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BMS564929

Catalog No. A12805
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Androgen receptor (AR) modulator

BMS-564929是一种新型，高效，口服活性，非甾体组织选择性雄激素受体（AR）调节剂，结合到雄激素受体，Ki 为 2.11±0.16 nM。该化合物已被推进临床试验，以治疗与年龄相关的功能衰退。了解更多

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Acolbifene (EM 652, SCH57068)

Catalog No. A12771
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estrogen receptor modulator

Acolbifene (EM 652,SCH57068)是第四代选择性的estrogen receptor拮抗剂，LC50 值为 22±3 nM。用于预防高乳腺癌女性的乳腺癌。盐酸阿科比芬与体内雌激素受体结合，阻断雌激素对乳房的作用。它是选择性雌激素受体调节剂（SERM）的一种。了解更多

Product Citations (2)

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- Sumit Bansal, .et al. Inhibition of Human Sulfotransferase 2A1-Catalyzed Sulfonation of Lithocholic Acid, Glycolithocholic Acid, and Taurolithocholic Acid by Selective Estrogen Receptor Modulators and Various Analogs and Metabolites, J Pharmacol Exp Ther, 2019, June, 369 (3) 389-405
- Lirit N. Franks, .et al. Selective Estrogen Receptor Modulators: Cannabinoid Receptor Inverse Agonists with Differential CB1 and CB2 Selectivity, Front Pharmacol, 2016, 7: 503 PMID: 28066250
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Vortioxetine (Lu AA21004) hydrobromide

Catalog No. A12602
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5-HT Receptor modulator

Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物，可抑制5-HT（1A），5-HT（1B），5-HT（3A），5-HT（7）和SERT，IC50为15 nM，33 nM，3.7 nM，19 nM和1.6 nM。了解更多

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PNU-120596

Catalog No. A11203
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Nicotinic (α7) Receptor Modulator

PNU-120596是α7神经元烟碱型乙酰胆碱受体的正变构调节剂。了解更多

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Ostarine (MK-2866, GTx-024)

Catalog No. A10253
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Androgen Receptor Modulators

Ostarine (MK-2866,GTX-024)是一种雄激素受体调节剂(SARM)。了解更多

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