“glucagon receptor”的搜索结果

产品 1 到 50 共 292个

每页
页面:
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

设置降序顺序
  1. Exendin-4 Acetate

    Catalog No. A21378
    Quick View
    glucagon-like peptide-1 receptor agonist
    Exendin-4 Acetate (Exenatide acetate), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. 了解更多
  2. Semaglutide

    Catalog No. A18908
    Quick View
    GLP-1 receptor agonist
    Semaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多
  3. (S)-Willardiine

    Catalog No. A21957
    Quick View
    AMPA/kainate receptors agonist
    (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. 了解更多
  4. L-APB

    Catalog No. A21872
    Quick View
    mGluRs M3 agonist
    L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. 了解更多
  5. Gaboxadol hydrochloride

    Catalog No. A21730
    Quick View
    GABAA receptors agonist
    Gaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多
  6. O-Phospho-L-serine

    Catalog No. A21159
    Quick View
    group III mGluR receptors agonist
    O-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2. 了解更多
  7. PSN632408

    Catalog No. A20902
    Quick View
    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多
  8. RU 24969

    Catalog No. A20857
    Quick View
    5-HT1A/5-HT1B receptors agonist
    RU 24969 is a selective agonist at the 5-HT1A and 5-HT1B receptors. 了解更多
  9. Carbetocin

    Catalog No. A18080
    Quick View
    peripheral oxytocin receptors agonist
    Carbetocin (Lonactene; Duratocin) is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth; an agonist at peripheral oxytocin receptors. 了解更多
  10. L-Glutamic acid monosodium salt

    Catalog No. A16591
    Quick View
    excitatory transmitter/agonist
    L-Glutamic acid monosodium salt acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). (S)-Glutamic acid shows a direct activating effect on the release of DA from dopaminergic terminals. 了解更多
  11. (S)-Glutamic acid

    Catalog No. A15458
    Quick View
    glutamate receptors agonist
    (S)-Glutamic acid acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). 了解更多
  12. Donitriptan

    Catalog No. A13145
    Quick View
    5-HT1B/1D receptors agonist
    Donitriptan is a potent, high efficacy agonist at 5-HT1B/1D receptors with pKis of 9.4 and 9.3, respectively. 了解更多
  13. DPI-3290

    Catalog No. A13699
    Quick View
    opioid receptors agonist
    DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively. 了解更多
  14. NMI 8739

    Catalog No. A12334
    Quick View
    dopamine D2 autoreceptor agonist
    NMI 8739 is a dopamine D2 autoreceptor agonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine. 了解更多
  15. Almitrine mesylate

    Catalog No. A18020
    Quick View
    Peripheral chemoreceptor agonist
    Almitrine mesylate, a peripheral chemoreceptor agonist, inhibits selectively the Ca2+-dependent K+ channel. 了解更多
  16. Cevimeline (AF-102B)

    Catalog No. A11372
    Quick View
    Muscarinic agonist
    Cevimeline (AF-102B) is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  17. Baclofen

    Catalog No. A18248
    Quick View
    GABA agonist
    Baclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. 了解更多
  18. Cevimeline hydrochloride

    Catalog No. A18092
    Quick View
    mAChR agonist
    Cevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  19. Dihydroergotamine Mesylate

    Catalog No. A17764
    Quick View
    Serotonin receptors agonist
    Dihydroergotamine Mesylate, also known as DHE or Migranal, is an ergot alkaloid used to treat migraines. It has similar actions to the triptans, acting as an agonist to the serotonin receptors and causing vasoconstriction of the intracranial blood vessels, but also interacts centrally with dopamine and adrenergic receptors. 了解更多
  20. Vilanterol

    Catalog No. A13125
    Quick View
    ultra-long-acting β? adrenoreceptor 激动剂
    Vilanterol是一种新的选择性β2-AR激动剂,PEC50值为10.37±0.05。 了解更多
  21. Cimaterol

    Catalog No. A13401
    Quick View
    β-adrenergic receptors 激动剂
    Cimaterol是β的有效激动剂;肾上腺素能受体(人β的pEC50 = 8.13、8.78和6.62;1β,2β和3β)。 了解更多
  22. BRL 37344 Na Salt

    Catalog No. A13676
    Quick View
    β3-adrenergic receptors 激动剂
    BRL 37344 Na Salt是具有脂解活性的β3-AR(β3-肾上腺素能受体)选择性激动剂。 了解更多
  23. BRL 52537 HCl

    Catalog No. A11210
    Quick View
    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  24. GW3965 HCl

    Catalog No. A11204
    Quick View
    LXR-like receptors 激动剂
    GW3965 HCl是一种选择性的口服活性肝X受体(LXR)完全激动剂。 了解更多
  25. Glucocorticoid receptor agonist

    Catalog No. A11431
    Quick View
    Glucocorticoid receptor agonist
    Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多
  26. H4 Receptor antagonist 1

    Catalog No. A18929
    Quick View
    histamine H4 receptor inverse agonist
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多
  27. Orexin 2 Receptor Agonist

