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Methiothepin mesylate
Catalog No. A19599 5-HT2 receptor antagonistMethiothepin mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C). 了解更多 -
N6-Cyclopentyladenosine
Catalog No. A19595 Adenosine A1 receptor agonistN6-Cyclopentyladenosine (CPA) is a selective Adenosine A1 receptor agonist, with Ki values of 2.3 nM, 790 nM and 43 nM for human A1, A2A and A3 receptors, respectively. 了解更多 -
N-Acetyl-5-hydroxytryptamine
Catalog No. A19581 Melatonin precursorN-Acetyl-5-hydroxytryptamine is a Melatonin precursor, and that it can potently activate TrkB receptor. 了解更多 -
SNIPER(BRD)-1
Catalog No. A19579 SNIPER inhibitorSNIPER(BRD4)-1 is a specific and nongenetic inhibitor of apoptosis protein (IAP)-dependent protein eraser (SNIPER) which acts as a protein degradation inducer of bromodomain-containing protein 4 (BRD4). 了解更多 -
4-(6-Bromo-2-benzothiazolyl)benzenamine
Catalog No. A19574 β-amyloid PET tracer4-(6-Bromo-2-benzothiazolyl)benzenamine is a β-amyloid PET (positron emission tomography) tracer that can be used in the diagnosis of neurological diseases, such as Alzheimer's and Down's syndrome. 了解更多 -
DL-Mevalonolactone
Catalog No. A19571 DL-Mevalonolactone ((±)-Mevalonolactone;Mevalolactone) is the δ-lactone form of mevalonic acid, a precursor in the mevalonate pathway. DL-Mevalonolactone (Mevalonolactone) decreases mitochondrial membrane potential (???m), NAD(P)H content and the capacity to retain Ca2+ in the brain, besides inducing mitochondrial swelling. 了解更多 -
2,2,5,7,8-Pentamethyl-6-Chromanol
Catalog No. A19565 2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol). 2,2,5,7,8-Pentamethyl-6-Chromanol has potent androgen receptor (AR) signaling modulation and anti-cancer activity against prostate cancer cell lines. 了解更多 -
BAY-678 racemate
Catalog No. A19564 HNE inhibitorBAY-678 racemate is a racemate of BAY-678. BAY-678 is an orally bioavailable, highly potent, selective and cell-permeable inhibitor of human neutrophil elastase (HNE), with an IC50 of 20 nM. BAY-678 is also nominated as a chemical probe to the public via the Structural Genomics Consortium (SGC). 了解更多 -
Veratryl alcohol
Catalog No. A19553 Veratryl alcohol (3,4-Dimethoxybenzenemethanol), a secondary metabolite of some lignin degrading fungi, is commonly used nonphenolic substrate for assaying ligninolytic activity. 了解更多 -
ATP synthase inhibitor 1
Catalog No. A19550 F1/FO-ATP synthase complex inhibitorATP synthase inhibitor 1 is a potent inhibitor of c subunit of the F1/FO-ATP synthase complex, inhibits mitochondrial permeability transition pore (mPTP) opening, does not affect ATP levels. 了解更多 -
Amibegron hydrochloride
Catalog No. A19549 β3-adrenoceptor agonistAmibegron hydrochloride is a selective β3-adrenoceptor agonist, with an EC50 of 3.5 nM for β-adrenoceptor in rat colon; Amibegron hydrochloride has anxiolytic and antidepressant activity. 了解更多 -
24-Norursodeoxycholic acid
Catalog No. A19546 24-norursodeoxycholic acid (norUDCA) is a side chain-shortened C23 homologue of UDCA and has shown potent anti-cholestatic, anti-inflammatory and anti-fibrotic properties. 了解更多 -
DSP-4 hydrochloride
Catalog No. A19539 DSP-4 hydrochloride (Neurotoxin DSP 4 hydrochloride) is a highly selective neurotoxin and readily passes the blood-brain barrier with neurotoxic effects on noradrenergic neurons of adult and developing rats, can be used for the temporary selective degradation of the central and peripheral noradrenergic neurons, mainly those from the locus coeruleus (LC). 了解更多 -
BMS-816336
Catalog No. A19528 11β-HSD1 inhibitorBMS-816336 is a novel, potent and orally bioavailable inhibitor against human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme with an IC50 of 3.0 nM. 了解更多 -
Ipsalazide
Catalog No. A19511 sulfasalazine analogIpsalazide is a novel sulfasalazine analog designed to release 5-aminosalicylic acid and a nontoxic carrier molecule in the gastrointestinal tract. 了解更多 -
Octaaminocryptand 1
Catalog No. A19497 -
N6-Methyladenosine 5'-monophosphate disodium salt
