“glucagon receptor”的搜索结果

产品 51 到 100 共 292个

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  1. PF-5190457

    Catalog No. A21784
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    ghrelin receptor inverse agonist
    PF-5190457 is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36. 了解更多
  2. SKF-82958 hydrobromide

    Catalog No. A21763
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    D1/D5 receptor full agonist
    SKF-82958 hydrobromide is a D1/D5 receptor full agonist. 了解更多
  3. Camicinal

    Catalog No. A21750
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    motilin receptor agonist
    Camicinal (GSK962040) is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. 了解更多
  4. Eprotirome

    Catalog No. A21743
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    thyroid hormone receptor agonist
    Eprotirome is a liver-selective thyroid hormone receptor agonist. 了解更多
  5. LY 344864 S-enantiomer

    Catalog No. A21742
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    5-HT1F receptor agonist
    LY 344864 S-enantiomer is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist. 了解更多
  6. MCOPPB triHydrochloride

    Catalog No. A21722
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    nociceptin receptor agonist
    MCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors. 了解更多
  7. Pipequaline hydrochloride

    Catalog No. A21712
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    partial benzodiazepine receptor agonist
    Pipequaline hydrochloride (PK-8165 hydrochloride) is a partial benzodiazepine receptor agonist with anxiolytic activity. 了解更多
  8. Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  9. diABZI STING agonist-1 trihydrochloride

    Catalog No. A21694
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    STING receptor agonist
    diABZI STING agonist-1 (trihydrochloride) is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 for human PBMCs. 了解更多
  10. diABZI STING agonist-1

    Catalog No. A21688
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    STING receptor agonist
    diABZI STING agonist-1 is a selective stimulator of interferon genes (STING) receptor agonist, with an EC50s of 130 nM for human PBMCs. 了解更多
  11. SAG hydrochloride

    Catalog No. A21678
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    Smo receptor agonist
    SAG (hydrochloride) is a potent Smo receptor agonist, and activates the Hedgehog signaling pathway, with a Kd of 59 nM. 了解更多
  12. (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
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    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  13. Norepinephrine hydrochloride

    Catalog No. A21605
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    β1-selective adrenergic receptor agonist
    Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  14. CGP-42112

    Catalog No. A21575
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    Angiotensin-II subtype 2 receptor(AT2 R) agonist
    CGP-42112(CGP-42112A) is a potent Angiotensin-II subtype 2 receptor(AT2 R) agonist. 了解更多
  15. (S)-Mapracorat

    Catalog No. A21528
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    glucocorticoid receptor agonist
    (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. 了解更多
  16. Camicinal hydrochloride

    Catalog No. A21415
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    motilin receptor agonist
    Camicinal hydrochloride (GSK962040 hydrochloride) is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. 了解更多
  17. CP-409092 hydrochloride

    Catalog No. A21397
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    GABAA receptor partial agonist
    CP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. 了解更多
  18. GI 181771

    Catalog No. A21396
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    cholecystokinin 1 receptor agonist
    GI 181771 is a cholecystokinin 1 receptor agonist investigated for the treatment of obesity. 了解更多
  19. Plecanatide acetate

    Catalog No. A21393
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    GC-C receptor agonist
    Plecanatide acetate is a guanylate cyclase-C (GC-C) receptor agonist, with an EC50 of 190 nM in T84 cells. Plecanatide acetate shows anti-inflammatory activity in models of murine colitis. 了解更多
  20. SR 146131

    Catalog No. A21391
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    nonpeptide cholecystokinin 1 receptor agonist
    SR 146131 is a potent, orally available, and selective nonpeptide (cholecystokinin 1) receptor agonist. 了解更多
  21. CYT-1010 hydrochloride

    Catalog No. A21348
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    mu-opioid receptor agonist
    CYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多
  22. Dagrocorat

    Catalog No. A21312
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    glucocorticoid receptor agonist
    Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. 了解更多
  23. Fosdagrocorat

    Catalog No. A21303
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    dissociated glucocorticoid receptor agonist
    Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. 了解更多
  24. WAY 163909

