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产品 501 到 550 共 2783个

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  1. UAA crosslinker 1

    Catalog No. A19947
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    UAA crosslinker 1 hydrochloride is an amber codon used for non-canonical amino acids (ncAAs) incorporation. The ncAAs can be incorporated into proteins in vivo by making use of the promiscuous activity of certain wildtype and engineered aminoacyl-tRNA synthetases. 了解更多
  2. 3',4'-Dihydroxyflavonol

    Catalog No. A19946
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    3',4'-Dihydroxyflavonol (DiOHF) is an effective antioxidant, which reduces superoxide and improves nitric oxide (NO) function in diabetic rat mesenteric arteries. 了解更多
  3. Oleoylethanolamide

    Catalog No. A19944
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    PPAR-α agonist
    Oleoylethanolamide is a high affinity endogenous PPAR-α agonist, which plays an important role in the treatment of obesity and arteriosclerosis. 了解更多
  4. DCP-LA

    Catalog No. A19943
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    DCP-LA (FR236924), a linoleic acid derivative, selectively and directly activates PKCε. 了解更多
  5. HMN-154

    Catalog No. A19940
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    HMN-154 is a novel benzenesulfonamide anticancer compound; inhibits KB and colon38 cells with IC50 values of 0.0026 and 0.003 μg/mL, respectively. 了解更多
  6. 1,4-Chrysenequinone

    Catalog No. A19937
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    aryl hydrocarbon receptor activator
    1,4-Chrysenequinone, a polycyclic aromatic quinone, acts as an activator of aryl hydrocarbon receptor (AhR). 了解更多
  7. 3,7,4'-Trihydroxyflavone

    Catalog No. A19936
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    3,7,4'-Trihydroxyflavone, isolated from Rhus javanica var. roxburghiana, is a flavonoid with DNA strand-scission activity. 了解更多
  8. Kanosamine hydrochloride

    Catalog No. A19932
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    Kanosamine hydrochloride is an antibiotic which inhibits the growth of plant-pathogenic oomycetes, certain fungi and a few bacterial species. Kanosamine inhibits Phytophthora medicaginis M2913 and Aphanomyces euteiches WI-98 with MICs of 25 and 60 ?g/mL, respectively. 了解更多
  9. 18:0 LYSO-PE

    Catalog No. A19930
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    18:0 LYSO-PE is an agent that can induce [Ca2+]i increase. 了解更多
  10. Ro 22-3581

    Catalog No. A19929
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    Tx synthetase inhibitor
    Ro 22-3581 (4'-(Imidazol-1-yl) acetophenone) is a selective thromboxane (Tx) synthetase inhibitor. 了解更多
  11. SNAP 94847

    Catalog No. A19925
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    MCHR1 antagonist
    SNAP 94847 is a novel, high affinity selective melanin-concentrating hormonereceptor1 (MCHR1) antagonist with (Ki= 2.2 nM, Kd=530 pM), it displays >80-fold and >500-fold selectivity over MCHα1A and MCHD2 receptors respectively. 了解更多
  12. JJKK 048

    Catalog No. A19924
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    MAGL inhibitor
    JJKK 048 is an ultrapotent and highly selective inhibitor of Monoacylglycerol lipase (MAGL). 了解更多
  13. GSK180

    Catalog No. A19923
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    KMO inhibitor
    GSK180 is a selective, competitive, and potent inhibitor of kynurenine-3-monooxygenase (KMO), a key enzyme of tryptophan metabolism (IC50, ~6 nM), but shows negligible activity against other enzymes on the tryptophan pathway. 了解更多
  14. N6-Ethyladenosine

    Catalog No. A19918
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    Adenosine receptor agonist
    N6-Ethyladenosine is an adenosine derivative, acts as a Adenosine receptor agonist, with Kis of 4.9 and 4.7 nM for hA1AR and hA3AR, respectively. 了解更多
  15. A 1120

    Catalog No. A19915
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    RBP4 antagonist
    A 1120, a nonretinoid retinol-binding protein 4 (RBP4) antagonist, has a high affinity with the Ki value of 8.3 nM, which disrupts the interaction between RBP4 and its binding partner transthyretin. 了解更多
  16. JNJ-678

    Catalog No. A19913
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    JNJ-678 (JNJ-53718678) is a novel fusion protein inhibitor in clinical trials for the treatment of respiratory syncytial virus (RSV). 了解更多
  17. NAI-N3

