“alpha ergocryptine”的搜索结果

产品 201 到 250 共 642个

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  1. Basmisanil

    Catalog No. A21321
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    GABAAα5 modulator
    Basmisanil is a highly selective GABAAα5 negative allosteric modulator. 了解更多
  2. ATN-161

    Catalog No. A21307
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    integrin α5β1 antagonist
    ATN-161 is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. 了解更多
  3. R1487 Hydrochloride

    Catalog No. A21231
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    p38α inhibitors
    R1487 (Hydrochloride) is highly potent and highly selective inhibitors of p38α. 了解更多
  4. MK-0429

    Catalog No. A21173
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    αvβ3 integrin antagonist
    MK-0429 (L-000845704) is an orally active, potent, selective and nonpeptide αvβ3 integrin antagonist with an IC50 of 80 nM. 了解更多
  5. Indeglitazar

    Catalog No. A21148
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    PPAR agonist
    Indeglitazar is an orally available peroxisome proliferator-activated receptor (PPAR) pan-agonist for all three PPAR subtypes alpha (α), delta (δ) and gamma (γ). 了解更多
  6. Alfacalcidol-D6

    Catalog No. A21142
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    VDR activator
    Alfacalcidol-D6, a deuterated Alfacalcidol (1-hydroxycholecalciferol; Alpha D3; 1.alpha.-Hydroxyvitamin D3), is a non-selective VDR activator medication. 了解更多
  7. EL-102

    Catalog No. A20925
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    HIF1α inhibitor
    EL102 is a inhibitor of HIF1α , Which can inhibit tubulin polymerisation and decreased microtubule stability. 了解更多
  8. Emiglitate

    Catalog No. A20917
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    α-glucoside hydrolase inhibitor
    Emiglitate (BAY o 1248) is a potent, selective and competitive inhibitor of α-glucoside hydrolase. 了解更多
  9. Integrin Antagonists 27

    Catalog No. A20895
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    integrin αvβ3 antagonist
    Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist with binding affinity of 18 nM, as s novel anticancer agent. 了解更多
  10. Oxytocin

    Catalog No. A17988
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    oxytocin receptor ligand
    Oxytocin (α-Hypophamine) is a mammalian neurohypophysial hormone; its actions are mediated by specific, high-affinity oxytocin receptors; ligand of oxytocin receptor. 了解更多
  11. Darbufelone mesylate

    Catalog No. A11789
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    PGF2α/LTB4 production inhibitor
    Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF2α and LTB4 production. Darbufelone potently inhibits PGHS-2 (IC50 = 0.19 μM) but is much less potent with PGHS-1 (IC50= 20 μM). 了解更多
  12. Rivanicline oxalate

    Catalog No. A11544
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    neuronal nicotinic receptor agonist
    Rivanicline oxalate (RJR-2403 oxalate; (E)-Metanicotine oxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 3.6 μM). 了解更多
  13. β3-AR agonist 1

    Catalog No. A12777
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    β3-adrenergic receptor agonist
    β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多
  14. MKC3946

    Catalog No. A12508
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    IRE1α inhibitor
    MKC3946 is a potent and soluble IRE1α inhibitor, used for cancer research. 了解更多
  15. KIRA6

    Catalog No. A12516
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    IRE1α RNase kinase inhibitor
    KIRA6 is an advanced small-molecule IRE1α RNase kinase inhibitor with an IC50 of 0.6 ?M. KIRA6 can trigger an apoptotic response. 了解更多
  16. Ercalcitriol

    Catalog No. A11414
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    Ercalcitriol (1α,25-Dihydroxy Vitamin D2) is an active metabolite of vitamin D2. 了解更多
  17. ZINC13466751

    Catalog No. A12522
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    HIF-1α/von Hippel-Lindau interaction inhibitor
    ZINC13466751 is a potent inhibitor of HIF-1α/von Hippel-Lindau interaction with an IC50 of 2.0 ?M. 了解更多
  18. STF-083010

    Catalog No. A16720
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    IRE1α inhibitor
    STF-083010 is a specific IRE1α inhibitor. STF-083010 inhibits Ire1 endonuclease activity, without affecting its kinase activity, after endoplasmic reticulum stress. 了解更多
  19. C 87

    Catalog No. A12313
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    TNFα inhibitor
    C87 is a novel small-molecule TNFα inhibitor; potently inhibits TNFα-induced cytotoxicity with an IC50 of 8.73 μM. 了解更多
  20. PAC

    Catalog No. A12939
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    PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab). 了解更多
  21. MD2-TLR4-IN-1

    Catalog No. A18452
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    MD2-TLR4 inhibitor
    MD2-TLR4-IN-1 (compound 22m) is an inhibitor of myeloid differentiation protein 2/toll-like receptor 4 (MD2-TLR4) complex, inhibiting lipopolysaccharides (LPS)-induced expression of tumor necrosis factor alpha (TNF-α) and interleukin-6 (IL-6) in macrophages with IC50 values of 0.89 μM and 0.53 μM, respectively. 了解更多
  22. PROTAC ER Degrader-3

    Catalog No. A18519
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    PROTAC ER Degrader-3 is an intermediate for synthesis of PAC. PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab). 了解更多
  23. 3,5-Diiodothyropropionic acid

    Catalog No. A19117
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    3,5-Diiodothyropropionic acid is a thyroid hormone analog, induces α-myosin heavy chain mRNA expression, binds to thyroid hormone receptor (TR), with Ka of 2.40 and 4.06 M-1 for TRα1 and TRβ1, respectively. 了解更多
  24. INH14