    Catalog No. A21282
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    5-HT(2C) receptor agonist
    WAY 163909 is a potent and selective 5-HT(2C) receptor agonist with a Ki of 10.5??1.1 nM. 了解更多
  25. Befiradol

    Catalog No. A21189
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    5-HT1A receptor agonist
    Befiradol (NLX-112) is a selective 5-HT1A receptor agonist. 了解更多
  26. L-655708

    Catalog No. A21181
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    GABAA receptor inverse agonist
    L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM). 了解更多
  27. LY2812223

    Catalog No. A21100
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    mGlu2 receptor agonist
    LY2812223 is a highly potent, functionally selective mGlu2 receptor agonist with mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively). 了解更多
  28. Nelonicline

    Catalog No. A21079
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    neuronal nicotinic receptor agonist
    Nelonicline (ABT-126) is a selective neuronal nicotinic receptor agonist. 了解更多
  29. APNEA

    Catalog No. A20845
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    A3 adenosine receptor agonist
    APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. 了解更多
  30. Quinagolide hydrochloride

    Catalog No. A18038
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    dopamine D2 receptor agonist
    Quinagolide hydrochloride is a selective dopamine D2 receptor agonist, also is a prolactin inhibitor. 了解更多
  31. Pyrantel tartrate

    Catalog No. A18032
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    antinematodal thiophene nicotinic receptor agonist
    Pyrantel tartrate is an antinematodal thiophene nicotinic receptor agonist and can elicit spastic muscle paralysis in parasitic worms due to prolonged activation of the excitatory nicotinic acetylcholine (nACh) receptors on body wall muscle. 了解更多
  32. (R)-Baclofen

    Catalog No. A16680
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    GABAB receptor agonist
    (R)-Baclofen(STX209) is a selective GABAB receptor agonist. 了解更多
  33. Dexamethasone acetate

    Catalog No. A16494
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    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. 了解更多
  34. Varenicline Tartrate

    Catalog No. A11618
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    nicotinic receptor partial agonist
    Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does. 了解更多
  35. Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  36. Rivanicline oxalate

    Catalog No. A11544
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    neuronal nicotinic receptor agonist
    Rivanicline oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 3.6 μM). 了解更多
  37. CGS 21680

    Catalog No. A11354
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    adenosine A2A receptor agonist
    CGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. 了解更多
  38. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多
  39. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  40. AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  41. Acamprosate calcium

    Catalog No. A11308
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    GABA receptor agonist
    Acamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. 了解更多
  42. PRX933 hydrochloride

    Catalog No. A12261
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    5-HT2c receptor agonist
    PRX933 hydrochloride is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1. 了解更多
  43. AC260584

    Catalog No. A12264
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    M1 muscarinic receptor allosteric agonist
    AC260584 is an M1 muscarinic receptor allosteric agonist with a pEC50 of 7.6. 了解更多
  44. AP521

    Catalog No. A12280
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    human 5-HT1A receptor agonist
    AP521 is an agonist of human 5-HT1A receptor with an IC50 of 94 nM. 了解更多
  45. CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  46. Pipequaline

    Catalog No. A12551
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    partial benzodiazepine receptor agonist
    Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. 了解更多
  47. BW 245C

    Catalog No. A13494
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    prostanoid DP-receptor (DP1) agonist
    BW 245C is a prostanoid DP-receptor (DP1) agonist, used to treat stroke. 了解更多
  48. SX-3228

    Catalog No. A13687
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    benzodiazepine1 (BZ1) receptor agonist
    SX-3228 is a selective benzodiazepine1 (BZ1) receptor agonist with an IC50 of 17 nM. 了解更多
  49. Norepinephrine

    Catalog No. A11306
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    β1-selective adrenergic receptor agonist
    Norepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多
  50. CP-809101

    Catalog No. A12481
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    5-HT2C receptor agonist
    CP-809101 is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively. 了解更多

产品 51 到 100 共 292个

每页
页面:
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

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