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Amisulpride hydrochloride
Catalog No. A21994 dopamine D2/D3 receptor antagonistAmisulpride hydrochloride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
Ziprasidone D8
Catalog No. A21989 5-HT / dopamine receptor antagonistZiprasidone D8 is deuterium labeled Ziprasidone, which is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多 -
Eplivanserin mixture
Catalog No. A21987 serotonin reuptake inhibitor/5-HT2A receptor antagonistEplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多 -
Niperotidine
Catalog No. A21981 histamine H2-receptor antagonistNiperotidine is a histamine H2-receptor antagonist. 了解更多 -
Ritanserin
Catalog No. A21976 5-HT2 receptor antagonistRitanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. 了解更多 -
Haloperidol D4'
Catalog No. A21971 dopamine D2 receptor antagonistHaloperidol D4' is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
Atenolol
Catalog No. A21962 -
Haloperidol D4
Catalog No. A21961 dopamine D2 receptor antagonistHaloperidol D4 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist. 了解更多 -
SB-224289 hydrochloride
Catalog No. A21920 5-HT1B receptor antagonistSB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
Olcegepant hydrochloride
Catalog No. A21900 CGRP1 receptor antagonistOlcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. 了解更多 -
Methoxy-PEPy
Catalog No. A21899 mGlu5 receptor antagonistMethoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. 了解更多 -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多 -
SB-269970 hydrochloride
Catalog No. A21889 5-HT7 receptor antagonistSB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多 -
Timapiprant sodium
Catalog No. A21883 D prostanoid receptor 2 antagonistTimapiprant sodium (OC000459 sodium) is a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist. 了解更多 -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多 -
Macitentan (n-butyl analogue)
Catalog No. A21845 endothelin ETA and ETB receptor antagonistMacitentan n-butyl analogue is a n-butyl analogue of Macitentan. Macitentan is an orally active, non-peptide dual endothelin ETA and ETB receptor antagonist for the potential treatment of idiopathic pulmonary fibrosis (IPF) and pulmonary arterial hypertension (PAH). 了解更多 -
Enclomiphene citrate
Catalog No. A21830 oestrogen receptor antagonistEnclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. 了解更多 -
Mavoglurant racemate
Catalog No. A21799 mGlu5 receptor antagonistMavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. 了解更多 -
GSK1521498 free base (hydrochloride)
Catalog No. A21792 μ-opioid receptor (MOR) antagonistGSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多 -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. 了解更多 -
H3B-6545 Hydrochloride
Catalog No. A21629 estrogen receptor covalent antagonistH3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多 -
Azilsartan D5
Catalog No. A21600 angiotensin II type 1 receptor antagonistAzilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多 -
Serlopitant
Catalog No. A21582 Neurokinin-1 (NK-1) receptor antagonistSerlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist. 了解更多 -
Losartan (D4 Carboxylic Acid)
Catalog No. A21578 angiotensin II receptor antagonistLosartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多 -
Fulvestrant R enantiomer
Catalog No. A21545 estrogen receptor antagonistFulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. 了解更多 -
Vofopitant dihydrochloride
Catalog No. A21543 NK1 receptor antagonistVofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist. 了解更多 -
L 888607 Racemate
Catalog No. A21482 DP1 antagonistL 888607 Racemate is a selective prostaglandin D2 receptor subtype 1 (DP1) antagonist, with Kis of 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively. 了解更多 -
JNJ-5207852
Catalog No. A21480 histamine H3 receptor antagonistJNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. 了解更多 -
Maropitant
Catalog No. A21473 -
(±)-Ibipinabant
Catalog No. A21439 CB-1 receptor antagonist(±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多 -
PF-03654746 Tosylate
Catalog No. A21434 histamine H3 receptor antagonistPF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
PF-03654746
Catalog No. A21429 histamine H3 receptor antagonistPF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
Batefenterol
Catalog No. A21387 muscarinic receptor antagonist and β2-adrenoceptor agonistBatefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively. 了解更多 -
SB-277011 dihydrochloride
Catalog No. A21353 dopamine D3 receptor antagonistSB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多 -
SB 242084 hydrochloride
Catalog No. A21349 5-HT2C receptor antagonistSB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多 -
SB290157 trifluoroacetate
Catalog No. A21347 C3a receptor antagonistSB290157 trifluoroacetate is a potent and selective C3a receptor antagonist with an IC50 of 200 nM. 了解更多 -
Darusentan
Catalog No. A21280 endothelin A (ETA) receptor antagonistDarusentan is a selective endothelin A (ETA) receptor antagonist. 了解更多 -
Lixivaptan
Catalog No. A21279 vasopressin receptor V2 antagonistLixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. 了解更多
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