    Catalog No. A19911
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    RNA acylation reagent
    NAI-N3 is a novel RNA acylation reagent that enables RNA purification. 了解更多
  18. Leelamine hydrochloride

    Catalog No. A19910
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    CB1 agonist
    Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees. Leelamine hydrochloride is a cannabinoid receptor type 1 (CB1) agonist and a inhibitor of SREBP1-regulated fatty acid/lipid synthesis in prostate cancer cells that is not affected by androgen receptor status. 了解更多
  19. Auxinole

    Catalog No. A19909
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    TIR1/AFB receptors auxin antagonist
    Auxinole is a potent auxin antagonist of TIR1/AFB receptors, binding TIR1 to block the formation of the TIR1-IAA-Aux/IAA complex and so inhibits auxin-responsive gene expression. 了解更多
  20. Reversan

    Catalog No. A19905
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    MRP1/Pgp inhibitor
    Reversan (CBLC4H10) is a potent and nontoxic multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp) inhibitor. 了解更多
  21. TES-991

    Catalog No. A19902
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    ACMSD inhibitor
    TES-991 is a potent and selective human α?Amino-β-carboxymuconate-ε-semialdehyde Decarboxylase (ACMSD) inhibitor, with an IC50 of 3 nM. 了解更多
  22. Homomangiferin

    Catalog No. A19899
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    Homomangiferin, isolated from the leaves of M. indica L., is mangiferin monomethyl ether. Homomangiferin has important medicinal properties and is widely used to relieve many symptoms, for example coughing and asthma. 了解更多
  23. Deriglidole

    Catalog No. A19898
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    peripheral adrenoceptor antagonist
    Deriglidole is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors. 了解更多
  24. Fmoc-1,6-diaminohexane

    Catalog No. A19892
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    Fmoc-1,6-diaminohexane is an analog of Osw-1 which can be used to treat Alzheimer's disease and cancer, extracted from patent US 20140135279 A1. 了解更多
  25. Chrysin-7-O-β-D-glucuronide

    Catalog No. A19889
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    Chrysin-7-O-β-D-glucuronide is a flavonoid. 了解更多
  26. Nitroxazepine

    Catalog No. A19888
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    serotonin-norepinephrine reuptake inhibitor
    Nitroxazepine is a tricyclic antidepressant (TCA) for the treatment of depression. Nitroxazepine acts as a serotonin-norepinephrine reuptake inhibitor. 了解更多
  27. INF39

    Catalog No. A19887
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    NLRP3 inhibitor
    INF39 is an irreversible and noncytotoxic NLRP3 inhibitor. 了解更多
  28. GSK3186899

    Catalog No. A19884
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    CRK12 inhibitor
    GSK3186899 (DDD-853651) is an inhibitor of cdc-2-related kinase 12 (CRK12), with an EC50 of 1.4 μM for L. donovani in an intra-macrophage assay. 了解更多
  29. STING agonist-3

    Catalog No. A19882
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    STING agonist
    STING agonist-3, compound 3, is a selective and non-nucleotide small-molecule STING agonist, which has durable anti-tumor effect and tremendous potential to improve treatment of cancer. 了解更多
  30. CAY 10465

    Catalog No. A19869
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    AhR agonist
    CAY 10465 is a selective and high-affinity AhR agonist, with a Ki of 0.2 nM, and shows no effect on estrogen receptor (Ki >100000 nM). 了解更多
  31. 2-HBA

    Catalog No. A19867
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    NQO1 inducer
    2-HBA is a potent inducer of NAD(P)H:quinone acceptor oxidoreductase 1 (NQO1) which can also activate caspase-3 and caspase-10. 了解更多
  32. AZD7594

    Catalog No. A19866
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    glucocorticoid receptor modulator
    AZD7594 is a potent selective nonsteroidal glucocorticoid receptor modulator, with an IC50 of 0.9 nM. 了解更多
  33. Nosantine racemate

    Catalog No. A19864
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    IL-2 inducer
    Nosantine racemate is the racemate of Nosantine. Nosantine is an inducer of IL-2 or enhancer of IL-2 induction by phytohemagglutinin (PHA). 了解更多
  34. GR 159897

    Catalog No. A19862
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    NK2 antagonist
    GR 159897 is a highly potent, selective, competitive, brain-penetrated non-peptide antagonist at tachykinin NK2 receptors, inhibits binding of [3H]GR100679 to hNK2-CHO cells and rat colon membranes with pKis of 9.51 and 10, respectively. Antagonizes bronchoconstriction, with anxiolytic-like activity. 了解更多
  35. QF0301B

