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Runcaciguat
Catalog No. A20200 soluble guanylate cyclase stimulatorRuncaciguat is an orally active stimulator of soluble guanylate cyclase, and is used in the research of cardiovascular and renal diseases combined with selective partial adenosine A1 receptor agonists. 了解更多 -
Oral antiplatelet agent 1
Catalog No. A20188 Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro as well as antithrombotic efficacy in a rat model. P2Y receptor antagonist. 了解更多 -
GRK2-IN-1
Catalog No. A20131 GRKs-IN-1, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=30 nM) and GRK5 (IC50=7.1 μM). GRKs-IN-1 is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine. 了解更多 -
GPR40/FFAR1 modulator 1
Catalog No. A20129 GPR40/FFAR1 agonistGPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1). 了解更多 -
RIP2 Kinase Inhibitor 3
Catalog No. A20109 RIP2 inhibitorRIP2 Kinase Inhibitor 3 is a highly potent and selective inhibitor of receptor interacting protein-2 (RIP2) Kinase with an IC50 of 1 nM . 了解更多 -
ML 145
Catalog No. A19953 GPR35/CXCR8 antagonistML 145 is a selective GPR35/CXCR8 antagonist with an IC50/EC50 of 20.1 nM, but not for the related GPR55 orphan receptor. GPR35 is expressed by various cells of the immune system and it may has potential as a therapeutic target in inflammatory disease. 了解更多 -
RG-12525
Catalog No. A19926 peptidoleukotrienes antagonistRG-12525 is a a specific, competitive and orally effective antagonist of the peptidoleukotrienes, LTC4, LTD4 and LTE4, inhibiting LTC4-, LTD4- and LTE4-inducd guinea pig parenchymal strips contractions, with IC50s of 2.6 nM, 2.5 nM and 7 nM, respectively; RG-12525 is also a peroxisome proliferator-activated receptor gamma (PPAR-gamma) agonist with IC50 of appr 60 nM and a potent inhibitor of CYP3A4, with a Ki value of 0.5 ?M. 了解更多 -
TR antagonist 1
Catalog No. A19919 TR antagonistTR antagonist 1 is a high-affinity thyroid hormone receptor (TR) antagonist with IC50s of 36 and 22 nM for TRα and TRβ, respectively. 了解更多 -
AHR antagonist 1
Catalog No. A19881 AHR antagonistAHR antagonist 1 is an aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2017202816A1, example 23, has an IC50 of 39.9 nM in human cell line. 了解更多 -
GSK3395879
Catalog No. A19861 TRPV4 antagonistGSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4. 了解更多 -
AZ10606120 dihydrochloride
Catalog No. A19853 P2X7R antagonistAZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10?nM. 了解更多 -
Broflanilide
Catalog No. A19824 Broflanilide is a potential insecticide and metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA receptor, and inhibits S. litura RDL GABAR, with an IC50 value of 1.3 nM. 了解更多 -
Foliglurax
Catalog No. A19753 mGluR4 modulatorFoliglurax (PXT002331) is a highly selective and potent, brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) with an EC50 of 79 nM. Antiparkinsonian effect. 了解更多 -
ORL1 antagonist 1
Catalog No. A19752 ORL1 antagonistORL1 antagonist 1 is an opioid receptor-like 1 (ORL1) antagonist with an IC50 of 61 nM. 了解更多 -
Estrone-N-O-C1-amido
Catalog No. A19746 estrogen ligandEstrone-N-O-C1-amido (ERα ligand 1) is an Estrone-based estrogen ligand, which targets estrogen receptor α (ERα). Estrone-N-O-C1-amido (ERα ligand 1) binds to cIAP1 ligand Bestatin via a linker to form SNIPER. 了解更多 -
Desisobutyryl-ciclesonide
Catalog No. A19718 Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide. Desisobutyryl-ciclesonide has affinity for the glucocorticoid receptor. 了解更多 -
DIM-C-pPhOCH3
Catalog No. A19708 Nur77 agonistDIM-C-pPhOCH3 is a Nur77 agonist. Nerve growth factor-induced Bα (NGFI-Bα, Nur77) is an orphan nuclear receptor. 了解更多 -
PROTAC ERα Degrader-2
Catalog No. A19697 ERα degraderPROTAC ERα Degrader-2 comprises a cIAP1 ligand binding group, a linker and an estrogen receptor α (ERα) binding group. PROTAC ERα Degrader-2 is an ERα degrader. 了解更多 -
Androstanolone acetate
Catalog No. A19688 androgen ligandAndrostanolone acetate is an androgen ligand, which targets androgen receptor (AR). Androstanolone acetate binds to cIAP1 ligand Bestatin via a linker to form PROTACs. 了解更多 -
PROTAC AR Degrader-4
Catalog No. A19678 AR degraderPROTAC AR Degrader-4 comprises a cIAP1 ligand binding group, a linker and an androgen receptor (AR) binding group. PROTAC AR Degrader-4 is an AR degrader. 了解更多 -
H4R antagonist 1
Catalog No. A19674 H4R antagonistH4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. 了解更多 -
PF-06747711
Catalog No. A19605 RORγt inverse agonistPF-06747711 is a potent, selective, and orally active retinoic acid receptor-related orphan C2 (RORC2, also known as RORγt) inverse agonist, with an IC50 of 4.1 nM. Anti-skin inflammatory activity. 了解更多 -
Proxalutamide
Catalog No. A19586 AR antagonistProxalutamide (GT0918) is a potent androgen receptor (AR) antagonist. 了解更多 -
N-Acetyl-5-hydroxytryptamine
Catalog No. A19581 Melatonin precursorN-Acetyl-5-hydroxytryptamine is a Melatonin precursor, and that it can potently activate TrkB receptor. 了解更多 -
IRAK4-IN-1
Catalog No. A19572 IRAK4 inhibitorIRAK4-IN-1 is an interleukin-1 receptor associated kinase 4 (IRAK4) inhibitor with an IC50 of 7 nM. 了解更多 -
2,2,5,7,8-Pentamethyl-6-Chromanol
Catalog No. A19565 2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol). 2,2,5,7,8-Pentamethyl-6-Chromanol has potent androgen receptor (AR) signaling modulation and anti-cancer activity against prostate cancer cell lines. 了解更多 -
GSK376501A
Catalog No. A19493 PPARγ modulatorGSK376501A is a selective peroxisome proliferator-activated receptor gamma (PPARγ) modulator for the treatment of type 2 diabetes mellitus. 了解更多
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