“glucagon receptor”的搜索结果

产品 101 到 150 共 471个

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  1. Tipelukast

    Catalog No. A21249
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    leukotriene receptor antagonist
    Tipelukast (KCA 757) is a sulfidopeptide leukotriene receptor antagonist, an orally bioavailable anti-inflammatory agent and used for the treatment of asthma. 了解更多
  2. Mavoglurant

    Catalog No. A21223
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    mGlu5 receptor antagonist
    Mavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist, has an IC50 of 30 nM in a functional assay with human mGluR5. 了解更多
  3. ELN-441958

    Catalog No. A21207
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    B1 receptor antagonist
    ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. 了解更多
  4. LAS101057

    Catalog No. A21203
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    A2B receptor antagonist
    LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. 了解更多
  5. MDL 105519

    Catalog No. A21192
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    NMDA receptor antagonist
    MDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多
  6. Velneperit

    Catalog No. A21190
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    NPY Y5 receptor antagonist
    Velneperit (S-2367) is a novel neuropeptide Y (NPY) Y5 receptor antagonist. 了解更多
  7. CE-224535

    Catalog No. A21183
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    P2X7 receptor antagonist
    CE-224535 is a selective P2X7 receptor antagonist. 了解更多
  8. SB-423562

    Catalog No. A21170
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    calcium-sensing receptor (CaR) antagonist
    SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. 了解更多
  9. SB-423557

    Catalog No. A21169
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    alcium-sensing receptor (CaR) antagonist
    SB-423557 is an orally active calcium-sensing receptor (CaR) antagonist (IC50=520 nM), precursor of SB-423562 (IC50=73 nM). 了解更多
  10. Tezosentan

    Catalog No. A21118
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    endothelin (ET) receptor antagonist
    Tezosentan (RO 610612) is an endothelin (ET) receptor antagonist, with pA2s of 9.5, 7.7 for ETA and ETB receptors, respectively. 了解更多
  11. Transcrocetinate disodium

    Catalog No. A21051
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    NMDA receptor antagonist
    Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多
  12. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  13. Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  14. Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  15. SYM2206

    Catalog No. A20843
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    AMPA receptor antagonist
    SYM 2206 is a novel, potent, non-competitive AMPA receptor antagonist. 了解更多
  16. Haloperidol hydrochloride

    Catalog No. A18304
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    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  17. Setiptiline

    Catalog No. A18090
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    serotonin receptor antagonist
    Setiptiline(Org-8282) is a serotonin receptor antagonist. 了解更多
  18. (Z)-Thiothixene

    Catalog No. A17891
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    Serotonergic receptor antagonist
    (Z)-Thiothixene is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1. 了解更多
  19. Ziprasidone hydrochloride

    Catalog No. A16790
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    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  20. WAY-100635 Maleate

    Catalog No. A16787
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    5-HT1A receptor antagonist
    WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. 了解更多
  21. SB-334867 free base

    Catalog No. A16695
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    orexin OX1 receptor antagonist
    SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. 了解更多
  22. Ifenprodil tartrate

    Catalog No. A16583
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    NMDA receptor antagonist
    Ifenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多
  23. SB 271046 Hydrochloride

    Catalog No. A11573
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    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  24. Montelukast sodium

    Catalog No. A11490
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    CysLT1 receptor antagonist
    Montelukast (sodium) (MK0476) is a potent, selective CysLT1 receptor antagonist. 了解更多
  25. JDTic

    Catalog No. A11468
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    κ-opioid receptor antagonist
    JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多
  26. RF9

    Catalog No. A12944
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    Neuropeptide FF receptor antagonist
    RF9 is a potent and selective Neuropeptide FF receptor antagonist, with Kis of 58??5 and 75??9 nM for hNPFF1R and hNPFF2R, respectively. 了解更多
  27. CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. 了解更多
  28. FR167344 free base

    Catalog No. A12964
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    nonpeptide bradykinin receptor B2 antagonist
    FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. 了解更多
  29. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  30. Amelubant

    Catalog No. A12968
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    LTB4 receptor antagonist
    Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist. 了解更多
  31. RPR104632

    Catalog No. A13385
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    NMDA receptor antagonist
    RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. 了解更多
  32. Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. 了解更多
  33. GLPG0187

    Catalog No. A13423
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    Integrin receptor antagonist
    GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activity; inhibits αvβ1-integrin with an IC50 of 1.3 nM. 了解更多
  34. GV-196771A

    Catalog No. A13438
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    NMDA receptor antagonist
    GV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多
  35. Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  36. Valsartan

    Catalog No. A10962
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    angiotensin II receptor antagonist
    Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure. 了解更多
  37. Zafirlukast

    Catalog No. A11004
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    LTD4 receptor antagonist
    Zafirlukast is a potent orally active leukotriene D4 (LTD4) receptor antagonist. 了解更多
  38. Ziprasidone hydrochloride monohydrate

    Catalog No. A11008
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    5-HT (serotonin) and dopamine receptor antagonist
    Ziprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  39. Sitaxsentan

    Catalog No. A11565
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    ETA receptor antagonist
    Sitaxsentan (IPI 1040; TBC-11251) is a selective endothelin A (ETA) receptor antagonist. Antihypertensive. Sitaxsentan is used in treatment of chronic heart failure. 了解更多
  40. DW-1350

    Catalog No. A12250
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    LTB4 receptor antagonist
    DW-1350 is a LTB4 receptor antagonist. 了解更多
  41. TY-52156

    Catalog No. A12265
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    S1P3 receptor antagonist
    TY-52156 is a potent and selective S1P3 receptor antagonist with a Ki value of 110 nM. 了解更多
  42. 5-HT4 antagonist 1

    Catalog No. A12268
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    5-HT4 receptor antagonist
    5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. 了解更多
  43. lumateperone Tosylate

    Catalog No. A12279
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    5-HT2A receptor antagonist
    Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM). 了解更多
  44. Veralipride

    Catalog No. A13132
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    D2 receptor antagonist
    Veralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多
  45. ZD-1611

    Catalog No. A13151
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    ETA receptor antagonist
    ZD-1611 is a potent, orally active, selective ETA receptor antagonist, used for the research of ischemic stroke. 了解更多
  46. SL910102

    Catalog No. A13591
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    Angiotensin AT1 receptor antagonist
    SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. 了解更多
  47. GSK598809

    Catalog No. A13695
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    dopamine D3 Receptor (DRD3) antagonist
    GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist, with a pKi of 8.9. 了解更多
  48. Mozavaptan

    Catalog No. A16622
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    nonpeptide vasopressin V2 receptor antagonist
    Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM. 了解更多
  49. Tripelennamine hydrochloride

    Catalog No. A16767
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    H1-receptor antagonist
    Tripelennamine hydrochloride, a H1-receptor antagonist, is a psychoactive drug and member of the pyridine andethylenediamine classes that is used as an antipruritic and first-generation antihistamine. 了解更多
  50. Pirenzepine dihydrochloride

    Catalog No. A17916
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    M1 muscarinic receptor antagonist
    Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist. 了解更多

产品 101 到 150 共 471个

每页
页面:
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  2. 2
  3. 3
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