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“glucagon receptor”的搜索结果

产品 1 到 50 共 55个

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  1. Ostarine (MK-2866, GTx-024)
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    Ostarine (MK-2866, GTx-024)

    Catalog No. A10253
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    Androgen Receptor Modulators
    Ostarine (MK-2866,GTX-024)是一种雄激素受体调节剂(SARM)。 了解更多
  2. PNU-120596
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    PNU-120596

    Catalog No. A11203
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    Nicotinic (α7) Receptor Modulator
    PNU-120596是α7神经元烟碱型乙酰胆碱受体的正变构调节剂。 了解更多
  3. Vortioxetine (Lu AA21004) hydrobromide
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    Vortioxetine (Lu AA21004) hydrobromide

    Catalog No. A12602
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    5-HT Receptor modulator
    Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物，可抑制5-HT（1A），5-HT（1B），5-HT（3A），5-HT（7）和SERT，IC50为15 nM，33 nM，3.7 nM，19 nM和1.6 nM。 了解更多
  4. Acolbifene (EM 652, SCH57068)
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    Acolbifene (EM 652, SCH57068)

    Catalog No. A12771
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    estrogen receptor modulator
    Acolbifene (EM 652,SCH57068)是第四代选择性的estrogen receptor拮抗剂，LC50 值为 22±3 nM。用于预防高乳腺癌女性的乳腺癌。 盐酸阿科比芬与体内雌激素受体结合，阻断雌激素对乳房的作用。 它是选择性雌激素受体调节剂（SERM）的一种。 了解更多
  5. BMS564929
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    BMS564929

    Catalog No. A12805
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    Androgen receptor (AR) modulator
    BMS-564929是一种新型，高效，口服活性，非甾体组织选择性雄激素受体（AR）调节剂，结合到雄激素受体，Ki 为 2.11±0.16 nM。该化合物已被推进临床试验，以治疗与年龄相关的功能衰退。 了解更多
  6. PU 02
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    PU 02

    Catalog No. A13757
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    5-HT3 Receptor Modulator
    PU 02是5-HT3受体的负变构调节剂。 了解更多
  7. Ospemifene
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    Ospemifene

    Catalog No. A14261
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    estrogen receptor modulator
    Ospemifene是一种非激素选择性雌激素受体调节剂（SERM）。 了解更多
  8. Farampator
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    Farampator

    Catalog No. A13798
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    AMPA receptor modulator
    Farampator是一种AMPA受体正调节剂，它可以改善短期记忆，但会损害情景记忆。 了解更多
  9. Indiplon
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    Indiplon

    Catalog No. A13769
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    GABAA receptor modulator
    Indiplon是吡唑并嘧啶，可作为GABAA受体的高亲和力正变构调节剂，以剂量依赖和可逆的方式增强GABA活化的氯离子电流。 了解更多
  10. MK-0773
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    MK-0773

    Catalog No. A15164
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    Androgen receptor modulator
    MK-0773是一种选择性雄激素受体调节剂（SARMs），是一种4-氮杂-类固醇，在人体中表现出组织选择性（IC50 = 6.6 nM）。 了解更多
  11. Toremifene
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    Toremifene

    Catalog No. A15265
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    Estrogen receptor modulator
    Toremifene是正在开发中的第二代选择性雌激素受体调节剂（SERM），用于预防骨质疏松症。 了解更多
  12. CBiPES HCl
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    CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂，IC50值为98.2 nM。 了解更多
  13. GSK-2881078
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    GSK-2881078

    Catalog No. A12645
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    androgen receptor modulator
    GSK-2881078是一种选择性雄激素受体调节剂（SARM），正在针对肌肉萎缩以改善其身体功能的受试者的肌肉生长和力量进行评估。 了解更多
  14. Ponesimod
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    Ponesimod

    Catalog No. A13307
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    S1P1 receptor modulator
    Ponesimod是一种口服活性，选择性鞘氨醇-1-磷酸受体1（S1P1）免疫调节剂，EC50为5.7 nM。 了解更多
  15. Lorediplon
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    Lorediplon

