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JNJ-5207852
Catalog No. A21480 histamine H3 receptor antagonistJNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. 了解更多 -
Maropitant
Catalog No. A21473 -
(±)-Ibipinabant
Catalog No. A21439 CB-1 receptor antagonist(±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多 -
PF-03654746 Tosylate
Catalog No. A21434 histamine H3 receptor antagonistPF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
PF-03654746
Catalog No. A21429 histamine H3 receptor antagonistPF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
Camicinal hydrochloride
Catalog No. A21415 motilin receptor agonistCamicinal hydrochloride (GSK962040 hydrochloride) is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. 了解更多 -
CP-409092 hydrochloride
Catalog No. A21397 GABAA receptor partial agonistCP-409092 hydrochloride is a partial agonist of GABAA receptor, with anti-anxiety activity. 了解更多 -
Plecanatide acetate
Catalog No. A21393 GC-C receptor agonistPlecanatide acetate is a guanylate cyclase-C (GC-C) receptor agonist, with an EC50 of 190 nM in T84 cells. Plecanatide acetate shows anti-inflammatory activity in models of murine colitis. 了解更多 -
Batefenterol
Catalog No. A21387 muscarinic receptor antagonist and β2-adrenoceptor agonistBatefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively. 了解更多 -
Foliglurax monohydrochloride
Catalog No. A21384 glutamate receptor 4 modulatorFoliglurax monohydrochloride (PXT002331 monohydrochloride) is a highly selective and potent, brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) , with an EC50 of 79 nM. Antiparkinsonian effect. 了解更多 -
Exendin-4 Acetate
Catalog No. A21378 glucagon-like peptide-1 receptor agonistExendin-4 Acetate (Exenatide acetate), a 39 amino acid peptide, is a long-acting glucagon-like peptide-1 receptor agonist with an IC50 of 3.22 nM. 了解更多 -
SB-277011 dihydrochloride
Catalog No. A21353 dopamine D3 receptor antagonistSB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多 -
SB 242084 hydrochloride
Catalog No. A21349 5-HT2C receptor antagonistSB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多 -
CYT-1010 hydrochloride
Catalog No. A21348 mu-opioid receptor agonistCYT-1010 hydrochloride is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. 了解更多 -
SB290157 trifluoroacetate
Catalog No. A21347 C3a receptor antagonistSB290157 trifluoroacetate is a potent and selective C3a receptor antagonist with an IC50 of 200 nM. 了解更多 -
Dagrocorat
Catalog No. A21312 glucocorticoid receptor agonistDagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. 了解更多 -
Fosdagrocorat
Catalog No. A21303 dissociated glucocorticoid receptor agonistFosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. 了解更多 -
WAY 163909
Catalog No. A21282 5-HT(2C) receptor agonistWAY 163909 is a potent and selective 5-HT(2C) receptor agonist with a Ki of 10.5??1.1 nM. 了解更多 -
Darusentan
Catalog No. A21280 endothelin A (ETA) receptor antagonistDarusentan is a selective endothelin A (ETA) receptor antagonist. 了解更多 -
Lixivaptan
Catalog No. A21279 vasopressin receptor V2 antagonistLixivaptan (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. 了解更多 -
Vortioxetine
Catalog No. A21266 5-HT1A/5-HT1B/5-HT3A/5-HT7 receptor/SERT inhibitorVortioxetine is a inhibitor of 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT, with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively. 了解更多 -
Tipelukast
Catalog No. A21249 leukotriene receptor antagonistTipelukast (KCA 757) is a sulfidopeptide leukotriene receptor antagonist, an orally bioavailable anti-inflammatory agent and used for the treatment of asthma. 了解更多 -
Mavoglurant
Catalog No. A21223 mGlu5 receptor antagonistMavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist, has an IC50 of 30 nM in a functional assay with human mGluR5. 了解更多 -
Capsazepine
Catalog No. A21208 TRPV1 receptorCapsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM. 了解更多 -
ELN-441958
Catalog No. A21207 B1 receptor antagonistELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. 了解更多 -
MDL 105519
Catalog No. A21192 NMDA receptor antagonistMDL 105519 is a potent and selective antagonist of glycine binding to the NMDA receptor. 了解更多 -
Velneperit
Catalog No. A21190 NPY Y5 receptor antagonistVelneperit (S-2367) is a novel neuropeptide Y (NPY) Y5 receptor antagonist. 了解更多 -
CE-224535
Catalog No. A21183 -
PF-4778574
Catalog No. A21157 AMPA receptor positive allosteric modulatorPF-4778574 is a potent AMPA receptor positive allosteric modulator (PAM) that has been shown to enhance cognition in animal models. 了解更多 -
Tezosentan
Catalog No. A21118 endothelin (ET) receptor antagonistTezosentan (RO 610612) is an endothelin (ET) receptor antagonist, with pA2s of 9.5, 7.7 for ETA and ETB receptors, respectively. 了解更多 -
Nelonicline
Catalog No. A21079 neuronal nicotinic receptor agonistNelonicline (ABT-126) is a selective neuronal nicotinic receptor agonist. 了解更多 -
Transcrocetinate disodium
Catalog No. A21051 NMDA receptor antagonistTranscrocetinate disodium, extracted from saffron (Crocus sativus L.), acts as an NMDA receptor antagonist with high affinity. 了解更多
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