Catalog No. A19489 rat adenylate kinase II inhibitorN6-Methyladenosine 5'-monophosphate disodium salt is an activator of glycogen phosphorylase b, with a Ka value of 22 ?M. N6-Methyladenosine 5'-monophosphate disodium salt is a non-competitive rat adenylate kinase II inhibitor. 了解更多 -
Apararenone
Catalog No. A19480 mineralocorticoid receptor antagonistApararenone (MT-3995) is a novel non-steroidal mineralocorticoid receptor antagonists under development for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis. 了解更多 -
5-Iodo-indirubin-3'-monoxime
Catalog No. A19479 GSK-3β, CDK5/P25 and CDK1/cyclin B inhibitor5-Iodo-indirubin-3'-monoxime is a potent GSK-3β, CDK5/P25 and CDK1/cyclin B inhibitor, competing with ATP for binding to the catalytic site of the kinase, with IC50s of 9, 20 and 25 nM, respectively. 了解更多 -
WAY127093B racemate
Catalog No. A19474 PDE-4 inhibitorWAY127093B racemate is the racemate of WAY127093B. WAY127093B is a novel, orallyactive phosphodiesterase IV inhibitor in guinea pigs and rats. 了解更多 -
Sinefungin
Catalog No. A19473 virion mRNA(guanine-7-)-methyltransferase inhibitorSinefungin is a potent inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral multiplication. 了解更多 -
Nacubactam
Catalog No. A19471 non-β-lactam-β-lactamase inhibitorNacubactam (OP0595 free acid) is a potent non-β-lactam-β-lactamase inhibitor with activity against class A and class C β-lactamases. 了解更多 -
Indirubin-3'-monoxime-5-sulphonic acid
Catalog No. A19470 CDK1, CDK5, and GSK-3βinhibitorIndirubin-3'-monoxime-5-sulphonic acid is a potent and selective inhibitor of CDK1, CDK5, and GSK-3β with IC50s of 5 nM, 7 nM, and 80 nM, respectively. 了解更多 -
SJ000291942
Catalog No. A19460 BMP activatorSJ000291942 is an activator of the canonical bone morphogenetic proteins (BMP) signaling pathway. BMPs are members of the transforming growth factor beta (TGFβ) family of secreted signaling molecules. 了解更多 -
Toyocamycin
Catalog No. A19458 XBP1 inhibitorToyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage, with an IC50 of 80 nM. 了解更多 -
(±)-Befunolol
Catalog No. A19441 -
Spastazoline
Catalog No. A19432 spastin inhibitorSpastazoline is a potent and selective spastin (a microtubule-severing AAA protein) inhibitor, with an IC50 of 99 nM for Human spastin. Spastazoline shows no effect on ATPase activity of a recombinant human VPS4. 了解更多 -
Aminooxyacetic acid hemihydrochloride
Catalog No. A19408 MAS inhibitorAminooxyacetic acid hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. 了解更多 -
NO-prednisolone
Catalog No. A19400 NO-prednisolone is a nitric oxide (NO)-releasing derivative of Prednisolone. NO-prednisolone potently stimulates IL-10 production in vivo. 了解更多 -
D-Ala-Lys-AMCA
Catalog No. A19387 D-Ala-Lys-AMCA is a known proton-coupled oligopeptide transporter 1 (PEPT1) substrate that emits blue fluorescence. D-Ala-Lys-AMCA may be transported into liver cancer cells and Caco-2 cells based on fluorescence analysis. 了解更多 -
AmPEG6C2-Aur0131
Catalog No. A19363 drug-linker conjugate for ADCAmPEG6C2-Aur0131 is a drug-linker conjugate for ADC (anti-CXCR4 ADC) with potent antitumor activity by using Aur0131 (an auristatin microtubule inhibitor), linked via the non-cleavable linker AmPEG6C2. 了解更多 -
β-Apo-13-carotenone
Catalog No. A19360 antagonist of RXRαβ-Apo-13-carotenone (D'Orenone) is a naturally occurring β-apocarotenoid functioned as an antagonist of RXRα. 了解更多 -
Pro-xylane
Catalog No. A19359 GAGs biosynthesisPro-xylane (Hydroxypropyl tetrahydropyrantriol) is a biologically active C-glycoside in aqueous media, acts as an activator of glycosaminoglycans (GAGs) biosynthesis. 了解更多 -
Ifenprodil glucuronide
Catalog No. A19353 platelet aggregation inhibitorIfenprodil glucuronide is a derivative of Ifenprodil. Ifenprodil is a vasodilator and an inhibitor of platelet aggregation, and Ifenprodil glucuronide has no effect on platelet aggregation and arterial contraction. 了解更多 -
Secoisolariciresinol diglucoside
Catalog No. A19345 Secoisolariciresinol diglucoside ((S,S)-SDG) is a major component of the lignans in flaxseed, scavenges free radical, with potent antioxidant activity. 了解更多
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