    Catalog No. A13449
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    GABAA receptor modulator
    Lorediplon 是一种新型的非苯二氮卓类催眠药，作为GABAA受体调节剂。 了解更多
  16. LY2452473
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    LY2452473

    Catalog No. A16873
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    androgen receptor modulator (SARM)
    LY2452473是一种口服生物利用型选择性雄激素受体调节剂（SARM），具有潜在的组织选择性雄激素/抗雄激素活性。 了解更多
  17. NSC-23026
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    NSC-23026

    Catalog No. A17151
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    CXCR4 receptor modulator
    NSC-23026是CXCR4受体调节剂。 了解更多
  18. VU0652835
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    VU0652835

    Catalog No. A18885
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    mGlu5 modulator
    VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM. 了解更多
  19. TAK-071
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    TAK-071

    Catalog No. A18626
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    M1 modulator
    TAK-071 is a novel, potent and highly selective muscarinic acetylcholine receptor 1 (M1R) positive allosteric modulator. EC50 of TAK-071 M1R agonist activities is 520 nM. 了解更多
  20. VU6005806
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    VU6005806

    Catalog No. A18488
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    M4 modulator
    VU6005806 (AZN-00016130) is a potent muscarnic acethylcholine receptor subtype 4 (M4) positive allosteric modulator (PAM), with EC50s of 94 nM, 28 nM, 87 nM and 68 nM for human, rat, dog and cyno M4, respectively. Used in the research of neuropsychiatric disorders. 了解更多
  21. MA-0204
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    MA-0204

    Catalog No. A19031
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    PPARδ modulator
    MA-0204 is a potent, highly selective and orally available peroxisome proliferator activated receptor δ (PPARδ) modulator with EC50s of 0.4 nM, 7.9 nM and 10 nM for human, mouse and rat PPARδ, respectively. Potential treatment for Duchene Muscular Dystrophy (DMD). 了解更多
  22. Rapacuronium bromide
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    Rapacuronium bromide

    Catalog No. A21119
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    mAChR modulator
    Rapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). 了解更多
  23. VU 0238429
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    VU 0238429

    Catalog No. A21519
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    positive allosteric modulator
    VU 0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5), with an EC50 of 1.16 μM. 了解更多
  24. PEPA
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    PEPA

    Catalog No. A21904
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    AMPA receptors allosteric modulator
    PEPA is an allosteric modulator of AMPA receptors; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity. 了解更多
  25. CMPDA
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    CMPDA

    Catalog No. A21909
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    AMPA receptors positive allosteric modulator
    CMPDA is a positive allosteric modulator of AMPA receptors with EC50s of 45.4 ?? 4.2 nM/63.4 ?? 5.6 nM for GluA2i/GluA2o receptor. 了解更多
  26. (Rac)-VU 6008667
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    (Rac)-VU 6008667

    Catalog No. A21939
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    mAChR M5 negative allosteric modulator
    (Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration. 了解更多
  27. Rovazolac
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    Rovazolac

    Catalog No. A18354
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    liver x receptor (LXR) modulator
    Rovazolac is a liver x receptor (LXR) modulator extracted from patent WO2013130892A1. 了解更多
  28. Lasofoxifene Tartrate
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    Lasofoxifene Tartrate

    Catalog No. A18097
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    selective Estrogen receptor modulator
    Lasofoxifene tartrate is a third-generation selective estrogen receptor modulator. 了解更多
  29. AZD9567
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    AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  30. D3-βArr
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    D3-βArr

    Catalog No. A18561
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    Thyrotropin receptor modulator
    D3-βArr is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 by direct TSHR activation and potentiates TSH-mediated preosteoblast differentiation in vitro. 了解更多
  31. Ryanodine
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    Ryanodine

    Catalog No. A12898
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    Ryanodine receptor modulator
    Ryanodine is a cell permeant ryanodine receptor modulator. Ryanodine can either stimulate or inhibit Ryanodine-mediated Ca2+ release depending on its concentrations. Poisonous diterpenoid found in Ryania speciosa. 了解更多
  32. Asoprisnil
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    Asoprisnil

