“receptor”的搜索结果

产品 501 到 550 共 1701个

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  1. Terutroban

    Catalog No. A20884
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    thromboxane-prostaglandin receptor antagonist
    Terutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多
  2. Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  3. Clopidogrel thiolactone

    Catalog No. A20862
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    P2Y12 receptor inhibitor
    Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent. 了解更多
  4. Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  5. APNEA

    Catalog No. A20845
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    A3 adenosine receptor agonist
    APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. 了解更多
  6. SYM2206

    Catalog No. A20843
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    AMPA receptor antagonist
    SYM 2206 is a novel, potent, non-competitive AMPA receptor antagonist. 了解更多
  7. Haloperidol hydrochloride

    Catalog No. A18304
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    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  8. Setiptiline

    Catalog No. A18090
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    serotonin receptor antagonist
    Setiptiline(Org-8282) is a serotonin receptor antagonist. 了解更多
  9. Quinagolide hydrochloride

    Catalog No. A18038
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    dopamine D2 receptor agonist
    Quinagolide hydrochloride is a selective dopamine D2 receptor agonist, also is a prolactin inhibitor. 了解更多
  10. Pyrantel tartrate

    Catalog No. A18032
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    antinematodal thiophene nicotinic receptor agonist
    Pyrantel tartrate is an antinematodal thiophene nicotinic receptor agonist and can elicit spastic muscle paralysis in parasitic worms due to prolonged activation of the excitatory nicotinic acetylcholine (nACh) receptors on body wall muscle. 了解更多
  11. Oxytocin

    Catalog No. A17988
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    oxytocin receptor ligand
    Oxytocin (α-Hypophamine) is a mammalian neurohypophysial hormone; its actions are mediated by specific, high-affinity oxytocin receptors; ligand of oxytocin receptor. 了解更多
  12. (Z)-Thiothixene

    Catalog No. A17891
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    Serotonergic receptor antagonist
    (Z)-Thiothixene is an antagonist of serotonergic receptor extracted from patent US 20150141345 A1. 了解更多
  13. Sunitinib

    Catalog No. A17858
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    multi-targeted receptor tyrosine kinase inhibitor
    Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase inhibitor with IC50s of 80 nM and 2 nM for VEGFR2 and PDGFRβ, respectively. 了解更多
  14. Trimethobenzamide hydrochloride

    Catalog No. A17648
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    D2 receptor blocker
    Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多
  15. Ziprasidone hydrochloride

    Catalog No. A16790
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    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  16. WAY-100635 Maleate

    Catalog No. A16787
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    5-HT1A receptor antagonist
    WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. 了解更多
  17. Tamoxifen

    Catalog No. A16738
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    selective estrogen receptor modulator (SERM)
    Tamoxifen (ICI 47699) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells. 了解更多
  18. SB-334867 free base

    Catalog No. A16695
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    orexin OX1 receptor antagonist
    SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. 了解更多
  19. (R)-Baclofen

    Catalog No. A16680
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    GABAB receptor agonist
    (R)-Baclofen(STX209) is a selective GABAB receptor agonist. 了解更多
  20. Ifenprodil tartrate

    Catalog No. A16583
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    NMDA receptor antagonist
    Ifenprodil tartrate is the atypical N-methyl-D-aspartate (NMDA) receptor antagonist, inhibits NMDA-induced currents at NR1A/NR2B receptors with high affinity (IC50 = 0.34 μM). 了解更多
  21. Dexamethasone acetate

    Catalog No. A16494
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    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. 了解更多
  22. Varenicline Tartrate

    Catalog No. A11618
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    nicotinic receptor partial agonist
    Varenicline Tartrate(CP 526555;Champix) is a nicotinic receptor partial agonist; it stimulates nicotine receptors more weakly than nicotine itself does. 了解更多
  23. Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  24. SB 271046 Hydrochloride

    Catalog No. A11573
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    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  25. SU14813 maleate

    Catalog No. A11556
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    multi-targeted receptor tyrosine kinases inhibitor
    SU14813 maleate is a multi-targeted receptor tyrosine kinases inhibitor with IC50s of 50, 2, 4, 15 nM for VEGFR2, VEGFR1, PDGFRβ and KIT. 了解更多
  26. Rivanicline oxalate

    Catalog No. A11544
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    neuronal nicotinic receptor agonist
    Rivanicline oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 3.6 μM). 了解更多
  27. Olcegepant

