“sb269970 hcl”的搜索结果

产品 301 到 325 共 325个

每页
页面:
  1. 3
  2. 4
  3. 5
  4. 6
  5. 7

设置升序顺序
  1. AZD1208 HCl

    Catalog No. A16927
    Quick View
    PIM kinases 抑制剂
    AZD1208 HCl是一种新型的,口服可生物利用的高选择性PIM激酶抑制剂。 了解更多
  2. RS 17053 HCl

    Catalog No. A16885
    Quick View
    α1A 拮抗剂
    RS 17053 HCl是α1A受体拮抗剂,对α1A受体具有很高的亲和力(pKi和pA2估计为9.1-9.9),选择性比α1B和α1D亚型高30-100倍(pKi和pA2估计为7.7- 7.8)。 了解更多
  3. Desformylflustrabromine HCl

    Catalog No. A17103
    Quick View
    Desformylflustrabromine HCl是α4β2的正变构调节剂,也是肌肉型nAChR抑制剂。 了解更多
  4. E6446 HCl

    Catalog No. A17149
    Quick View
    E6446 HCl是核酸敏感TLR的合成拮抗剂。 了解更多
  5. S38093 HCl

    Catalog No. A17148
    Quick View
    H3 receptors
    S38093 HCl是组胺H3受体的反向激动剂。 了解更多
  6. Anavex2-73 HCl

    Catalog No. A17145
    Quick View
    ??1 激动剂
    Anavex2-73 HCl是毒蕈碱/中度sigma1受体激动剂,可减轻东pol碱和地佐西平引起的学习障碍。 了解更多
    • 最新产品

    TCS-OX2-29 HCl

    Catalog No. A17136
    Quick View
    OX2 receptor 拮抗剂
    TCS-OX2-29 HCl是一种选择性OX2受体拮抗剂,IC50值为40 nM。 了解更多
  7. Procyclidine HCl

    Catalog No. A17371
    Quick View
    Muscarinic antagonist
    Procyclidine hydrochloride is a muscarinic antagonist that crosses the blood-brain barrier and is used in the treatment of drug-induced extrapyramidal disorders and in Parkinsonism. 了解更多
    • 最新产品

    SAR-7334 HCl

    Catalog No. A17237
    Quick View
    TRPC6 inhibitor
    SAR7334 is a novel, highly potent and bioavailable inhibitor of TRPC6 channels that opens new opportunities for the investigation of TRPC channel function in vivo. SAR7334 inhibited TRPC6, TRPC3 and TRPC7-mediated Ca(2+) influx into cells with IC50 s of 9.5, 282 and 226 nM, whereas TRPC4 and TRPC5-mediated Ca(2+) entry was not affected. 了解更多
  8. Ractopamine HCl

    Catalog No. A17372
    Quick View
    beta-Adrenergic agonist
    Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多
  9. Acecainide HCl

    Catalog No. A22660
    Quick View
    Class III antiarrhythmic agent
    Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide. Acecainide is a Class III antiarrhythmic agent. It can be given either intravenously or orally, and is eliminated primarily by renal excretion. 了解更多
  10. MK-212 HCl

    Catalog No. A22531
    Quick View
    MK 212 hydrochloride is a 5-HT receptor agonist; displays selectivity for 5-HT2C over 5-HT2A (IC50 values are 0.028 and 0.42 μM for human 5-HT2C and 5-HT2A receptors expressed in HEK293 cells respectively). 了解更多
  11. Varenicline HCl

    Catalog No. A22519
    Quick View
    Varenicline is a nicotinic receptor partial agonist. 了解更多
  12. AVN-101 HCl

    Catalog No. A22498
    Quick View
    5-HT7 receptor antagonist
    AVN-101 is a very potent 5-HT7 receptor antagonist, with slightly lesser potency toward 5-HT6, 5-HT2A, and 5HT-2C receptors. It is a milti-target drug candidate for the treatment of CNS disorders. 了解更多
  13. UK-371804 HCl

    Catalog No. A22379
    Quick View
    uPA inhibitor
    UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). 了解更多
  14. SEL24-B489 HCl

    Catalog No. A22203
    Quick View
    pan-PIM/FLT3 inhibitor
    SEL24-B489 HCl is a potent, dual pan-PIM/FLT3 inhibitor. 了解更多
  15. Prexasertib HCl

    Catalog No. A22156
    Quick View
    ATP-competitive CHK1 inhibitor
    Prexasertib (LY2606368) is an ATP-competitive CHK1 inhibitor with a Ki value of 0.9 nmol/L. For CHK2 and RSK, its IC50 values are 8 nM and 9 nM respectively in cell-free assay. 了解更多
  16. 17-DMAG HCl (Alvespimycin)

    Catalog No. A10011
    Hsp90 抑制剂
    17-DMAG HCl (Alvespimycin)是17-AAG和格尔德霉素的水溶性类似物,与Hsp90的ATP结合位点结合并抑制其伴侣活性。显示出比17-AAG更有效的抗肿瘤活性。 了解更多
  17. MLN4924 (HCL Salt)

    Catalog No. A11499
    Quick View
    NAE 抑制剂
    MLN4924 (HCL Salt)是一种有效,选择性的 NEDD8 活化酶 (NEDD8-activating enzyme) 抑制剂。 了解更多
  18. SB203186 HCl

    Catalog No. A22523
    Quick View
    5-HT4 receptor antagonist
    SB203186 is potent 5-HT4 receptor antagonist. 了解更多
  19. TP0427736 HCl

    Catalog No. A22382
    Quick View
    ALK5 kinase activity inhibitor
    TP0427736 is a potent inhibitor of ALK5 kinase activity with an IC50 of 2.72 nM and this effect is 300-fold higher than the inhibitory effect on ALK3 (IC50 = 836 nM for ALK3). It also inhibits Smad2/3 phosphorylation in A549 cells induced by TGF-β1 with an IC50 value of 8.68 nM. 了解更多
  20. AMG-073 HCl (Cinacalcet HCl)

    Catalog No. A10219
    Quick View
    CaSR activator
    AMG-073 HCl(Cinacalcet HCl)是一种用于治疗甲状旁腺功能亢进的化合物,称为拟钙剂,通过增加甲状旁腺钙敏感受体(CaR)对细胞外钙的敏感性来减少甲状旁腺激素(PTH)的合成和分泌 。 了解更多
  21. P005672 HCl (Sarecycline HCl)

    Catalog No. A11283
    Quick View
    P005672 HCl (Sarecycline HCl)是用于抗菌/消炎痤疮治疗的II期药物。 了解更多
  22. SB-269970 hydrochloride

    Catalog No. A21889
    Quick View
    5-HT7 receptor antagonist
    SB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多
  23. SB269970 HCl

    Catalog No. A11925
    Quick View
    5-HT7 receptor 拮抗剂
    SB269970 HCl是有效的选择性5-HT7受体拮抗剂。 了解更多

产品 301 到 325 共 325个

每页
页面:
  1. 3
  2. 4
  3. 5
  4. 6
  5. 7

设置升序顺序
Rewards