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Blarcamesine (AVex-73)
Catalog No. A21095 muscarinic M1 agonistBlarcamesine, also known as AVex-73 and AE-37, is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease. It is an σ receptor ligand. 了解更多 -
Pridopidine
Catalog No. A22009 D2R antagonistPridopidine, a dopamine (DA) stabilizer, acts as a low affinity dopamine D2 receptor (D2R) antagonist. 了解更多 -
Calcitriol Impurities D
Catalog No. A20825 impurity of CalcitriolCalcitriol Impurities D is the impurity of Calcitriol, Calcitriol is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). 了解更多 -
GSK2798745
Catalog No. A20799 TRPV4 ion channel blockerGSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively. 了解更多 -
WAY-204688
Catalog No. A20757 NF-κB inhibitorWAY-204688 is an estrogen receptor (ER-α) selective, orally active inhibitor of NF-κB transcriptional activity with an IC50 of 122?±?30 nM for NF-κB-luciferase (NF-κB-luc) in HAECT-1 cells. 了解更多 -
GSK180736A
Catalog No. A20736 GRK2 inhibitorGSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM. 了解更多 -
Fezolinetant
Catalog No. A20706 NK3R antagonistFezolinetant is an antagonist of the neurokinin 3 receptor (NK3R), used for the treatment of menopausal hot flushes. 了解更多 -
Setmelanotide
Catalog No. A20689 MC4R agonistSetmelanotide (RM-493; BIM-22493; IRC-022493) is a selective melanocortin 4 receptor (MC4R) agonist with EC50s of 0.27 nM and 0.28 nM for human and rat MC4R, respectively. 了解更多 -
CCR2-RA-[R]
Catalog No. A20644 CCR2 antagonistCCR2-RA-[R] is an allosteric antagonist of the C-C chemokine receptor type 2 (CCR2) with an IC50 of 103 nM. 了解更多 -
Saroglitazar
Catalog No. A20636 PPAR agonistSaroglitazar is a novel peroxisome proliferator-activated receptor (PPAR) agonist with predominant PPARα and moderate PPARγ activity with EC50 values of 0.65 pM and 3 nM in HepG2 cells, respectively. 了解更多 -
Calcitriol Impurities A
Catalog No. A20633 Calcitriol Impurities A is the impurity of Calcitriol, Calcitriol is the hormonally active form of vitamin D, Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor (VDR). 了解更多 -
Azeliragon
Catalog No. A20622 RAGE inhibitorAzeliragon (TTP488) is an orally bioavailable inhibitor of the receptor for advanced glycation end products (RAGE) in development as a potential treatment to slow disease progression in patients with mild Alzheimer??s disease (AD). Azeliragon also can cross the blood-brain barrier (BBB). 了解更多 -
GSK682753A
Catalog No. A20519 EBI2 inverse agonistGSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2) with an IC50 of 53.6 nM. 了解更多 -
Mivotilate
Catalog No. A20504 AhR activatorMivotilate is a nontoxic, potent activator of the aryl hydrocarbon receptor (AhR), and acts as a hepatoprotective agent. 了解更多 -
Agmatine sulfate
Catalog No. A20485 NO synthase inhibitorAgmatine sulfate exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide synthesis. It is an endogenous agonist at imidazoline receptor and a NO synthase inhibitor. 了解更多 -
CCR2 antagonist 3
Catalog No. A20467 -
(-)-(S)-Equol
Catalog No. A20465 (-)-(S)-Equol is a high affinity ligand for estrogen receptor β with a Ki of 0.73 nM. 了解更多 -
Trifarotene
Catalog No. A20458 RAR agonistTrifarotene (CD5789) is a retinoic acid receptor (RAR) agonist with Kdapp of 2, 15 and 500 nM for RARγ, RARβ and RARα, respectively. 了解更多 -
TCS-OX2-29
Catalog No. A20457 OX2R antagonistTCS-OX2-29 is a potent, high affinities and selective orexin-2 receptor (OX2R) antagonist with an IC50 value of 40 nM and a pKI value of 7.5. TCS-OX2-29 displays ~250-fold selectivity for OX2 over OX1. 了解更多 -
WAY-200070
Catalog No. A20442 ERRβ agonistWAY-200070 is a selective estrogen receptor β (ERRβ) agonist with an IC50 of 2.3 nM. 了解更多 -
Nitromifene
Catalog No. A20417 -
LXRβ agonist-2
Catalog No. A20405 LXRβ agonistLXRβ agonist-2 is a highly potent and β-selective liver X receptor (LXRβ) agonist with EC50 of 7 nM, displays 28.5-fold selectivity over LXRα (EC50=200 nM) and used in the treatment of atherosclerosis. 了解更多 -
BMS-986020
Catalog No. A20393 LPA1 antagonistBMS-986020 is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. 了解更多 -
Adenosine antagonist-1
Catalog No. A20383 AA3R antagonistAdenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist. 了解更多 -
Fisogatinib
Catalog No. A20354 FGFR4 inhibitorFisogatinib (BLU-554) is a potent, highly selective and orally active fibroblast growth factor receptor 4 (FGFR4) inhibitor with an IC50 of 5 nM. 了解更多 -
5-HT1A modulator 1
Catalog No. A20319 5-HT1A modulator5-HT1A modulator 1 displays very high affinities for the 5HT1A, adrenergic α1 and dopamine D2 receptor with IC50s of 2 ±0.3 nM, 10 ± 3 nM and 40 ±9 nM, respectively. 了解更多 -
CNS-5161 hydrochloride
Catalog No. A20308 NMDA ion-channel antagonistCNS-5161 hydrochloride is a novel NMDA ion-channel antagonist that interacts with the NMDA receptor/ion channel site to produce a noncompetitive blockade of the actions of glutamate. 了解更多 -
SSTR5 antagonist 1
Catalog No. A20218 SSTR5 antagonistSSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a). 了解更多
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