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CGP71683 hydrochloride
Catalog No. A19844 neuropeptide Y5 receptor antagonistCGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes. 了解更多 -
CJ-42794
Catalog No. A21948 EP4 antagonistCJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多 -
Risperidone hydrochloride
Catalog No. A21458 dopamine D2 receptor antagonistRisperidone hydrochloride is a serotonin 5-HT2 receptor blocker and a potent dopamine D2 receptor antagonist, with Kis of 0.16, 1.4 nM for 5-HT2 and D2 receptor, respectively. 了解更多 -
L-371,257
Catalog No. A21219 oxytocin receptor antagonistL-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM). 了解更多 -
Cutamesine
Catalog No. A21152 sigma 1 receptor agonistCutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多 -
Pipamperone
Catalog No. A12621 D2 receptor antagonistPipamperone (Floropipamide; McN-JR 3345; R 3345) is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7). 了解更多 -
Nemorexant
Catalog No. A12685 Orexin receptor antagonistNemorexant (ACT-541468) is a potent orexin receptor antagonist extracted from patent WO2015083094A1, compound example 7, has IC50s of 2 nM and 3 nM for Ox1 receptor and Ox2 receptor, respectively. 了解更多 -
JNJ-54175446
Catalog No. A18675 P2X7 receptor antagonistJNJ-54175446 is a potent and selective brain penetrant P2X7 receptor antagonist, with pIC50s of 8.46 and 8.81 for hP2X7 receptor and rP2X7 receptor, respectively. 了解更多 -
Seratrodast
Catalog No. A18134 thromboxane A2 (TXA2) receptor (TP receptor) antagonistSeratrodast is a thromboxane A2 (TXA2) receptor (TP receptor) antagonist used primarily in the treatment of asthma. 了解更多 -
SCH-23390 maleate
Catalog No. A22592 dopamine D1-like receptor antagonistSCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively. 了解更多 -
Aganepag
Catalog No. A20794 Prostanoid EP2 receptor agonistAganepag is a potent Prostanoid EP2 receptor agonist, with an EC50 of 0.19 nM, and shows no activity at EP4 receptor. Aganepag can be used in the research of wound healing, scar reduction, scar prevention and wrinkle treatment and prevention. 了解更多 -
Masupirdine free base
Catalog No. A20245 5-HT6 receptor antagonistMasupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多 -
Sigma-LIGAND-1
Catalog No. A20242 Sigma-LIGAND-1 is a selective sigma receptor ligand, has receptor IC50s of 16 nM at the DTG site, 19 nM at the PPP site, and a Ki of 4000 nM at the dopamine D2 receptor. 了解更多 -
5-HT7 agonist 1
Catalog No. A20143 5-HT7 receptor agonist5-HT7 agonist 1 is a selective 5-HT7 receptor agonist, with an IC50 of 222.93 nM, can be used for the 5-HT7 receptor related disease, such as CNS disorders. 了解更多 -
ZD 7155 hydrochloride
Catalog No. A19959 AT1 receptor antagonistZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist. 了解更多 -
L-368,899 hydrochloride
Catalog No. A19843 oxytocin receptor antagonistL-368,899 hydrochloride is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively, used as a tocolytic agent. 了解更多 -
ReN-1869 hydrochloride
Catalog No. A19610 histamine H1 receptor antagonistReN 1869 hydrochloride is a novel, selective histamine H1 receptor antagonist, which demonstrates affinity to the histamine H1 receptor (guinea pig brain) with Ki of 0.19±0.04 μM and the non-selective ?? site (guinea pig brain) with Ki of 0.45 μM. 了解更多 -
J-2156
Catalog No. A19264 SST4 receptor agonistJ-2156 is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. 了解更多 -
Nomegestrol
Catalog No. A19235 full progesterone receptor agonistNomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity. 了解更多 -
![N-[(4-Aminophenyl)methyl]adenosine](https://www.adooq.cn/media/catalog/product/cache/1/small_image/9df78eab33525d08d6e5fb8d27136e95/a/1/a12659-n-4-aminophenyl-methyl-adenosine_1.gif)
N-[(4-Aminophenyl)methyl]adenosine
Catalog No. A12659 Adenosine receptor inhibitorN-[(4-Aminophenyl)methyl]adenosine is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5??-Nucleotidase. IC50 value: 29.0 ± 1.7 nM (Ki) Target: Adenosine Receptor 了解更多 -
Cariprazine
Catalog No. A21202 D3 receptor and D2 receptor partial agonistCariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). 了解更多 -
Dihydrexidine
Catalog No. A21949 D1-like dopamine receptor (D1/D5) agonistDihydrexidine (DAR-0100) is a high potent, selective and full efficacy D1-like dopamine receptor (D1/D5) agonist with an IC50 of 10 nM for D1 receptor. Dihydrexidine exhibits potent antiparkinsonian activity. 了解更多 -
AZD9496 maleate
Catalog No. A21726 estrogen receptor (ERα) antagonistAZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多 -
Tarafenacin D-tartrate
Catalog No. A21477 M3 muscarinic receptor antagonistTarafenacin D-tartrate (SVT-40776 D-tartrate) is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor. 了解更多 -
JNJ-37822681 dihydrochloride
Catalog No. A21470 dopamine D2 receptor antagonistJNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多 -
Risperidone mesylate
Catalog No. A21463 dopamine D2 receptor antagonistRisperidone mesylate(R 64 766 mesylate) is a serotonin 5-HT2 receptor blocker(Ki= 0.16 nM) and a potent dopamine D2 receptor antagonist(Ki= 1.4 nM). 了解更多 -
Masupirdine mesylate
Catalog No. A21409 5-HT6 receptor antagonistMasupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). 了解更多 -
Ditolylguanidine
Catalog No. A21268 Sigma receptor agonistDitolylguanidine (1,3-Di-o-tolylguanidine) is an agonist of sigma receptor (??1/??2 receptor). 了解更多 -
Zonampanel
Catalog No. A21199 glutamate receptor subtype antagonistZonampanel (YM 872) is a selective antagonist of the glutamate receptor subtype, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) receptor. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
Pexacerfont
Catalog No. A14105 CRF1 receptor antagonistPexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多 -
LY-2940094
Catalog No. A19125 NOP receptor antagonistLY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models. 了解更多 -
Fimasartan
Catalog No. A17477 non-peptide angiotensin II receptor antagonistFimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多
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