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搜索结果：“alpha ergocryptine”

“alpha ergocryptine”的搜索结果

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MRK-016

Catalog No. A12046
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GABAA α5 receptor agonist

MRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多

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NS11394

Catalog No. A21425
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GABA(A) receptor modulator

NS11394 is a potent and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors. 了解更多

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TPA 023

Catalog No. A20140
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GABAA α2/α3 agonist

TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. 了解更多

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Basmisanil

Catalog No. A21321
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GABAAα5 modulator

Basmisanil is a highly selective GABAAα5 negative allosteric modulator. 了解更多

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Gaboxadol hydrochloride

Catalog No. A21730
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GABAA receptors agonist

Gaboxadol hydrochloride (Lu 02-030 hydrochloride) is a selective agonist at GABAA receptors that contain α4-δ subunits, and has anxiolytic and sedative effects. 了解更多

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L-655708

Catalog No. A21181
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GABAA receptor inverse agonist

L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM). 了解更多

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