“alpha ergocryptine”的搜索结果

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  1. Labetalol HCl

    Catalog No. A14239
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    alpha1/beta adrenergic receptors 拮抗剂
    Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多
  2. Ritanserin

    Catalog No. A21976
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    5-HT2 receptor antagonist
    Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. 了解更多
  3. Tamsulosin

    Catalog No. A12657
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    alpha-1A/alpha-1B-adrenoceptor 拮抗剂
    Tamsulosin是一种α1a-选择性α受体阻滞剂,用于对症治疗前列腺增生(BPH)。 了解更多
  4. NRA-0160

    Catalog No. A20128
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    Dopamine D4 receptor antagonist
    NRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). 了解更多
  5. AS2717638

    Catalog No. A18630
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    LPA5 antagonist
    AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia. 了解更多
  6. Pimozide

    Catalog No. A17375
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    Dopamine receptor antagonist
    Pimozide is a dopamine receptor antagonist, with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozide also inhibits STAT3 and STAT5. 了解更多
  7. Urapidil

    Catalog No. A17074
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    α1 adrenoreceptor 拮抗剂
    Urapidil是一种α1肾上腺素受体拮抗剂和5-HT1A受体激动剂。 了解更多
  8. Rauwolscine

    Catalog No. A13426
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    α2-adrenergic receptor 拮抗剂
    Rauwolscine是一种天然生物碱,具有选择性和可逆性α2肾上腺素能受体拮抗剂(Ki = 12 nM)。 了解更多
  9. Atipamezole HCl

    Catalog No. A13902
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    α2 adrenergic receptor 拮抗剂
    Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂(α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm)。已经被证明是大脑的渗透剂。 了解更多

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