    Catalog No. A19030
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    Progesterone receptor modulator
    Asoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. 了解更多
  33. Lu AF21934
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    Lu AF21934

    Catalog No. A12140
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    mGlu4 receptor modulator
    Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多
  34. VU6001376
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    VU6001376

    Catalog No. A13763
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    metabotropic glutamate receptor 4 modulator
    VU6001376 is a potent and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu4 PAM) with an EC50 of 50.1 nM. 了解更多
  35. Endothelin Mordulator 1
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    Endothelin Mordulator 1

    Catalog No. A13040
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    endothelin receptor modulator
    Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多
  36. IRAK inhibitor 3
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    IRAK inhibitor 3

    Catalog No. A11457
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    IL-1 receptor-associated kinase (IRAK) kinase modulator
    IRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator extracted from patent WO2008030579 A2. 了解更多
  37. Tamoxifen
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    Tamoxifen

    Catalog No. A16738
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    selective estrogen receptor modulator (SERM)
    Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells. 了解更多
  38. GLPG0492
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    GLPG0492

    Catalog No. A21105
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    androgen receptor modulator
    GLPG0492 is a novel selective androgen receptor modulator; exhibited anabolic activity on muscle, strongly dissociated from the androgenic activity on prostate after oral dosing. 了解更多
  39. PF-4778574
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    PF-4778574

    Catalog No. A21157
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    AMPA receptor positive allosteric modulator
    PF-4778574 is a potent AMPA receptor positive allosteric modulator (PAM) that has been shown to enhance cognition in animal models. 了解更多
  40. TCN238
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    TCN238

    Catalog No. A21191
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    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  41. RAD140
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    RAD140

    Catalog No. A21205
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    androgen receptor modulator
    RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM). 了解更多
  42. AZD8797
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    AZD8797

    Catalog No. A21230
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    human CX3CR1 receptor modulator
    AZD8797 is an allosteric non-competitive and orally active modulator of the human CX3CR1 receptor; antagonizes CX3CR1 and CXCR2 with Kis of 3.9 and 2800 nM, respectively. 了解更多
  43. Estetrol
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    Estetrol

    Catalog No. A21291
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    nuclear estrogen receptor modulator
    Estetrol, a natural estrogen synthesized exclusively during pregnancy by the human fetal liver, is a selective nuclear estrogen receptor modulator. 了解更多
  44. Foliglurax monohydrochloride
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    Foliglurax monohydrochloride

    Catalog No. A21384
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    glutamate receptor 4 modulator
    Foliglurax monohydrochloride (PXT002331 monohydrochloride) is a highly selective and potent, brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) , with an EC50 of 79 nM. Antiparkinsonian effect. 了解更多
  45. NS11394
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    NS11394

    Catalog No. A21425
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    GABA(A) receptor modulator
    NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors. 了解更多
  46. LUF6000
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    LUF6000

    Catalog No. A21532
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    A3 adenosine receptor allosteric modulator
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). 了解更多
  47. Pipendoxifene hydrochloride
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    Pipendoxifene hydrochloride

    Catalog No. A21623
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    estrogen receptor modulators
    Pipendoxifene hydrochloride is a selective estrogen receptor modulators (SERMs). 了解更多
  48. 4-Hydroxytamoxifen
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    4-Hydroxytamoxifen

    Catalog No. A20955
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    estrogen receptor modulator
    4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM). 了解更多
  49. Ulipristal acetate
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    Ulipristal acetate

    Catalog No. A21041
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    progesterone receptor modulator
    Ulipristal (acetate) is a novel selective progesterone receptor modulator (SPRM) for the treatment of benign gynecological conditions such as uterine myoma. 了解更多
  50. VU 0361737
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    VU 0361737

    Catalog No. A12467
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    mGlu4 receptors modulator
    VU 0361737是mGluR-4的选择性正变构调节剂（人和大鼠受体的EC50值分别为240和110 nM）。 了解更多

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