微信关注
China
Total item
Cart Subtotal
￥ 0.00 “receptor”的搜索结果
-
Ziprasidone hydrochloride monohydrate
Catalog No. A11008 5-HT (serotonin) and dopamine receptor antagonistZiprasidone hydrochloride monohydrate (CP 88059 hydrochloride monohydrate) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多 -
Acamprosate calcium
Catalog No. A11308 GABA receptor agonistAcamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. 了解更多 -
Sitaxsentan
Catalog No. A11565 ETA receptor antagonistSitaxsentan (IPI 1040; TBC-11251) is a selective endothelin A (ETA) receptor antagonist. Antihypertensive. Sitaxsentan is used in treatment of chronic heart failure. 了解更多 -
Elacestrant
Catalog No. A12244 Estrogen receptor degraderElacestrant (RAD1901) is an orally available selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. 了解更多 -
DW-1350
Catalog No. A12250 -
PRX933 hydrochloride
Catalog No. A12261 5-HT2c receptor agonistPRX933 hydrochloride is a 5-HT2c receptor agonist extracted from patent WO 2014140631 A1. 了解更多 -
5-HT4 antagonist 1
Catalog No. A12268 5-HT4 receptor antagonist5-HT4 antagonist 1 is a 5-HT4 receptor antagonist with a pKi of 9.6. 了解更多 -
lumateperone Tosylate
Catalog No. A12279 5-HT2A receptor antagonistLumateperone Tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a SERT blocker (Ki = 61 nM). 了解更多 -
Pipequaline
Catalog No. A12551 partial benzodiazepine receptor agonistPipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. 了解更多 -
Endothelin Mordulator 1
Catalog No. A13040 endothelin receptor modulatorEndothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多 -
Veralipride
Catalog No. A13132 D2 receptor antagonistVeralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. 了解更多 -
Chlorantraniliprole
Catalog No. A13214 Chlorantraniliprole is an insecticide that potently and selectively activates insect ryanodine receptor, with EC50s of 40 nM and 50 nM for Drosophila melanogaster and H. virescens ryanodine receptor, and ?300-fold more potent than that in the mouse myoblast cell line, C2C12 (EC50, 14 μM). 了解更多 -
Mozavaptan
Catalog No. A16622 nonpeptide vasopressin V2 receptor antagonistMozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM. 了解更多 -
Tripelennamine hydrochloride
Catalog No. A16767 H1-receptor antagonistTripelennamine hydrochloride, a H1-receptor antagonist, is a psychoactive drug and member of the pyridine andethylenediamine classes that is used as an antipruritic and first-generation antihistamine. 了解更多 -
Pirenzepine dihydrochloride
Catalog No. A17916 M1 muscarinic receptor antagonistPirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist. 了解更多 -
Norepinephrine
Catalog No. A11306 β1-selective adrenergic receptor agonistNorepinephrine (Levarterenol; L-Noradrenaline) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. 了解更多 -
CAY10471 Racemate
Catalog No. A11760 Prostaglandin D2 receptor CRTH2 antagonistCAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多 -
Darenzepine
Catalog No. A12333 muscarinic receptor inhibitorDarenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多 -
MRK-016
Catalog No. A12046 GABAA α5 receptor agonistMRK-016 is a selective, orally bioavailable inverse agonist of GABAA α5 receptor, with an EC50 of 3 nM for GABAA α5, and Kis of 0.83, 0.85, 0.77?and 1.4?nM for human?GABAA?α1β3γ2, GABAA?α2β3γ2, GABAA?α3β3γ2, and GABAA?α5β3γ2, respectively; MRK-016 also readily penetrates the CNS. 了解更多 -
Tecadenoson
Catalog No. A13302 A1 adenosine receptor agonistTecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多 -
