Cannabinoid Receptors

Quick View
AM630

Catalog No. A14993
Quick View

添加到收藏
CB2 拮抗剂

AM630是一种选择性CB2拮抗剂，Ki为31.2 nM，选择性是CB1受体的150倍以上。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Md Shah Sufian, .et al. Early suppression of the endocannabinoid degrading enzymes FAAH and MAGL alters locomotor development in zebrafish, J Exp Biol, 2021, 21 JUNE
Quick View
Otenabant

Catalog No. A15200
Quick View

添加到收藏
CB1 receptor 拮抗剂

Otenabant是最近发现的选择性，高亲和力，竞争性CB1受体拮抗剂，Ki为0.7 nM。了解更多

Bulk Inquiry Free Sample
Quick View
AM251

Catalog No. A12914
Quick View

添加到收藏
CB1 receptor 拮抗剂

AM251是有效的CB1受体拮抗剂（IC50 = 8 nM，Ki = 7.49 nM），其选择性是CB2受体的306倍。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Potential for pharmacological manipulation of human embryonic stem cells. Br J Pharmacol. 2013 May; 169(2): 269–289.
Quick View
CP 945598 HCl (Otenabant HCl)

Catalog No. A11942
Quick View

添加到收藏
CB1 拮抗剂

CP 945598 HCl (Otenabant HCl)是一种有效且高度选择性的CB1拮抗剂。了解更多

Bulk Inquiry
Quick View
Taranabant racemate

Catalog No. A21699
Quick View

添加到收藏
CB1 antagonist/inverse agonist

Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多

Bulk Inquiry
Quick View
(±)-Ibipinabant

Catalog No. A21439
Quick View

添加到收藏
CB-1 receptor antagonist

(±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多

Bulk Inquiry
Quick View
JD-5037

Catalog No. A20837
Quick View

添加到收藏
CB1R antagonist

JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. 了解更多

Bulk Inquiry
Quick View
CB1 antagonist 2

Catalog No. A18810
Quick View

添加到收藏
CB1 antagonist

CB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多

Bulk Inquiry