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VU 0238429
Catalog No. A21519 positive allosteric modulatorVU 0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5), with an EC50 of 1.16 μM. 了解更多 -
mAChR-IN-1
Catalog No. A21518 mAChR antagonistmAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM. 了解更多 -
RGX-104 free Acid
Catalog No. A21513 LXR agonistRGX-104 free Acid is an orally bioavailable and potent liver-X nuclear hormone receptor (LXR) agonist that modulates innate immunity via transcriptional activation of the ApoE gene. 了解更多 -
BMS-819881
Catalog No. A21500 MCHR1 antagonistBMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM. 了解更多 -
EC-17 disodium salt
Catalog No. A21492 FRα targeting contrast agentEC-17 (disodium salt) is a folate receptor alpha (FRα) targeting contrast agent with fluorescent properties in the visible light spectrum. 了解更多 -
PNU-282987 S enantiomer free base
Catalog No. A21459 PNU-282987 S enantiomer free base is the S-enantiomer of PNU-282987 free base. PNU-282987 is an α7 nicotinic acetylcholine receptor (α7 nAChR) agonist. 了解更多 -
mAChR-IN-1 hydrochloride
Catalog No. A21398 mAChR antagonistmAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM. 了解更多 -
TAS-115 mesylate
Catalog No. A21389 c-Met/HGFR inhibitorTAS-115 mesylate is a potent VEGFRand hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase inhibitor, with IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively. 了解更多 -
PF-00446687
Catalog No. A21382 MC4R agonistPF-00446687 is a potent, selective melanocortin-4 receptor (MC4R) agonist with EC50 of 12????1 nM. Pf-446687 is brain penetrant. 了解更多 -
FTY720 (S)-Phosphate
Catalog No. A21324 S1PR1 agonistFTY720 (S)-Phosphate is an agonist of S1P receptor 1 (S1PR1), used in the research of acute inflammatory diseases such as acute lung injury. 了解更多 -
LPA1 antagonist 1
Catalog No. A21301 LPA1 antagonistLPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM. 了解更多 -
Fedovapagon
Catalog No. A21286 V2R agonistFedovapagon is a selective vasopressin V2 receptor (V2R) agonist with an EC50 of 24 nM, which is being developed for the treatment of nocturia. 了解更多 -
Capromorelin Tartrate
Catalog No. A21238 GHSR agonistCapromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. 了解更多 -
OT-R antagonist 1
Catalog No. A21216 OT-R antagonistOT-R antagonist 1 is a new potent and selective nonpeptide low molecular weight OT-R antagonist. 了解更多 -
(R)-Elagolix
Catalog No. A21184 GnRHR antagonistElagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多 -
Pavinetant
Catalog No. A21174 NK3R antagonistPavinetant (MLE-4901) is a neurokinin-3 receptor (NK3R) antagonist. 了解更多 -
Methionine
Catalog No. A21171 chemoprotective agentMethionine (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor activation. 了解更多 -
Indeglitazar
Catalog No. A21148 PPAR agonistIndeglitazar is an orally available peroxisome proliferator-activated receptor (PPAR) pan-agonist for all three PPAR subtypes alpha (α), delta (δ) and gamma (γ). 了解更多 -
Arhalofenate
Catalog No. A21135 PPARγ agonistArhalofenate (MBX 102) is a selective partial agonist of peroxisome proliferator-activated receptor (PPAR)-γ, used for the treatment of type 2 diabetes. 了解更多 -
Evatanepag
Catalog No. A21129 PGE2 agonistEvatanepag (CP-533536) is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation with EC50 of 0.3 nM. 了解更多 -
Rapacuronium bromide
Catalog No. A21119 mAChR modulatorRapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR). 了解更多 -
Indirubin Derivative E804
Catalog No. A21052 IGF1R inhibitorE 804 is a potent inhibitor of Insulin-like Growth Factor 1 Receptor (IGF1R), with an IC50 of 0.65 μM for IGF1R. 了解更多 -
Tesaglitazar
Catalog No. A20891 PPAR alpha/gamma agonistTesaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha/gamma agonist that is more potent on PPARγ than on PPARα, with EC50s of 13.4 μM and 3.6 μM for rat PPARα and human PPARα, respectively. 了解更多 -
Levalbuterol tartrate
Catalog No. A20864 Levosalbutamol tartrate(levalbuterol) is the R-enantiomer of the short-acting β2-adrenergic receptor agonist salbutamol. 了解更多 -
Eltoprazine
Catalog No. A20861 Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor. 了解更多 -
Metixene hydrochloride hydrate
Catalog No. A18028 anticholinergic antiparkinsonian agentMetixene hydrochloride hydrate is an anticholinergic antiparkinsonian agent, potently inhibits binding of quinuclidinyl benzilate (QNB) to the muscarinic receptor in rat brain cortical tissue, with an IC50 of 55 nM and a Kd of 15 nM. 了解更多 -
Alimemazine hemitartrate
Catalog No. A17754 antipruritic agentAlimemazine hemitartrate is a phenothiazine derivative that is generally used as an antipruritic agent and also a hemagglutinin (HA)-receptor antagonist. 了解更多 -
Resatorvid
Catalog No. A11543 TLR4 inhibitorResatorvid (TAK-242) is a selective Toll-like receptor 4 (TLR4) inhibitor and plays pivotal role in various inflammatory diseases. 了解更多 -
Pitolisant
Catalog No. A11525 nonimidazole inverse agonistPitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). 了解更多 -
NPS-2143 hydrochloride
Catalog No. A11505 CaSR antagonistNPS-2143 hydrochloride (SB-262470A hydrochloride), an orally active calcilytic agent, is a selective and potent calcium ion-sensing receptor (CaSR) antagonist. 了解更多 -
IRAK inhibitor 4
Catalog No. A11458 IRAK4 inhibitorIRAK inhibitor 4 is an interleukin-1 receptor associated kinase 4(IRAK4) inhibitor. 了解更多 -
Kynurenic acid sodium
Catalog No. A20000 GPR35/CXCR8 agonistKynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多 -
MT-7716 hydrochloride
Catalog No. A20004 NOP agonistMT-7716 hydrochloride (W-212393 hydrochloride) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. 了解更多 -
EGFR-IN-3
Catalog No. A15847 -
Propyl pyrazole triol
Catalog No. A13329 ERα agonistPropyl pyrazole triol (PPT) is an estrogen receptor alpha (ERα) agonist. 了解更多
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