“MK-2206 dihydrochloride”的搜索结果
-
PPARγ 激动剂
Inolitazone dihydrochloride是一种新型的高亲和力PPARγ激动剂,可激活PPARγ,其EC50约为罗格列酮的EC50,对RIE细胞无影响。
了解更多
-
MAO-A inhibitor
Minaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression.
了解更多
-
PPARβ/δ inverse 激动剂
DG-172是一种口服活性强效PPARβ/δ反向激动剂 (IC50 = 26.9 nM)。DG-172在体外抑制小鼠成肌细胞中Angptl4基因的表达 (IC50 = 9.5 nM)。
了解更多
-
CYP450 dependent inhibitor
Liarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).
了解更多
-
PDE-5 inhibitor
Mirodenafil dihydrochloride (SK3530 dihydrochloride) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction.
了解更多