“glucagon receptor”的搜索结果

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  1. 5-hydroxymethyl tolterodine (PNU 200577)

    Catalog No. A11166
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    muscarinic receptor 拮抗剂
    5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物,tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。 了解更多
  2. Biperiden HCl

    Catalog No. A10147
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    Muscarinic receptor antagonist
    Biperiden HCl是毒蕈碱受体拮抗剂,对M1亚型表现出一定的选择性。 了解更多
  3. Tolterodine tartrate (Detrol LA)

    Catalog No. A10937
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    muscarinic receptor 拮抗剂
    Tolterodine tartrate (Detrol LA)是毒蕈碱受体拮抗剂。 了解更多
  4. Solifenacin succinate

    Catalog No. A11215
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    muscarinic M3 receptor antagoinst
    Solifenacin succinate是毒蕈碱M3受体拮抗剂,用于治疗尿失禁。 了解更多
  5. SVT-40776 (Tarafenacin)

    Catalog No. A10808
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    muscarinic receptor 拮抗剂
    SVT-40776 (Tarafenacin)是新型M3毒蕈碱受体拮抗剂,用于治疗膀胱过度活动症。 了解更多
  6. Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。 了解更多
  7. Bethanechol chloride

    Catalog No. A10180
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    Muscarinic receptor 激动剂
    Bethanechol chloride是拟副交感神经的胆碱氨基甲酸酯,可选择性刺激毒蕈碱受体,而不会对烟碱样受体产生任何影响。 了解更多
  8. PF-3635659

    Catalog No. A13548
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    muscarinic M(3) receptor 拮抗剂
    PF-3635659是有效的毒蕈碱M3受体拮抗剂。 了解更多
  9. Umeclidinium bromide

    Catalog No. A15268
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    Muscarinic receptor 拮抗剂
    Umeclidinium bromide (GSK573719A)是毒蕈碱受体拮抗剂,可用于治疗慢性阻塞性肺疾病(COPD)。 了解更多
  10. Metanicotine

    Catalog No. A11545
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    Nicotinic receptor 激动剂
    Metanicotine是一种神经元的尼古丁受体激动剂,对α4β2亚型具有高选择性(Ki = 26 nM)。选择性是α7受体(Ki = 36000 nM)的1,000倍以上。 了解更多
  11. Revefenacin

    Catalog No. A15986
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    muscarinic receptor 拮抗剂
    Revefenacin是正在研发中的有效,选择性毒蕈碱受体拮抗剂,可用于治疗COPD。 了解更多
  12. Atropine methyl bromide

    Catalog No. A18026
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    mAChR antagonist
    Atropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and a mydriatic for dilation of the pupil during ophthalmic examination. It is introduced for relieving pyloric spasm in infants for its highly polar nature. It penetrates less readily into the central nervous system than atropine. 了解更多
  13. Rapacuronium bromide

    Catalog No. A21119
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    mAChR modulator
    Rapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). 了解更多
  14. mAChR-IN-1 hydrochloride

    Catalog No. A21398
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    mAChR antagonist
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多
  15. mAChR-IN-1

    Catalog No. A21518
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    mAChR antagonist
    mAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多
  16. (Rac)-VU 6008667

    Catalog No. A21939
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    mAChR M5 negative allosteric modulator
    (Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration. 了解更多
  17. Oxotremorine M iodide

    Catalog No. A21977
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    mAChR agonist
    Oxotremorine M iodide is a potent and non-selective muscarinic acetylcholine receptor (mAChR) agonist. 了解更多
  18. Darenzepine

    Catalog No. A12333
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    muscarinic receptor inhibitor
    Darenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多
  19. Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  20. Oxybutynin

    Catalog No. A10684
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    Oxybutynin (Ditropan)是一种抗胆碱能药物,是一种竞争性的muscarinic acetylcholine receptorM1,M2,和M3拮抗剂,用于缓解尿道和膀胱疾病。 了解更多
  21. Imidafenacin

    Catalog No. A15490
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    M3 receptors 抑制剂
    Imidafenacin是一种有效的选择性M3受体抑制剂,Kb为0.317 nM。对M2受体的效力较低(IC50 = 4.13 nM)。 了解更多
  22. Cevimeline hydrochloride

    Catalog No. A18092
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    mAChR agonist
    Cevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多
  23. Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多

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