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￥ 0.00 “sb269970 hcl”的搜索结果
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BRL 52537 HCl
Catalog No. A11210 Opioid Receptors 激动剂BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂（Ki = 0.24 nM）。比吗啡强25倍。 了解更多 -
Rotigotine HCl
Catalog No. A11118 Dopamine Receptor 激动剂Rotigotine hydrochloride是一种多巴胺D2和D3受体激动剂。D2和D3的Ki值分别为13和0.71 nM。 了解更多 -
Phenylephrine HCl
Catalog No. A11666 α1-adrenergic receptor 激动剂Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂，主要用作减充血剂，扩张瞳孔和增加血压的药物。 了解更多 -
Clomipramine HCl
Catalog No. A10231 5-HT Receptor 激动剂Clomipramine HCl是下列转运蛋白的阻滞剂：5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM)，去甲肾上腺素转运蛋白（NET）(Ki = 54 nM)，多巴胺转运蛋白（DAT）(Ki = 3，020 nM)，甘氨酸转运蛋白（GlyT/LeuT）。 了解更多 -
Roxatidine acetate hydrochloride
Catalog No. A11921 Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多 -
Phenoxybenzamine hydrochloride
Catalog No. A10719 α-adrenergic (AR) 拮抗剂/CaM 抑制剂Phenoxybenzamine hydrochloride是一种细胞可渗透的，非特异性的，不可逆的α-肾上腺素（AR）拮抗剂，也可作为CaM抑制剂。 了解更多 -
Olopatadine hydrochloride
Catalog No. A10671 Olopatadine hydrochloride是一种双重作用的组胺H1受体拮抗剂和肥大细胞稳定剂。 了解更多 -
Oxymetazoline hydrochloride
Catalog No. A10686 -
Tetrahydrozoline Hydrochloride
Catalog No. A13080 -
lorcaserin hydrochloride (APD-356)
Catalog No. A12598 serotonin 2C receptor 激动剂lorcaserin hydrochloride (APD-356)是血清素2C受体激动剂，可指示与减少热量饮食和增加体育锻炼以减轻慢性体重成人管理。 了解更多 -
Octopamine hydrochloride
Catalog No. A13419 Octopamine hydrochloride是一种无脊椎生物胺神经递质，与去甲肾上腺素相关，是肾上腺素受体激动剂。 了解更多 -
Xylazine HCl
Catalog No. A13434 -
SB-408124 HCl
Catalog No. A15231 OX Receptor 拮抗剂SB408124 Hydrochloride是OX1受体的非肽拮抗剂，全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。 了解更多 -
AMD-070 HCl
Catalog No. A14997 CXCR4 拮抗剂在CXCR4 125I-SDF抑制结合试验中，AMD-070 HCl是一种有效的选择性CXCR4拮抗剂，IC50值为13 nM，抑制T-4型HIV-1（NL4.3株）在MT-4细胞中的复制和PBMC。 了解更多 -
Asenapine HCl
Catalog No. A15002 adrenergic receptor/5-HT receptor 抑制剂Asenapine hydrochloride抑制肾上腺素能受体（α1，α2A，α2B，α2C）的Ki为0.25-1.2 nM，还抑制5-HT受体（1A，1B，2A，2B，2C，5A，6、7），Ki为0.03- 4.0 nM。 了解更多 -
Atrasentan HCl
Catalog No. A15007 Endothelin 拮抗剂 receptorAtrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体（IC50 = 0.0551 nM，ETA）。 了解更多 -
SCH 23390 HCl
Catalog No. A13066 -
Promazine hydrochloride
Catalog No. A17638 D2DR inhibitorPromazine Hydrochloride is a phenothiazine compound and D2DR inhibitor. Promazine Hydrochloride has been employed in studies investigating dopamine-stimulated glycosylation of brain proteins in vitro. It has actions similar to chlorpromazine but with less antipsychotic activity. 了解更多 -
Moxisylyte hydrochloride
Catalog No. A17725 alpha-adrenergic blocking agentMoxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomimetic agents. 了解更多 -
Metipranolol hydrochloride
