“glucagon receptor”的搜索结果

产品 1 到 50 共 1712个

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  1. Glucagon receptor antagonists-1

    Catalog No. A11428
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    glucagon receptor antagonist
    Glucagon receptor antagonists-1 is a highly potent glucagon receptor antagonist. 了解更多
  2. Glucagon receptor antagonists-3

    Catalog No. A11430
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    Glucagon receptor antagonist
    Glucagon receptor antagonists-3 is a highly potent glucagon receptor antagonist. 了解更多
  3. Glucagon receptor antagonists-2

    Catalog No. A11429
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    Glucagon receptor antagonist
    Glucagon receptor antagonists-2 is a highly potent glucagon receptor antagonist. 了解更多
  4. Glucagon HCl

    Catalog No. A17906
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    Glucagon is a peptide hormone, produced by alpha cells of the pancreas. It works to raise the concentration of glucose in the bloodstream. Its effect is opposite that of insulin, which lowers the glucose. 了解更多
  5. Glucagon-Like Peptide 1 (7-36) Amide

    Catalog No. A16895
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    Glucagon-Like Peptide 1 (7-36) Amide是一种强效葡萄糖依赖性促胰岛素肽,它是通过肠道L细胞中胰高血糖素原的翻译后加工而产生的。 了解更多
  6. Glucagon Human, His

    Catalog No. AP3258
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    Glucagon Human Recombinant, His Tag 了解更多
  7. Glucagon Human

    Catalog No. AP3257
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    Glucagon Human 了解更多
  8. Glucagon Human

    Catalog No. AP3256
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    Glucagon Human Recombinant 了解更多
  9. Glucagon (19-29), human

    Catalog No. A14875
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    Ca 2+ /Mg 2+ -ATPase 抑制剂
    Glucagon (19-29), human是有效的Ca2+/Mg2+ -ATPase抑制剂。 了解更多
  10. PF-06291874

    Catalog No. A20635
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    glucagon receptor antagonist
    PF-06291874 (Glucagon receptor antagonists-4) is a highly potent and orally active glucagon receptor antagonist. It displays low in vivo clearance in both rats and dogs. 了解更多
  11. GRA Ex-25

    Catalog No. A20625
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    glucagon receptor inhibitor
    GRA Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and human glucagon receptors, respectively. 了解更多
  12. Exendin-4

    Catalog No. A21580
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    glucagon-like peptide-1 receptor agonist
    Exendin-4 (Exenatide), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. 了解更多
  13. GLP-1R Antagonist 1

    Catalog No. A20679
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    glucagon-like peptide 1 receptor antagonist
    GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC50 of 650 nM. 了解更多
  14. Adomeglivant

    Catalog No. A20647
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    glucagon receptor antagonist
    Adomeglivant is a potent and selective glucagon receptor antagonist that is used in clinical trial for type 2 diabetes mellitus. 了解更多
  15. LGD-6972

    Catalog No. A21840
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    glucagon receptor antagonist
    LGD-6972 is a glucagon receptor antagonist. 了解更多
  16. Exendin-4 Acetate

    Catalog No. A21378
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    glucagon-like peptide-1 receptor agonist
    Exendin-4 Acetate (Exenatide acetate), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. 了解更多
  17. Semaglutide

    Catalog No. A18908
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    GLP-1 receptor agonist
    Semaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多
  18. Vildagliptin dihydrate

    Catalog No. A21898
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    DPP4 inhibitor
    Vildagliptin (LAF237 dihydrate;NVP-LAF 237 dihydrate) is a dipeptidyl peptidase 4 (DPP4) inhibitor that delays the degradation of glucagon-like peptide-1 (GLP-1). 了解更多
  19. GLP 2 Human

    Catalog No. AP3254
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    Human Glucagon Like Peptide-2 了解更多
  20. GLP 1 Human

    Catalog No. AP3253
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    Human Glucagon Like Peptide-1 了解更多
  21. GLP-1 Human (31 a.a.)

    Catalog No. AP3252
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    Glucagon Like Peptide-1 (31 a.a.) Human Recombinant 了解更多
  22. GLP 1 Human (37 a.a.)

    Catalog No. AP3251
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    Human Glucagon Like Peptide-1 (37 a.a.) 了解更多
  23. GLP-1 receptor agonist 1

    Catalog No. A19885
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    GLP-1 receptor agonist
    GLP-1 receptor agonist 1 is a glucagon-like peptide-1 (GLP-1) receptor agonist extracted from patent WO2018056453A1, Compound 67. 了解更多
  24. GLP-1 receptor agonist 2

    Catalog No. A19722
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    GLP-1R agonist
    GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist. 了解更多
  25. PF-06882961

    Catalog No. A22492
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    GLP-1R agonist
    PF-06882961 is a potent, orally bioavailable agonist of the glucagon-like peptide-1 receptor agonist (GLP-1R) 了解更多
  26. NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多
  27. VU0453379

    Catalog No. A18796
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    GLP-1R modulator
    VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM. 了解更多
  28. GCGR Human

    Catalog No. AP3255
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    Glucagon Receptor Human Recombinant 了解更多
  29. 4BP-TQS

    Catalog No. A22084
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    neuronal nicotinic acetylcholine receptors agonist
    4BP-TQS is an allosteric agonist of α7 subunit-containing neuronal nicotinic acetylcholine receptors (nAChRs). 了解更多
  30. FLTX1

    Catalog No. A22120
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    antiestrogenic properties
    FLTX1 is a fluorescent Tamoxifen derivative that can specifically label intracellular Tamoxifen-binding sites (estrogen receptors) under permeabilized and non-permeabilized conditions. FLTX1 exhibits the potent antiestrogenic properties of Tamoxifen in breast cancer cells. FLTX1 is devoid of the estrogenic agonistic effect on the uterus. 了解更多
  31. LDN-193189 2HCl