    Catalog No. A19119
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    IKKα/IKKβ inhibitor
    INH14 is a cell permeable inhibitor of IKKα/IKKβ, with IC50s of 8.97 and 3.59 μM, respectively. 了解更多
  25. GSK5182

    Catalog No. A19383
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    ERRγ agonist
    GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. 了解更多
  26. LJ570

    Catalog No. A20081
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    PPARα/PPARγ dual agonist
    LJ570 is a PPARα/PPARγ dual agonist with EC50s of 1.05 and 0.12 μM, respectively. 了解更多
  27. Pictilisib dimethanesulfonate

    Catalog No. A11444
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    PI3Kα/δ inhibitor
    Pictilisib dimethanesulfonate (GDC-0941 dimethanesulfonate) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM, with modest selectivity against p110β (11-fold) and p110γ (25-fold). 了解更多
  28. 6-Thioinosine

    Catalog No. A18412
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    6-?Thioinosine (6TI) is a purine antimetabolite, acts as an anti-adipogenesis agent, downregulates mRNA levels of PPAR γ and C/EBPα, as well as PPAR γ target protein such as LPL, CD36, aP2, and LXRα. 了解更多
  29. BNC375

    Catalog No. A18503
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    α7 nAChR Modulator
    BNC375 is a Potent, Selective, and Orally Available Type I Positive Allosteric Modulator of α7 nAChRs. 了解更多
  30. VERU-111

    Catalog No. A18743
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    oral α and β tubulin inhibitor
    VERU-111 is a novel, oral α and β tubulin inhibitor that blocks tubulin polymerization and is not a substrate for multi-drug resistance mechanisms. 了解更多
  31. (-)-(S)-B-973B

    Catalog No. A18761
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    α7 nAChR modulator
    -)-(S)-B-973B is a potent allosteric agonist and positive allosteric modulator of α7 nAChR, with antinociceptive activity. 了解更多
  32. MW-150

    Catalog No. A18798
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    p38α MAPK inhibitor
    MW150 (MW01-18-150SRM) is a selective, CNS penetrant, and orally active inhibitor of p38α MAPK with a Ki of 101 nM. 了解更多
  33. Epristeride

    Catalog No. A18231
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    5 alpha-reductase inhibitor
    Epristeride is a selective and specific uncompetitive inhibitor of human steroid 5 alpha-reductase isoform 2. 了解更多
  34. Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多
  35. Lofexidine

    Catalog No. A18151
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    α2-receptor agonist
    Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. 了解更多
  36. Limaprost

    Catalog No. A18129
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    platelet adhesion inhibitor
    Limaprost(OP1206) is a PGE1 analog and potent platelet adhesion inhibitor. 了解更多
  37. Midodrine

    Catalog No. A17758
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    adrenergic alpha-1 agonist
    Midodrine is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of HYPOTENSION. 了解更多
  38. Midodrine hydrochloride

    Catalog No. A17757
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    Adrenergic alpha-1 agonist
    Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多
  39. Moxisylyte hydrochloride

    Catalog No. A17725
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    alpha-adrenergic blocking agent
    Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomimetic agents. 了解更多
  40. Methoxamine HCl

    Catalog No. A17365
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    alpha-1 adrenergic agonist
    Methoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction. 了解更多
  41. Lobeline hydrochloride

    Catalog No. A17333
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    nicotinic receptor agonist
    Lobeline hydrochloride, a nicotinic receptor agonist, acting as a potent antagonist at both α3β2 and α4β2 neuronal nicotinic receptor subtypes. 了解更多
  42. Xylometazoline HCl

    Catalog No. A17251
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    α-adrenoceptor agonist
    Xylometazoline hydrochloride is an α-adrenoceptor agonist commonly used as nasal decongestant. 了解更多
  43. Piperoxan hydrochloride

    Catalog No. A18336
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    α2 adrenoceptor antagonist
    Piperoxan hydrochloride is an α2 adrenoceptor antagonist. 了解更多
  44. R-BC154

    Catalog No. A17184
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    α4β1/α9β1 抑制剂
    R-BC154是高亲和力的荧光α4β1/α9 9β1抑制剂。 了解更多
  45. BOP sodium salt

    Catalog No. A17201
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    α9β1/α4β1 integrin 抑制剂
    BOP sodium salt是新型的双重alpha9beta1/alpha4beta1整联蛋白抑制剂。 了解更多
  46. Lipoic acid

    Catalog No. A14822
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    Lipoic acid是衍生自辛酸的有机硫化合物。ALA通常在动物体内制成,并且对于有氧代谢至关重要。 了解更多
  47. Deoxygalactonojirimycin HCl

    Catalog No. A14016
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    Alpha-galactosidase 抑制剂
    Deoxygalactonojirimycin Hydrochloride是一种有效且选择性的Alpha-gal A(Alpha-半乳糖苷酶)抑制剂。 了解更多
  48. Tamsulosin

    Catalog No. A12657
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    alpha-1A/alpha-1B-adrenoceptor 拮抗剂
    Tamsulosin是一种α1a-选择性α受体阻滞剂,用于对症治疗前列腺增生(BPH)。 了解更多
  49. Hyodeoxycholic acid

    Catalog No. A10460
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    Hyodeoxycholic (HDCA) acid是二级胆汁酸,是肠道细菌的代谢副产物之一。 了解更多
  50. BMS453

    Catalog No. A22082
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    RARβ agonist
    BMS453 (BMS-189453), a synthetic retinoid, is a RARβ agonist and a RARα/RARγ antagonist. 了解更多

产品 201 到 250 共 642个

每页
页面:
  1. 3
  2. 4
  3. 5
  4. 6
  5. 7

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