Catalog No. A18064 β-adrenergic receptor antagonistMetipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多 -
Metoclopramide hydrochloride hydrate
Catalog No. A18072 Dopamine D2 antagonistMetoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. 了解更多 -
MK 3207 HCl
Catalog No. A10598 CGRP Receptor 拮抗剂MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂，IC50为0.12 nM。 了解更多 -
Moxonidine Hydrochloride
Catalog No. A13416 imidazoline receptor 1 激动剂Moxonidine Hydrochloride (BDF5895)是咪唑啉1型受体（I1-R）选择性激动剂，为降压剂。 了解更多 -
CBiPES HCl
Catalog No. A15811 -
Melitracen hydrochloride
Catalog No. A17494 dopamine D1/2 receptor antagonistMelitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多 -
Nefazodone hydrochloride
Catalog No. A17622 5-HT2 receptors inhibitorNefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多 -
Ziprasidone hydrochloride
Catalog No. A16790 5-HT (serotonin)/dopamine receptor antagonistZiprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多 -
MCOPPB 3HCl
Catalog No. A10561 -
Naftopidil 2HCl
Catalog No. A10619 5-HT1A and α1-adrenergic receptor 拮抗剂Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂，IC50分别为0.1μM和0.2μM。 了解更多 -
Vanoxerine 2HCl (GBR-12909)
Catalog No. A10725 dopamine re-uptake 抑制剂Vanoxerine 2HCl (GBR-12909)是哌嗪衍生物，是一种有效的、选择性的多巴胺摄取（dopamine uptake）抑制剂。 了解更多 -
Plerixafor 8HCl (DB06809)
Catalog No. A10913 CXCR4 拮抗剂Plerixafor 8HCl (DB06809)是CXCR4趋化因子受体拮抗剂，作用于CXCR4和CXCL12介导调节的趋化性， IC50分别为44 nM和5.7 nM。 了解更多 -
Pramipexole dihydrochloride monohyrate
Catalog No. A10747 Dopamine Receptor 激动剂Pramipexole dihydrochloride monohyrate是非麦角灵类的多巴胺激动剂，适用于治疗早期帕金森氏病（PD）和不安腿综合征（RLS）。 了解更多 -
B-HT 920 2HCl
Catalog No. A11341 -
GBR-12935 2HCl
Catalog No. A11937 -
Cetirizine Dihydrochloride
Catalog No. A10195 Cetirizine Dihydrochloride是第二代抗组胺药，是羟嗪的主要代谢产物，是用于治疗过敏，花粉症，血管性水肿和荨麻疹的消旋选择性H1受体反向激动剂。 了解更多 -
A 943931 2HCl
Catalog No. A13442 -
Cyclizine 2HCl
Catalog No. A16472 -
Azelastine HCl (Allergodil)
Catalog No. A10117 Azelastine HCl (Allergodil)是有效的第二代选择性组胺拮抗剂（组胺-H1-受体拮抗剂）。 了解更多 -
Promethazine HCl
Catalog No. A14248 -
Cyclobenzaprine HCl
Catalog No. A14255 -
SKF38393 HCl
Catalog No. A15839 -
Buspirone HCl
Catalog No. A15687 5HT(1A) receptor 激动剂Buspirone hydrochloride是一种具有5-D（2）多巴胺能作用的血清素能（5HT（1A）受体激动剂）抗焦虑药，用于焦虑症。 了解更多 -
Isoprenaline HCl
Catalog No. A10484 β adrenoceptor 激动剂Isoprenaline HCl或isoproterenol是非选择性β肾上腺素能激动剂，在结构上类似于肾上腺素。 了解更多 -
CP 945598 HCl (Otenabant HCl)
Catalog No. A11942 -
SDZ 205-557 HCl
Catalog No. A13766 -
SB 399885 HCl
Catalog No. A14102 5-HT6 拮抗剂SB 399885 hydrochloride是一种有效的，脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍（对于人类重组，天然大鼠和天然人类SR-6受体，pKi值分别为9.11、8.81和9.02）。 了解更多 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多
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