    Catalog No. A11512
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    CGRP1 receptor
    Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. 了解更多
  28. Montelukast sodium

    Catalog No. A11490
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    CysLT1 receptor antagonist
    Montelukast (sodium) (MK0476) is a potent, selective CysLT1 receptor antagonist. 了解更多
  29. JDTic

    Catalog No. A11468
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    κ-opioid receptor antagonist
    JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. 了解更多
  30. IRAK inhibitor 3

    Catalog No. A11457
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    IL-1 receptor-associated kinase (IRAK) kinase modulator
    IRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator extracted from patent WO2008030579 A2. 了解更多
  31. IRAK inhibitor 2

    Catalog No. A11456
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    interleukin-1 receptor associated kinase inhibitor
    IRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多
  32. CGS 21680

    Catalog No. A11354
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    adenosine A2A receptor agonist
    CGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. 了解更多
  33. Cabozantinib S-malate

    Catalog No. A11349
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    multiple receptor tyrosine kinases inhibitor
    Cabozantinib S-malate (XL184 S-malate) is a potent multiple receptor tyrosine kinases inhibitor that inhibits VEGFR2, c-Met, Kit, Axl and Flt3 with IC50s of 0.035, 1.3, 4.6, 7 and 11.3 nM, respectively. 了解更多
  34. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多
  35. RF9

    Catalog No. A12944
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    Neuropeptide FF receptor antagonist
    RF9 is a potent and selective Neuropeptide FF receptor antagonist, with Kis of 58??5 and 75??9 nM for hNPFF1R and hNPFF2R, respectively. 了解更多
  36. Lesopitron dihydrochloride

    Catalog No. A12950
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    5-HT1A receptor agonist
    Lesopitron dihydrochloride is a full and selective 5-HT1A receptor agonist with IC50 of 125 nM in rat hippocampal membranes. 了解更多
  37. CP-96486

    Catalog No. A12471
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    LTD4/PAF receptor antagonist
    CP-96486 is a potent and orally active leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor antagonist with Kis of 20 and 24 nM, respectively. 了解更多
  38. FR167344 free base

    Catalog No. A12964
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    nonpeptide bradykinin receptor B2 antagonist
    FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. 了解更多
  39. Pancopride

    Catalog No. A12967
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    5-HT3 receptor antagonist
    Pancopride is a new potent and selective 5-HT3 receptor antagonist. 了解更多
  40. Amelubant

    Catalog No. A12968
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    LTB4 receptor antagonist
    Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist. 了解更多
  41. RPR104632

    Catalog No. A13385
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    NMDA receptor antagonist
    RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. 了解更多
  42. Foropafant

    Catalog No. A13388
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    PAF receptor antagonist
    Foropafant (SR27417) highly potent, competitive, selective and orally active antagonist of platelet-activating factor (PAF) receptor. 了解更多
  43. AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  44. Edicotinib

    Catalog No. A13008
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    CSF-1 receptor inhibitor
    Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease. 了解更多
  45. GLPG0187

    Catalog No. A13423
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    Integrin receptor antagonist
    GLPG0187 is a broad spectrum integrin receptor antagonist with antitumor activity; inhibits αvβ1-integrin with an IC50 of 1.3 nM. 了解更多
  46. LED209

    Catalog No. A12219
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    bacterial receptor QseC inhibitor
    LED209 is a potent small molecule inhibitor of bacterial receptor QseC, is a potent prodrug that is highly selective for QseC. 了解更多
  47. GV-196771A

    Catalog No. A13438
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    NMDA receptor antagonist
    GV-196771A is the sodium salt form of GV196771, is an NMDA receptor antagonist. 了解更多
  48. Tiotropium Bromide

    Catalog No. A10934
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    muscarinic acetylcholine receptor (mAChR) antagonist
    Tiotropium Bromide (BA679 BR) is a muscarinic acetylcholine receptor (mAChR) antagonist that blocks the binding of the acetylcholine ligand and subsequent opening of the ligand-gated ion channel. 了解更多
  49. Valsartan

    Catalog No. A10962
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    angiotensin II receptor antagonist
    Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure. 了解更多
  50. Zafirlukast

    Catalog No. A11004
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    LTD4 receptor antagonist
    Zafirlukast is a potent orally active leukotriene D4 (LTD4) receptor antagonist. 了解更多

产品 501 到 550 共 1701个

每页
页面:
  1. 9
  2. 10
  3. 11
  4. 12
  5. 13

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