Cannabinoid Receptors
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Taranabant ((1R,2R)stereoisomer)
Catalog No. A21705 CB1 receptor inverse agonistTaranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多 -
Taranabant
Catalog No. A11578 CB1 receptor inverse agonistTaranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多 -
Rimonabant hydrochloride
Catalog No. A11548 -
AM1241
Catalog No. A16397 -
Bay 59-3074
Catalog No. A16328 CB1/CB2 receptor 激动剂Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂,对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多 -
GW842166X
Catalog No. A11253 -
WIN 55,212-2 mesylate
Catalog No. A11932 CB receptor 激动剂WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂,在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多