-Aminophenol was commonly used as a developer for black-and-white film, marketed under the name Rodinal. 了解更多
  8. CDC123 Human

    Catalog No. AP0672
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    Cell Division Cycle 123 Human Recombinant 了解更多
  9. Cetylpyridinium Chloride

    Catalog No. A16439
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    Cetylpyridinium Chloride是用作口咽防腐剂的阳离子季铵化合物。 了解更多
  10. 2-Aminoheptane

    Catalog No. A16383
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    2-Aminoheptane是一种鼻减充血药,是一种拟交感神经兴奋剂和血管收缩药。 了解更多
  11. Azelaic acid

    Catalog No. A16150
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    Azelaic acid是通过油酸的臭氧分解产生的有机化合物。头发和皮肤调理剂的成分。 了解更多
  12. 6-Diazo-5-oxo-L-nor-Leucine

    Catalog No. A20846
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    6-Diazo-5-oxo-L-norleucine 是一种从链霉菌中分离出来的抗生素,一种 glutaminase 的拮抗剂对cKGA(肾脏型谷氨酰胺酶)的IC50值约为1 mM。 了解更多
  13. Auranofin

    Catalog No. A18996
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    Auranofin is a gold salt classified by the World Health Organization as an antirheumatic agent. It is a gold-thiol complex with anti-inflammatory and immunosuppressive actions. 了解更多
  14. Angiotensin III

    Catalog No. A18943
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    angiotensin 1 (AT1) and AT2 receptor agonist
    Angiotensin III is an angiotensin 1 (AT1) and AT2 receptor agonist. 了解更多
  15. Pertussis Toxin

    Catalog No. A19356
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    protein-based AB5-type exotoxin
    Pertussis Toxin is a protein-based AB5-type exotoxin produced by the bacterium Bordetella pertussis, which causes whooping cough. 了解更多
  16. Lignine

    Catalog No. A20324
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    Lignine (Lignin) is a complex organic polymer, which plays an important role in plant cell wall structure. 了解更多
  17. Chitosan oligosaccharide

    Catalog No. A20304
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    Chitosan oligosaccharide (COS) is an oligomer of β-(1??4)-linked D-glucosamine. Chitosan oligosaccharide (COS) activates AMPK and inhibits inflammatory signaling pathways including NF-κB and MAPK pathways. 了解更多
  18. Avelumab

    Catalog No. A18234
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    PD-1/PD-L1
    Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody with potential antibody-dependent cell-mediated cytotoxicity. 了解更多
  19. BMS-1001

    Catalog No. A22061
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    PD-1/PD-L1 interaction inhibitor
    BMS-1001 is a potent inhibitor of PD-1/PD-L1 interaction with EC50 of 253 nM. 了解更多
  20. 9-ING-41

    Catalog No. A22066
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    glycogen synthase kinase-3β (GSK-3β) inhibitor
    9-ING-41 is a maleimide-based ATP-competitive and selective glycogen synthase kinase-3β (GSK-3β) inhibitor with an IC50 of 0.71 μM. 了解更多
  21. BAY 2416964

    Catalog No. A22067
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    aryl hydrocarbon receptor (AHR) antagonist
    BAY 2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 192, has an IC50 of 341 nM. BAY 2416964 has the potential for solid tumors treatment. 了解更多
  22. CYM50308

    Catalog No. A22072
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    sphingosine-1-phosphate receptor 4 (S1P4-R) agonist
    CYM50308 (ML248) is a potent, selective and high affinity sphingosine-1-phosphate receptor 4 (S1P4-R) agonist with an EC50 of 56 nM. 了解更多
  23. ASN03576800

    Catalog No. A22080
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    ASN03576800 is an inhibitor of the VP40 matrix protein. 了解更多
  24. BMS453

    Catalog No. A22082
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    RARβ agonist
    BMS453 (BMS-189453), a synthetic retinoid, is a RARβ agonist and a RARα/RARγ antagonist. 了解更多
  25. CYM 2503

    Catalog No. A22092
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    positive allosteric modulator (PAM)
    CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. 了解更多
  26. RBC10

    Catalog No. A22098
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    inhibitor of Ral binding to RALBP1
    RBC10 is an inhibitor of Ral binding to RALBP1 (the effector). 了解更多
  27. NIBR-0213

    Catalog No. A22099
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    S1P(1) antagonist
    NIBR-0213 is a potent and selective antagonist of S1P(1) with efficacy in experimental autoimmune encephalomyelitis. 了解更多
  28. PD-089828

    Catalog No. A22103
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    ATP competitive inhibitor of FGFR-1, PDGFR-β and EGFR
    PD089828 is an ATP competitive inhibitor of FGFR-1, PDGFR-β and EGFR with IC50 of 0.15 ?M, 1.76 ?M, and 5.47 ?M, respectively. 了解更多
  29. AEM1

    Catalog No. A22108
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    inhibitor of deregulated NRF2 transcriptional activity
    AEM1 is an inhibitor of deregulated NRF2 transcriptional activity in cancer. 了解更多
  30. RO5203648 hydrochloride

    Catalog No. A22118
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    partial agonist of Trace amine-associated receptor 1
    RO5203648 hydrochloride is a partial agonist of Trace amine-associated receptor 1 (TAAR1). 了解更多
  31. R243