    Catalog No. A19856
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    α1 adrenergic receptor antagonist
    QF0301B is an α1 adrenergic receptor antagonist and a low α2 adrenoceptor, 5-HT2A, and histamine H1 receptor blocker. 了解更多
  36. Statine

    Catalog No. A19855
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    Statine is an unusual amino acid that occurs twice in the sequence of pepstatin, a protease inhibitor that is active against pepsin and other acid proteases. 了解更多
  37. VH032-thiol-C6-NH2

    Catalog No. A19847
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    VH032-thiol-C6-NH2 (VHL Ligand-Linker Conjugates 14) is a synthesized E3 ligase ligand-linker conjugate that incorporates the VH032 based VHL ligand and a linker used in PROTAC technology. 了解更多
  38. CGP71683 hydrochloride

    Catalog No. A19844
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    neuropeptide Y5 receptor antagonist
    CGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes. 了解更多
  39. L-368,899 hydrochloride

    Catalog No. A19843
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    oxytocin receptor antagonist
    L-368,899 hydrochloride is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively, used as a tocolytic agent. 了解更多
  40. VU0467154

    Catalog No. A19842
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    mAChR modulator
    VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor (mAChR), potentiating the response to ACh with pEC50s of 7.75, 6.2 and 6 for rat, human and cynomolgus monkey M4 receptor, respectively. 了解更多
  41. AMPD2 inhibitor 1

    Catalog No. A19839
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    AMPD2 inhibitor
    AMPD2 inhibitor 1 is an adenosine monophosphate deaminase 2 (AMPD2) inhibitor, used in the research of sugar craving, salt craving, umami craving, and addictions including drug, tobacco, nicotine and alcohol addictions. 了解更多
  42. Aristeromycin

    Catalog No. A19832
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    AHCY inhibitor
    Aristeromycin, an adenosine analog, is an antibiotic and a potent S-adenosylhomocysteine hydrolase (AHCY) inhibitor. 了解更多
  43. ARQ 531

    Catalog No. A19823
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    BTK inhibitor
    ARQ 531 is a reversible non-covalent inhibitor of Bruton??s Tyrosine Kinase (BTK), with IC50s of 0.85 nM and 0.39 nM for WT-BTK and C481S-BTK, respectively. 了解更多
  44. PD 90780

    Catalog No. A19821
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    NGF antagonist
    PD 90780 is a non peptide antagonist of nerve growth factor (NGF) binding to the P75 NGF receptor, inhibits NGF-p75 NTR interaction with IC50s values of 23.1 ?M and 1.8 ?M in PC12 cells and PC12 nnr5 cells, respectively . 了解更多
  45. S-1-Propenyl-L-cysteine

    Catalog No. A19819
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    S-1-Propenyl-L-cysteine is a stereoisomer of S-allyl-l-cysteine, extracted from garlic, with immunomodulatory effects and reduces blood pressure in a hypertensive animal model. 了解更多
  46. BCECF

    Catalog No. A19817
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    fluorescent agent
    Cardiogreen is fluorescent agent with low toxicity has been widely used in medical diagnostics. 了解更多
  47. LY2955303

    Catalog No. A19816
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    RARγ antagonist
    LY2955303 is a potent and selective retinoic acid receptor gamma (RARγ) antagonist with a Ki of 1.09 nM. 了解更多
  48. CG-806

    Catalog No. A19814
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    FLT3/BTK inhibitor
    CG-806 is an orally active, potent and non-covalent pan-FLT3/pan-BTK inhibitor with an IC50 of 0.08 μM for FLT3. CG-806 has an IC50 of 11 nM against FLT3 wild type (WT)-transfected Ba/F3 cells. 了解更多
  49. RT-NH2

    Catalog No. A19813
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    RealThiol prototype
    RT-NH2 is a RealThiol prototype without the carboxylic acid groups. RT-NH2 is fairly hydrophobic and cannot distribute in the nucleus, which is a hallmark of protein binding for fluorescent probe. 了解更多
  50. EP1-antanoist-1

    Catalog No. A19810
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    EP1 antagonist
    EP1-antanoist-1 is a EP1 antagonist with a pKi of 7.54 and an pIC50 of 8.5. 了解更多

产品 501 到 550 共 2783个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

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