    Catalog No. A15982
    Quick View
    Orexin 2 receptor 激动剂
    Orexin 2 Receptor Agonist一种有效的选择性Orexin2受体激动剂。 了解更多
  28. TGR5-Receptor-Agonist

    Catalog No. A13732
    Quick View
    TGR5(GPCR19) 激动剂
    TGR5 Receptor Agonist是一种有效的TGR5(GPCR19)激动剂,在U2-OS细胞分析(pEC50 = 6.8)和黑素细胞(pEC50 = 7.5)中显示出增强的效力。 了解更多
  29. Pardoprunox hydrochloride

    Catalog No. A21624
    Quick View
    partial dopamine D2 and D3 receptor agonist
    Pardoprunox hydrochloride is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) and D3 receptor (pKi = 8.6) partial agonist and 5-HT1A receptor (pKi = 8.5) full agonist. 了解更多
  30. Cutamesine

    Catalog No. A21152
    Quick View
    sigma 1 receptor agonist
    Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多
  31. Ralinepag

    Catalog No. A21073
    Quick View
    IP receptor agonist
    Ralinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively. 了解更多
  32. U-101017

    Catalog No. A13357
    Quick View
    Benzodiazepine receptor/GABAA receptor agonist
    U-101017 is a partial agonist of benzodiazepine receptor and GABAA receptor, with anxiolytic effects. 了解更多
  33. Cariprazine

    Catalog No. A21202
    Quick View
    D3 receptor and D2 receptor partial agonist
    Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多
  34. Dihydrexidine

    Catalog No. A21949
    Quick View
    D1-like dopamine receptor (D1/D5) agonist
    Dihydrexidine (DAR-0100) is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist with an IC50 of 10 nM for D1 receptor. Dihydrexidine exhibits potent antiparkinsonian activity. 了解更多
  35. Ditolylguanidine

    Catalog No. A21268
    Quick View
    Sigma receptor agonist
    Ditolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多
  36. YM348

    Catalog No. A12290
    Quick View
    5-HT2C receptor agonist
    YM348 is a potent and orally active 5-HT2C receptor agonist, which shows a high affinity for cloned human 5-HT2C receptor (Ki: 0.89 nM). 了解更多
  37. TCPOBOP

    Catalog No. A18376
    Quick View
    Androstane receptor agonist
    TCPOBOP is an agonist of the constitutive androstane receptor (CAR) (EC50 = 20 nM). TCPOBOP enhances the nuclear receptor CAR transactivation of cytochrome P450 (CYP), as dose-dependent direct agonist of CAR. 了解更多
  38. Lobeline hydrochloride

    Catalog No. A17333
    Quick View
    nicotinic receptor agonist
    Lobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes. 了解更多
  39. N6-Cyclohexyladenosine

    Catalog No. A21008
    Quick View
    A1 receptor agonist
    N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多
  40. Eglumegad

    Catalog No. A21005
    Quick View
    group II (mGlu2/3) receptor agonist
    Eglumegad (LY354740) is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively. 了解更多
  41. AVE 0991

    Catalog No. A20997
    Quick View
    angiotensin-(1-7) receptor agonist
    AVE 0991 is a nonpeptide and orally active angiotensin-(1-7) receptor agonist with an IC50 of 21 nM. 了解更多
  42. MK-0354

    Catalog No. A22008
    Quick View
    GPR109a receptor agonist
    MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多
  43. Aripiprazole (D8)

    Catalog No. A22004
    Quick View
    human 5-HT1A receptor partial agonist
    Aripiprazole D8 (OPC-14597 D8) is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. 了解更多
  44. Ro 10-5824 dihydrochloride

    Catalog No. A21986
    Quick View
    dopamine D4 receptor partial agonist
    Ro 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist, with Ki of 5.2 nM. 了解更多
  45. Mapracorat

    Catalog No. A21953
    Quick View
    glucocorticoid receptor agonist
    Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. 了解更多
  46. MT-7716 free base

    Catalog No. A21928
    Quick View
    non-peptide nociceptin receptor (NOP) agonist
    MT-7716 free base (W-212393) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. 了解更多
  47. AR-M 1000390 hydrochloride

    Catalog No. A21911
    Quick View
    δ opioid receptor agonist
    AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2??0.9 nM for δ agonist potency. 了解更多
  48. Vilazodone D8

    Catalog No. A21876
    Quick View
    SSR inhibitor / 5-HT1A receptor partial agonist
    Vilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多
  49. SKF 82958

    Catalog No. A21866
    Quick View
    D1/D5 receptor full agonist
    SKF 82958 is a D1/D5 receptor full agonist. 了解更多
  50. Nomegestrol acetate

    Catalog No. A21829
    Quick View
    progesterone receptor agonist
    Nomegestrol acetate is a potent, highly selective progestogen, which is characterized as a full agonist at the progesterone receptor, with no or minimal binding to other steroid receptors, including the androgen and glucocorticoid receptors. 了解更多

产品 1 到 50 共 292个

每页
页面:
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

设置降序顺序
Rewards