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Minodronic acid
Catalog No. A21975 purinergic P2X2/3 receptors antagonistMinodronic acid (YM-529) is an antagonist of purinergic P2X2/3 receptors involved in pain. 了解更多 -
Gaboxadol hydrochloride
Catalog No. A21730 GABAA receptors agonistGaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多 -
Baclofen
Catalog No. A18248 GABA agonistBaclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing It acts at spinal and supraspinal sites, reducing excitatory transmission. 了解更多 -
Anisodamine
Catalog No. A18215 alpha-1 adrenergic receptors / mAChRs inhibitorAnisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多 -
Cevimeline hydrochloride
Catalog No. A18092 mAChR agonistCevimeline (Evoxac) Hcl is a parasympathomimetic and muscarinic agonist, with particular effect on M3 receptors; used in the treatment of dry mouth associated with sjogren's syndrome. 了解更多 -
Cangrelor Tetrasodium
Catalog No. A17919 P2Y12 receptors inhibitorCangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多 -
Ro 25-6981 maleate
Catalog No. A13144 -
RO 25-6981 maleate
Catalog No. A16083 NMDA receptors blockerRO 25-6981 maleate是含有NR2B亚基的NMDA受体的强效和选择性活性依赖性阻断剂。克隆的受体亚基组合NR1C/NR2B和NR1C/NR2A的IC50值分别为0.009和52 uM。 了解更多 -
Imidafenacin
Catalog No. A15490 M3 receptors 抑制剂Imidafenacin是一种有效的选择性M3受体抑制剂，Kb为0.317 nM。对M2受体的效力较低（IC50 = 4.13 nM）。 了解更多 -
CIQ
Catalog No. A15523 -
NVP-AAM077 Tetrasodium Hydrate (PEAQX)
Catalog No. A14071 -
2-Hydroxysaclofen
Catalog No. A13696 -
Oxybutynin
Catalog No. A10684 Oxybutynin (Ditropan)是一种抗胆碱能药物，是一种竞争性的muscarinic acetylcholine receptorM1，M2，和M3拮抗剂，用于缓解尿道和膀胱疾病。 了解更多 -
JNJ-54175446
Catalog No. A18675 P2X7 receptor antagonistJNJ-54175446 is a potent and selective brain penetrant P2X7 receptor antagonist, with pIC50s of 8.46 and 8.81 for hP2X7 receptor and rP2X7 receptor, respectively. 了解更多 -
Rislenemdaz
Catalog No. A21907 NMDA receptor GluN2B antagonistRislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively. 了解更多 -
SDZ 220-581 hydrochloride, SDZ220-581, SDZ-220-581
Catalog No. A21897 NMDA receptor antagonistSDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. 了解更多 -
7-Chlorokynurenic acid sodium salt
Catalog No. A21879 NMDA receptor antagonist7-Chlorokynurenic acid sodium salt is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM). 了解更多 -
CP-409092 hydrochloride
Catalog No. A21397 GABAA receptor partial agonistCP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. 了解更多 -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多 -
CE-224535
Catalog No. A21183 -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多 -
Clopidogrel thiolactone
Catalog No. A20862 P2Y12 receptor inhibitorClopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent. 了解更多 -
(R)-Baclofen
Catalog No. A16680 GABAB receptor agonist(R)-Baclofen(STX209) is a selective GABAB receptor agonist. 了解更多 -
Ifenprodil tartrate
Catalog No. A16583 NMDA receptor antagonistIfenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多 -
GV-196771A
Catalog No. A13438 NMDA receptor antagonistGV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多 -
Tiotropium Bromide
Catalog No. A10934 muscarinic acetylcholine receptor (mAChR) antagonistTiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多 -
Acamprosate calcium
Catalog No. A11308 GABA receptor agonistAcamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. 了解更多 -
Darenzepine
Catalog No. A12333 muscarinic receptor inhibitorDarenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多 -
MRK-016
Catalog No. A12046 GABAA α5 receptor agonistMRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多 -
Homotaurine
Catalog No. A17944 GABA receptor agonistTramiprosate, also known as homotaurine, is a gamma-Aminobutyric acid (GABA) receptor agonist and a glycosaminoglycan mimetic used in the treatment of Alzheimer's disease. 了解更多 -
Mephenesin
Catalog No. A17493 NMDA receptor antagonistMephenesin is an NMDA receptor antagonist, is a centrally acting muscle relaxant. 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多 -
Clopidogrel
Catalog No. A21206 platelet inhibitorClopidogrel is a well-known and orally active platelet inhibitor that targets P2Y12 receptor. Clopidogrel is used to inhibit blood clots in coronary artery disease, peripheral vascular disease, and cerebrovascular disease. 了解更多 -
Oxotremorine M iodide
Catalog No. A21977 mAChR agonistOxotremorine M iodide is a potent and non-selective muscarinic acetylcholine receptor (mAChR) agonist. 了解更多 -
(Rac)-VU 6008667
Catalog No. A21939 mAChR M5 negative allosteric modulator(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration. 了解更多 -
Varenicline Hydrochloride
Catalog No. A21539 α4β2 nAChR partial agonistVarenicline Hydrochloride (CP 526555 hydrochloride) is a high affinity, selective α4β2 nicotine acetylcholine receptor (nAChR) partial agonist and full α7 nAChR agonist. 了解更多 -
mAChR-IN-1
Catalog No. A21518 mAChR antagonistmAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多 -
mAChR-IN-1 hydrochloride
Catalog No. A21398 mAChR antagonistmAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多
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