    Catalog No. A22123
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    inhibitor of CCR8 signaling and chemotaxis
    R243 is an inhibitor of CCR8 signaling and chemotaxis. 了解更多
  32. MN58b

    Catalog No. A22129
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    choline kinase α (CHKα) inhibitor
    MN58b is a selective choline kinase α (CHKα) inhibitor, and results in inhibition of phosphocholine synthesis. 了解更多
  33. ASLAN003

    Catalog No. A22140
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    Dihydroorotate Dehydrogenase (DHODH) inhibitor
    ASLAN003 is an orally active and potent Dihydroorotate Dehydrogenase (DHODH) inhibitor with an IC50 of 35 nM for human DHODH enzyme. 了解更多
  34. Takeda103A

    Catalog No. A22142
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    bovine tubulin oxidation inhibitor
    Takeda103A is a potent GRK2-dependent bovine tubulin oxidation inhibitor. 了解更多
  35. Soporidine

    Catalog No. A22145
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    strigolactone (SL) antagonist
    Soporidine is a strigolactone (SL) antagonist and inhibitor of germination in their biological assays. It binds AtHTL and specifically interferes with SL signaling. 了解更多
  36. Aka Lumine

    Catalog No. A22152
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    luciferin analogue
    Aka Lumine, a luciferin analogue, is a luciferase substrate emitting red, green, and blue light. The longest emission wavelength of Aka Lumine is recorded at 675 nm, which is within the NIR region. 了解更多
  37. Prexasertib HCl

    Catalog No. A22156
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    ATP-competitive CHK1 inhibitor
    Prexasertib (LY2606368) is an ATP-competitive CHK1 inhibitor with a Ki value of 0.9 nmol/L. For CHK2 and RSK, its IC50 values are 8 nM and 9 nM respectively in cell-free assay. 了解更多
  38. iFSP1

    Catalog No. A22277
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    glutathione-independent inhibitor
    iFSP1 is a potent, selective and glutathione-independent inhibitor of ferroptosis suppressor protein 1 (FSP1) (AIFM2) with an EC50 of 103 nM. 了解更多
  39. AC1903

    Catalog No. A22296
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    TRPC5 inhibitor
    AC1903 is a specific and selective inhibitor of TRPC5 and has podocyte-protective properties. 了解更多
  40. Ribociclib hydrochloride

    Catalog No. A22303
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    CDK4/6 inhibitor
    Ribociclib hydrochloride (LEE011 hydrochloride) is a highly specific CDK4/6 inhibitor with IC50 values of 10 nM and 39 nM, respectively, 了解更多
  41. Gallein

    Catalog No. A22304
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    Gβγ subunit signalling inhibitor
    Gallein is a G protein βγ (Gβγ) subunit signalling inhibitor. Gallein disrupts the interaction of Gβγ subunits with the PI3Kγ. Anticancer agent. 了解更多
  42. BAY-474

    Catalog No. A22330
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    tyrosine-protein kinase c-Met inhibitor
    BAY-474 is a tyrosine-protein kinase c-Met inhibitor. BAY-474 acts as an epigenetics probe. 了解更多
  43. Decursinol angelate

    Catalog No. A22340
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    cytotoxic and protein kinase C (PKC) activating agent
    Decursinol angelate, a cytotoxic and protein kinase C (PKC) activating agent from the root of Angelica gigas, possesses anti-tumor and anti-inflammatory activities. 了解更多
  44. Solamargine

    Catalog No. A22357
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    anticancer agent
    Solamargine, a derivative from the steroidal solasodine in Solanum species, exhibits anticancer activities in numerous types of cancer. Solamargine induces non-selective cytotoxicity and P-glycoprotein inhibition. 了解更多
  45. SEL24-B489 HCl

    Catalog No. A22203
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    pan-PIM/FLT3 inhibitor
    SEL24-B489 HCl is a potent, dual pan-PIM/FLT3 inhibitor. 了解更多
  46. Perlapine

    Catalog No. A22204
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    hM3Dq DREADD agonist
    Perlapine is a potent and selective hM3Dq DREADD agonist (EC50 = 2.8 nM). This drug exhibits >10,000-fold selectivity for hM3Dq over hM3. 了解更多
  47. Dehydroascorbic acid

    Catalog No. A12366
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    potent cerebroprotection
    Dehydroascorbic acid, a blood-brain barrier transportable form of vitamin C, mediates potent cerebroprotection in experimental stroke. 了解更多
  48. CB-103

    Catalog No. A22160
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    protein-protein interaction (PPI) inhibitor
    CB-103 is a first-in-class, orally active protein-protein interaction (PPI) inhibitor of the NOTCH transcriptional activation complex. CB-103 has anti-tumor activity. 了解更多
  49. Laninamivir octanoate

    Catalog No. A22166
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    neuraminidase (NA) inhibitor
    Laninamivir octanoate (CS-8958), a prodrug of Laninamivir, is a long-acting neuraminidase (NA) inhibitor with anti-influenza virus activity. 了解更多
  50. ML382

    Catalog No. A22168
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    MRGPRX1 positive allosteric modulator
    ML382 is a potent and selective MRGPRX1 (Mas-related G protein-coupled receptor X1, MrgX1) positive allosteric modulator, with an EC50 of 190 nM. 了解更多

产品 1 到 50 共 7371个

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