    Catalog No. A22307
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    BMP signaling inhibitor
    LDN193189 HCl (DM-3189) is the hydrochloride salt of LDN193189, which is a selective BMP signaling inhibitor, and inhibits the transcriptional activity of the BMP type I receptors ALK2 and ALK3 with IC50 of 5 nM and 30 nM in C2C12 cell lines, respectively, 200-fold selectivity for BMP versus TGF-β. 了解更多
  32. BIO-013077-01

    Catalog No. A22185
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    antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4
    BIO-013077-01, Novel potent antagonist of the TGFbeta family type I receptors, Alk5 and/or Alk4. 了解更多
  33. AP1189 acetate

    Catalog No. A22488
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    AP1189 is a biased agonist at receptors MC1 and MC3. AP1189 reduced cytokine release, an effect reliant on both MC1 and MC3 as evident from the use of Mc1r(-/-) and Mc3r(-/-) macrophages. 了解更多
  34. PNU-282987 free base

    Catalog No. A22518
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    PNU 282987 is a highly selective α7 nAChR agonist (Ki = 26 nM) displaying negligible blockade of α1β1γδ and α3β4 nAChRs (IC50 ?? 60 μM). Found to be inactive against a panel of 32 receptors at 1 μM, except 5-HT3 receptors (Ki = 930 nM). 了解更多
  35. NMP-7

    Catalog No. A22619
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    agonist of the CB1 and CB2 cannabinoid receptors
    NMP-7 is a non-selective agonist of the CB1 and CB2 cannabinoid receptors that acts by blocking T-type calcium channels. 了解更多
  36. YM 298198 Hydrochloride

    Catalog No. A22630
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    mGlu1 receptorsant agonist
    YM 298198 Hydrochloride is a non-competitive antagonist with high affinity and selectivity for mGlu1 receptors (Ki = 19 nM). 了解更多
  37. NPS2390

    Catalog No. A22631
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    group I mGlu antagonist
    NPS2390 is a group I mGlu antagonist. It displays noncompetitive antagonist activity at both mGlu1 and mGlu5 receptors. NPS2390 is thought to act on a site separate from the glutamate binding pocket. 了解更多
  38. Galnon

    Catalog No. A22633
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    agonist at the galanin receptors GALR
    Galnon is a selective, non-peptide agonist at the galanin receptors GALR. 了解更多
  39. Tracazolate

    Catalog No. A22635
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    pyrazolopyridine anxiolytic
    Tracazolate is a pyrazolopyridine anxiolytic known to interact with gamma-aminobutyric acid (GABA)(A) receptors, adenosine receptors, and phosphodiesterases. 了解更多
  40. Gardenoside

    Catalog No. A15630
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    hepatoprotective agent
    Gardenoside is a natural compound found in Gardenia fruits, with hepatoprotective properties. Gardenoside suppresses the pain of chronic constriction injury by regulating the P2X3 and P2X7 receptors. Gardenoside has an inhibitory effect on free fatty acids (FFA)-induced cellular steatosis. 了解更多
  41. SSR-241586

    Catalog No. A20773
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    neurokinin receptors antagonist
    SSR-241586 is an antagonist of neurokinin receptors. SSR-241586 is shown to be active in the treatment of depression, schizophrenia, urinary trouble, emesis, and irritable bowel syndrome (IBS). 了解更多
  42. AMG-009

    Catalog No. A20759
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    prostaglandin D2 antagonist
    AMG-009 is a potent antagonist of prostaglandin D2, with IC50 of 3 nM and 12 nM for CRTH2 and DP receptors, respectively. 了解更多
  43. Calcipotriol Impurity C

    Catalog No. A20634
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    Calcipotriol Impurity C is the impurity of Calcipotriol, Calcipotriol is a ligand of VDR-like receptors. 了解更多
  44. L-Cysteinesulfinic acid

    Catalog No. A20585
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    metabotropic glutamate receptors agonist
    L-Cysteinesulfinic acid is a potent agonist at several rat metabotropic glutamate receptors (mGluRs) with pEC50s of 3.92±0.03, 4.6±0.2, 3.9±0.2, 2.7±0.2, 4.0±0.2, and 3.94±0.08 for mGluR1, mGluR5, mGluR2, mGluR4, mGluR6, and mGluR8, respectively. 了解更多
  45. Ro 67-7476

    Catalog No. A20562
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    mGlu1 receptors modulator
    Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors. 了解更多
  46. DFMTI

    Catalog No. A20558
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    mGluR1 receptors
    DFMTI is an allosteric negative modulator of mGluR1 receptors. 了解更多
  47. DREADD agonist 21

    Catalog No. A20534
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    hM3Dq agonist.
    DREADD agonist 21 is a potent human muscarinic acetylcholine M3 receptors (hM3Dq) agonist(EC50=1.7 nM). 了解更多
  48. CGP 25454A

    Catalog No. A20448
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    dopamine autoreceptor antagonist
    CGP 25454A is a novel and selective presynaptic dopamine autoreceptor antagonist. 了解更多
  49. Fenobam

    Catalog No. A20372
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    mGluR5 antagonist
    Fenobam is a selective, orally active, and non-competitive mGluR5 antagonist acting at an allosteric modulatory site (Kd values are 54 and 31 nM for rat and human recombinant mGlu5 receptors, respectively). 了解更多
  50. SYM 2081

    Catalog No. A20332
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    kainate receptors agonist
    SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively. 了解更多

产品 1 到 50 共 1712个

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