“glucagon receptor”的搜索结果

产品 301 到 350 共 1712个

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  1. L-159282

    Catalog No. A20703
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    nonpeptide angiotensin II receptor antagonist
    L-159282 is a highly potent, orally active, nonpeptide angiotensin II receptor antagonist, with anti-hypertensive activity. 了解更多
  2. CP-105696

    Catalog No. A20701
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    Leukotriene B4 Receptor antagonist
    CP-105696 is a potent and selective Leukotriene B4 Receptor antagonist, with an IC50 of 8.42 nM. 了解更多
  3. gamma-DGG

    Catalog No. A20685
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    AMPA receptor blocker
    gamma-DGG is a competitive AMPA receptor blocker. 了解更多
  4. AZD-6280

    Catalog No. A20684
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    GABAA(α2/3) receptor modulator
    AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. 了解更多
  5. Sultopride

    Catalog No. A20663
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    dopamine D2 receptor antagonist
    Sultopride (LIN-1418) is a selective antagonist of dopamine D2 receptor. 了解更多
  6. JNJ-18038683

    Catalog No. A20659
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    5-HT7 receptor antagonist
    JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively. 了解更多
  7. GSK1521498

    Catalog No. A20649
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    μ-opioid receptor (MOR) antagonist
    GSK1521498 is a potent and selective μ-opioid receptor (MOR) antagonist. GSK1521498 is being used for the treatment of disorders of compulsive consumption of food, alcohol, and drugs. 了解更多
  8. Taprenepag isopropyl

    Catalog No. A20604
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    EP2 receptor agonist
    Taprenepag isopropyl is a highly selective EP2 receptor agonist. 了解更多
  9. Sufugolix

    Catalog No. A20589
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    LHRH receptor antagonist
    Sufugolix (TAK-013) is a highly potent and orally available luteinizing hormone-releasing hormone (LHRH) receptor antagonist with an IC50 of 0.1 nM. 了解更多
  10. PZM21

    Catalog No. A20586
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    μ opioid receptor agonist
    PZM21 is a potent and selective μ opioid receptor agonist with an EC50 of 1.8 nM. 了解更多
  11. Quinolinic acid

    Catalog No. A20575
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    NMDA receptor agonist
    Quinolinic acid is an endogenous N-methyl-D-aspartate (NMDA) receptor agonist synthesized from L-tryptophan via the kynurenine pathway and thereby has the potential of mediating N-methyl-D-aspartate neuronal damage and dysfunction. 了解更多
  12. Isoguvacine hydrochloride

    Catalog No. A20563
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    GABA receptor agonist
    Isoguvacine hydrochloride is a GABA receptor agonist. 了解更多
  13. JNJ16259685

    Catalog No. A20545
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    mGlu1 receptor antagonist
    JNJ16259685 is a selective antagonist of mGlu1 receptor, and inhibits the synaptic activation of mGlu1 in a concentration-dependent manner with IC50 of 19 nM. 了解更多
  14. Naltrindole hydrochloride

    Catalog No. A20541
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    δ opioid receptor antagonist
    Naltrindole hydrochloride is a highly potent and selective non-peptide δ opioid receptor antagonist with a Ki of 0.02 nM. 了解更多
  15. Nicotinamide N-oxide

    Catalog No. A20532
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    CXCR2 receptor antagonist
    Nicotinamide N-oxide, an in vivo nicotinamide metabolite, is a potent, and selective antagonist of the CXCR2 receptor. 了解更多
  16. Org-26576

    Catalog No. A20502
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    AMPA receptor modulator
    Org-26576 is a AMPA receptor positive allosteric modulator. 了解更多
  17. PCO371

    Catalog No. A20493
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    PTHR1 agonist
    PCO371 is an orally active full agonist of parathyroid hormone receptor 1 (PTHR1), with no effect on PTH type 2 receptor. 了解更多
  18. CYM-5541

    Catalog No. A20489
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    S1P3 receptor agonist
    CYM-5541 (ML249) is an selective and allosteric S1P3 receptor agonist with an EC50 between 72 and 132 nM. 了解更多
  19. Sarmazenil

    Catalog No. A20487
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    benzodiazepine receptor antagonist
    Sarmazenil is a benzodiazepine receptor antagonist. 了解更多
  20. Tiodazosin

    Catalog No. A20463
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    ostsynaptic alpha adrenergic receptor antagonist
    Tiodazosin is a potent competitive postsynaptic alpha adrenergic receptor antagonist. 了解更多
  21. Org41841

    Catalog No. A20396
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    LHCGR/TSHR agonist
    Org41841 is a partial agonist of both luteinizing hormone/chorionic gonadotropin receptor (LHCGR) and thyroid-stimulating hormone receptor (TSHR) with EC50s of 0.2 and 7.7 μM, respectively. 了解更多
  22. Pirolate

    Catalog No. A20363
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    histamine H1 receptor
    Pirolate is a histamine H1 receptor. 了解更多
  23. JYL 1421

    Catalog No. A20350
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    TRPV1 receptor antagonist
    JYL 1421 is a TRPV1 receptor antagonist, with an IC50 of 8 nM. 了解更多
  24. (+)-Dihydrexidine hydrochloride

    Catalog No. A20339
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    dopamine D1 receptor agonist
    (+)-Dihydrexidine hydrochloride ((+)-DAR-0100 hydrochloride) is a dopamine D1 receptor agonist with an EC50 of 72± 21 nM. 了解更多
  25. L162389