Lu AF21934
Catalog No. A12140 mGlu4 receptor modulatorLu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多 -
Beperidium iodide
Catalog No. A12382 competitive antagonistic effect against acetylcholine receptorBeperidium iodide shows a competitive antagonistic effect against acetylcholine receptor with a pA2 of 7.93. 了解更多 -
GSK1059865
Catalog No. A12401 -
Dexamethasone palmitate
Catalog No. A18453 Dexamethasone palmitate (DXP) is a prodrug of Dexamethasone, which is a glucocorticoid receptor agonist. Dexamethasone palmitate (DXP) has a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Anti-inflammatory agent. 了解更多 -
ROR agonist-1
Catalog No. A18569 ROR 激动剂ROR agonist-1 is a potent and orally bioavailable inverse agonist of the retinoic acid receptor-related orphan receptor C2 (RORC2), inhibition of IL-17A production from human primary TH 17 cells with a pIC50 of 7.5. 了解更多 -
PROTAC ERRα Degrader-2
Catalog No. A18904 ERRa degraderPROTAC ERRalpha Degrader-2 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRalpha Degrader-2 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多 -
Semaglutide
Catalog No. A18908 GLP-1 receptor agonistSemaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多 -
PROTAC ERRα Degrader-1
Catalog No. A18910 ERRα DegraderPROTAC ERRα Degrader-1 comprises a MDM2 ligand binding group, a linker and an estrogen-related receptor alpha (ERRa) binding group. PROTAC ERRα Degrader-1 is an estrogen-related receptor alpha (ERRa) degrader. 了解更多 -
AZD2906
Catalog No. A18936 glucocorticoid receptor agonistAZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多 -
PF-05231023
Catalog No. A18949 FGF21-receptor agonistPF-05231023, a long-acting fibroblast growth factor 21 (FGF21) analog, is a FGF21-receptor agonist, suitable for development as a potential treatment for T2DM. 了解更多 -
GSK1521498 free base
Catalog No. A18994 μ-opioid receptor antagonistGSK1521498 free base is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 free base is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多 -
Asoprisnil
Catalog No. A19030 Progesterone receptor modulatorAsoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. 了解更多
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
FILTER BY:
购物选项
- 分类
-
- Epigenetics (2)
- Apoptosis (9)
- Protein Tyrosine Kinases (21)
- Angiogenesis (15)
- JAK / Stat (7)
- Cell Cycle (1)
- Cytoskeleton (2)
- Cell Metabolism (31)
- Autophagy Signaling (11)
- Immunology & Inflammation (31)
- GPCR / G Protein (493)
- TGF-β / Smad (6)
- Neuronal Signaling (101)
- Proteases (2)
- Microbiology (4)
- Membrane Transporters/Ion Channels (26)
- Endocrinology / Hormones (88)
- PROTACs (5)
- Others (12)
- Natural Products (2)
- Ready to Use Solution (71)
- Products On Sale (131)
- Recombinant Proteins (100)
- Neurotrophins (7)
- Growth Factors (16)
- Hormones (1)
- Monoclonal Antibodies (27)
- Natural Proteins (1)
- Viral Antigens (5)
- CD Antigens (3)
- Cytokines (78)
- Enzymes (42)
- COVID-19 Related Products (1)
- 作用机制
-
- Inhibitor (抑制剂) (109)
- Agonist (激动剂) (292)
- Antagonist (拮抗剂) (471)
- Activator (激活剂) (2)
- Modulator (调节剂) (55)
- Blocker (阻断剂) (13)
- Degrader (降解剂) (7)
- Potentiator (增强剂) (2)
- 靶点
-
- A1 adenosine receptor (1)
- A3 adenosine receptor (1)
- Aurora A (1)
- Aurora B (1)
- Aurora C (1)
- COX-1 (1)
- COX-2 (1)
- CSF1R (1)
- CXCL8 (1)
- CXCR1 (1)
- CXCR2 (1)
- CXCR4 (2)
- Ecdysone receptor (1)
- Histamine H1 receptor (1)
ADOOQ 产品质量保证
We promise all products to perform as described.