    Catalog No. A20297
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    angiotensin AT1 receptor antagonist
    L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM. 了解更多
  26. Abaperidone

    Catalog No. A20286
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    5-HT2A/dopamine D2 antagonist
    Abaperidone is a potent antagonist of 5-HT2A?receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM. 了解更多
  27. MRZ 2-514

    Catalog No. A20277
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    NMDA receptor (glycineB) antagonist
    MRZ 2-514 is an antagonist of the strychnine-insensitive modulatory site of the NMDA receptor (glycineB), with Ki of 33 μM. 了解更多
  28. Lidanserin

    Catalog No. A20266
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    5-HT2A/α1-adrenergic receptor antagonist
    Lidanserin is a drug which acts as a combined 5-HT2A and α1-adrenergic receptor antagonist. 了解更多
  29. Spirendolol

    Catalog No. A20254
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    β adrenergic receptor antagonist
    Spirendolol is a β adrenergic receptor antagonist. 了解更多
  30. Foscarbidopa

    Catalog No. A20221
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    dopamine receptor agonist
    Foscarbidopa (Carbidopa 4??-monophosphate) is a prodrug of Carbidopa, acts as a dopamine receptor agonist. 了解更多
  31. Foslevodopa

    Catalog No. A20212
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    dopamine receptor agonist
    Foslevodopa is a dopamine receptor agonist. 了解更多
  32. ALB-127158(a)

    Catalog No. A20211
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    MCH1 receptor antagonist
    ALB-127158(a) is a potent and selective melanin concentrating hormone 1 (MCH1) receptor antagonist. 了解更多
  33. NK-1 Antagonist 1

    Catalog No. A20201
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    NK-1 receptor antagonist
    NK-1 Antagonist 1 (Rolapitant intermediate) is an antagonist of NK-1 receptor, used in the research of NK-1 related diseases and conditions such as cough, overactive bladder, alcohol dependency and depression. 了解更多
  34. Taminadenant

    Catalog No. A20190
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    adenosine receptor antagonist
    Taminadenant is an antagonist of adenosine receptor. 了解更多
  35. Wy 49051

    Catalog No. A20176
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    H1 receptor antagonist
    Wy 49051 is a potent, orally active H1 receptor antagonist, with IC50 of 44 nM. 了解更多
  36. FK1052 hydrochloride

    Catalog No. A20164
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    5-HT3 /5-HT4 receptor dual antagonist
    FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist. 了解更多
  37. Saredutant

    Catalog No. A20096
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    NK2 receptor antagonist
    Saredutant is a selective NK2 receptor antagonist. 了解更多
  38. Apimostinel

    Catalog No. A20075
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    NMDA receptor partial agonist
    Apimostinel (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist. 了解更多
  39. AR-A 2

    Catalog No. A20051
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    5-HT1B receptor antagonist
    AR-A 2 is a selective 5-HT1B receptor antagonist. 了解更多
  40. FITM

    Catalog No. A20047
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    mGlu1 receptor modulator
    FITM is a negative allosteric modulator of mGlu1 receptor with a Ki of 2.5 nM. 了解更多
  41. AP5

    Catalog No. A20042
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    AP5 exhibits potent and selective agonism for the GPR40 receptor with positive allosteric modulation of endogenous ligands (AgoPAM). AP5 demonstrates a rat hIP1 EC50 of 0.49±0.28 nM against the GPR40 receptor. 了解更多
  42. Pargolol hydrochloride

    Catalog No. A20035
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    β adrenergic receptor antagonist
    Pargolol hydrochloride is a β adrenergic receptor antagonist. 了解更多
  43. YK11

    Catalog No. A20033
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    Androgen receptor partial agonist
    YK11 is a partial agonist of androgen receptor, with osteogenic activity. 了解更多
  44. MK-8318

    Catalog No. A20030
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    CRTh2 receptor antagonist
    MK-8318 is a potent and selective CRTh2 receptor antagonist with a Ki of 5.0 nM. 了解更多
  45. ODM-204

    Catalog No. A20025
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    androgen receptor/CYP17A1 dual inhibitor
    ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme, with IC50s of 80?nM and 22 nM, respectively. 了解更多
  46. N6-(2-Phenylethyl)adenosine

    Catalog No. A20011
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    A1 adenosine receptor agonist
    N6-(2-Phenylethyl)adenosine is a selective A1 adenosine receptor agonist. 了解更多
  47. D4-abiraterone

    Catalog No. A19987
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    androgen receptor antagonist
    D4-abiraterone is a major metabolite of abiraterone. D4-abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid-5a-reductase (SRD5A) and also an antagonist of androgen receptor. 了解更多
  48. Sulamserod

    Catalog No. A19984
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    5-HT4 receptor antagonist
    Sulamserod is a 5-HT4 receptor antagonist, with antiarrhythmic activities. 了解更多
  49. H3B-5942

    Catalog No. A19960
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    estrogen receptor covalent antagonist
    H3B-5942 is a selective, irreversible and orally active estrogen receptor covalent antagonist, inactivates both wild-type and mutant ERα by targeting Cys530, with Kis of 1 nM and 0.41 nM, respectively. 了解更多
  50. 1,4-Chrysenequinone

    Catalog No. A19937
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    aryl hydrocarbon receptor activator
    1,4-Chrysenequinone, a polycyclic aromatic quinone, acts as an activator of aryl hydrocarbon receptor (AhR). 了解更多

产品 301 到 350 共 1712个

每页
页面:
  1. 5
  2. 6
  3. 7
  4. 8
  5. 9

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